GENTILI, Francesco

GENTILI, Francesco  

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14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry 1-gen-2003 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma ORGANIZZAZIONE DI EVENTI
16th Camerino-Noordwijkerhout Symposium - An Overview of Receptor Chemistry 1-gen-2007 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma ORGANIZZAZIONE DI EVENTI
2-(2-Phenylcyclopropyl)imidazolines: Reversed Enantioselective Interaction at I1 and I2 Imidazoline Receptors 1-gen-1999 Quaglia, Wilma; Bousquet, P.; Pigini, Maria; Carotti, A.; Carrieri, A.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Maranca, F.; Piergentili, Alessandro; Brasili, L. Articolo
Agonists and antagonists targeting the different alpha(2)-adrenoceptor subtypes 1-gen-2007 Gentili, Francesco; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario Articolo
Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole 1-gen-2002 Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria Articolo
alpha(2)-Adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha2C-subtype 1-gen-2004 Gentili, Francesco; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Vesprini, C.; Crassous, A.; Paris, H.; Carrieri, A. Articolo
Alpha(2)-Adrenoreceptors Profile Modulation. 3. (R)-(+)-m-Nitrobiphenyline, a New Efficient and alpha(2C)-Subtype Selective Agonist. 1-gen-2007 Crassous, P. A.; Cardinaletti, C; Carrieri, A; Bruni, B; DI VAIRA, M; Gentili, Francesco; Ghelfi, F; Giannella, Mario; Paris, H; Piergentili, Alessandro; Quaglia, Wilma; Schaak, S; Vesprini, C; Pigini, Maria Articolo
alpha(2)-adrenoreceptors profile modulation. 4. From antagonist, to agonist behavior 1-gen-2008 Gentili, Francesco; Cardinaletti, C.; Vesprini, C.; Carrieri, A.; Ghelfi, F.; Farande, A.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Laurila, J. M.; Huhtinen, A.; Scheinin, M.; Pigini, Maria Articolo
Binding of Tracizolines to the Imidazoline Receptor. Role of Lipophilicity in Quantitative Structure-Activity Relationship Models. 1-gen-1999 Pigini, Maria; Bousquet, P; Brasili, L; Carrieri, A; Dontenwill, M; Gentili, Francesco; Giannella, Mario; Leonetti, F; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A. Articolo
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives 1-gen-2002 Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma Articolo
Hyperphagic effect of novel compounds with high affinity for imidazoline I2 binding sites 1-gen-2000 Polidori, Carlo; Gentili, Francesco; Pigini, Maria; Quaglia, Wilma; Panocka, I.; Massi, M. Articolo
Imidazoline binding sites (IBS) profile modulation: Key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues 1-gen-2003 Gentili, Francesco; Bousquet, P.; Brasili, L.; Dontenwill, M.; Feldman, J.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria Articolo
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models 1-gen-1998 Pigini, Maria; Bousquet, P.; Brasili, L.; Carrieri, A.; Cavagna, R.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Leonetti, F.; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A. Articolo
Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine 1-gen-2003 Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario Articolo
Novel ligands rationally designed for characterizing I2-imidazoline binding sites nature and functions 1-gen-2008 Gentili, Francesco; Cardinaletti, Claudia; Vesprini, C.; Ghelfi, Francesca; Farande, ANIKET VIJAYKUMAR; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Mattioli, Laura; Perfumi, Marina Cecilia; Hudson, A.; Pigini, Maria Articolo
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands 1-gen-2004 Nicolotti, O.; Carotti, A.; Carrieri, A.; Pigini, Maria; Gentili, Francesco; Brasili, L.; Giannella, Mario; Quaglia, Wilma; Piergentili, Alessandro; Bousquet, P.; Dontenwill, M. Articolo
Rational design of new alpha(2)-adrenoreceptor agonists 1-gen-2007 Gentili, Francesco; Cardinaletti, C.; Carrieri, A.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, Maria Articolo
Solution-phase synthesis of ICG-001, a beta-turn peptidomimetic molecule inhibitor of beta-catenin-Tcf-mediated transcription 1-gen-2007 Piergentili, Alessandro; DEL BELLO, Fabio; Gentili, Francesco; Giannella, Mario; Quaglia, Wilma; Vesprini, Christian; Thomas, R. J.; Robertson, G. M. Articolo
Structure-activity relationship at alpha-adrenergic receptors within a series of imidazoline analogues of cirazoline 1-gen-2000 Pigini, Maria; Quaglia, Wilma; Gentili, Francesco; Marucci, Gabriella; Cantalamessa, F.; Franchini, S.; Sorbi, C.; Brasili, L. Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes 1-gen-2002 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C. Articolo