Sfoglia per Autore
“Tetraamines as Lead Compounds for the “Pharmacological Evaluation of Prazosin and Doxazosin-related Compounds with Modified Piperazine Ring”.
1996-01-01 Giardinà, D; Crucianelli, M; Marucci, Gabriella; Melchiorre, C; Polidori, Carlo; Pompei, Pierluigi; Massi, Maurizio
SAR Studies on the Potent and Selective Muscarinic Antagonist 2-Ethylthio-2,2-diphenylacetic Acid N,N-Diethylaminoethyl Ester
1997-01-01 Scapecchi, S; Angeli, Piero; Dei, S; Ghelardini, C; Gualtieri, F; Marucci, Gabriella; Paparelli, F; Romanelli, M. N.; Teodori, E.
“Synthesis and α1-Antagonist Activity of New Prazosin-and Benextramine-Related Tetraamine Disulfides”.
1997-01-01 Giardinà, D; Crucianelli, M; Gulini, U; Marucci, Gabriella; Melchiorre, C; Spampinato, S.
Synthesis and alpha-Adrenoceptor Blocking Activity of the Enantiomers of Benzyl- (2-chloroethyl)-[2-(2-methoxyphenoxy)-1-methylethyl] amine Hydrochloride
1997-01-01 Giardina', Dario; Crucianelli, M; Marucci, Gabriella; Angeli, Piero; Melchiorre, C; Antolini, L.
Synthesis and pharmacological characterization of enantiomerically pure muscarinic agonists: difluoromuscarines
1997-01-01 Angeli, Piero; Cantalamessa, Franco; Cavagna, Roberto; Conti, Paola; De Amici, Marco; De Micheli, Marco; Gamba, Anna; Marucci, Gabriella
Simplified analogues of Ritanserin and their affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors
1998-01-01 Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Marucci, Gabriella; DI STEFANO, A.; Gessi, S.; Siniscalchi, A.; Borea, P. A.
Synthesis and antagonistic activity at muscarinic receptor subtypes of some 2-carbonyl derivatives of diphenidol
1999-01-01 Varoli, L; Angeli, Piero; Burnelli, S; Marucci, Gabriella; Recanatini, M.
Structure-Activity Relationships in 1,4-Benzodioxan-Related Compounds. 6. Role of the Dioxane Unit on Selectivity for Alpha1-Adrenoreceptor Subtypes
1999-01-01 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Poggesi, E.; Leonardi, A.; Melchiorre, C.
4-(4-Fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2c serotonin receptors
1999-01-01 Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Accorroni, Beatrice; Marucci, Gabriella; Gessi, S; Siniscalchi, A; Borea, Pa
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine
2000-01-01 DE AMICI, M.; Dallanoce, C.; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; DE MICHELIS, C.
Pharmacological profile of enantiomerically pure chiral muscarinic agonists - desoxymuscarines
2000-01-01 DE AMICI, M; Dallanoce, C; DE MICHELI, C; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; Sparapassi, L.
"[4-[[N-(3-Chlorophenyl)carbamoyl]-2-butynyl]-trimethylammonium (McN-A-343)-Related Compounds. Effect of the Butynyl Chain Inclusion into an Aromatic Unit of the Potency for Muscarinic Receptors
2000-01-01 Tumiatti, V; Angeli, Piero; Andrisano, V; Bolognesi, Ml; Cavalli, A; Marucci, Gabriella; Minarini, A; Recanatini, M; Rosini, M; Melchiorre, C.
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety
2000-01-01 Melchiorre, C.; Angeli, Piero; Bolognesi, M. L.; Chiarini, A.; Giardinà, D.; Gulini, U.; Leonardi, A.; Marucci, Gabriella; Minarini, A.; Pigini, Maria; Quaglia, Wilma; Rosini, M.; Tumiatti, V.
Structure-activity relationship at alpha-adrenergic receptors within a series of imidazoline analogues of cirazoline
2000-01-01 Pigini, Maria; Quaglia, Wilma; Gentili, Francesco; Marucci, Gabriella; Cantalamessa, F.; Franchini, S.; Sorbi, C.; Brasili, L.
Synthesis and α1-antagonist activity of derivatives of 4-chloro-5-{4-[2-(2-methoxyphenoxy)-ethyl]-1-piperazinyl}-3(2H)-pyridazinone
2000-01-01 Strappaghetti, Giovannella; Barbaro, Roberta; Marucci, Gabriella
Synthesis, Absolute Configuration and Antimuscarinic Activity of the Enantiomers of [1-(2,2-Diphenyl-[1,3]dioxolan-4-yl)-ethyl]-dimethyl-amine.
2001-01-01 Gulini, Ugo; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Giardina', Dario; Antolini, L; Franchini, S; Sorbi, C; Brasili, L.
Structure-Activity Relationships in 2,2-Diphenyl-2-ethylthioacetic Acid Esters: Unexpected Agonist Activity in a Series of Muscarinic Antagonists.
2001-01-01 Scapecchi, S.; Marucci, Gabriella; Matucci, R.; Angeli, Piero; Bellucci, C.; Buccioni, Michela; Dei, S.; Gualtieri, F.; Manetti, D.; Romanelli, M. N.; Teodori, E.
Analogues of Prazosin That Bear a Benextramine-Related Polyamine Backbone Exhibit Different Antagonism toward alpha1-Adrenoceptor Subtypes
2001-01-01 Bolognesi, M. L.; Marucci, Gabriella; Angeli, Piero; Buccioni, Michela; Minarini, A.; Rosini, M.; Tumiatti, V.; Melchiorre, C.
Structure-activity relationships among novel phenoxybenzamine-related beta-chloroethylamines
2002-01-01 Giardina', Dario; Crucianelli, M.; Angeli, Piero; Buccioni, M.; Gulini, Ugo; Marucci, Gabriella; Sagratini, Gianni; Melchiorre, C.
Structure-Activity Relatioships Among Novel Phenoxybenzamine-Related Beta-Chloroethylamines.
2002-01-01 Giardina', Dario; Crucianelli, M; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Gulini, Ugo; Sagratini, Gianni; Melchiorre, C.
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
“Tetraamines as Lead Compounds for the “Pharmacological Evaluation of Prazosin and Doxazosin-related Compounds with Modified Piperazine Ring”. | 1-gen-1996 | Giardinà, D; Crucianelli, M; Marucci, Gabriella; Melchiorre, C; Polidori, Carlo; Pompei, Pierluigi; Massi, Maurizio | Articolo | |
SAR Studies on the Potent and Selective Muscarinic Antagonist 2-Ethylthio-2,2-diphenylacetic Acid N,N-Diethylaminoethyl Ester | 1-gen-1997 | Scapecchi, S; Angeli, Piero; Dei, S; Ghelardini, C; Gualtieri, F; Marucci, Gabriella; Paparelli, F; Romanelli, M. N.; Teodori, E. | Articolo | |
“Synthesis and α1-Antagonist Activity of New Prazosin-and Benextramine-Related Tetraamine Disulfides”. | 1-gen-1997 | Giardinà, D; Crucianelli, M; Gulini, U; Marucci, Gabriella; Melchiorre, C; Spampinato, S. | Articolo | |
Synthesis and alpha-Adrenoceptor Blocking Activity of the Enantiomers of Benzyl- (2-chloroethyl)-[2-(2-methoxyphenoxy)-1-methylethyl] amine Hydrochloride | 1-gen-1997 | Giardina', Dario; Crucianelli, M; Marucci, Gabriella; Angeli, Piero; Melchiorre, C; Antolini, L. | Articolo | |
Synthesis and pharmacological characterization of enantiomerically pure muscarinic agonists: difluoromuscarines | 1-gen-1997 | Angeli, Piero; Cantalamessa, Franco; Cavagna, Roberto; Conti, Paola; De Amici, Marco; De Micheli, Marco; Gamba, Anna; Marucci, Gabriella | Articolo | |
Simplified analogues of Ritanserin and their affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors | 1-gen-1998 | Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Marucci, Gabriella; DI STEFANO, A.; Gessi, S.; Siniscalchi, A.; Borea, P. A. | Articolo | |
Synthesis and antagonistic activity at muscarinic receptor subtypes of some 2-carbonyl derivatives of diphenidol | 1-gen-1999 | Varoli, L; Angeli, Piero; Burnelli, S; Marucci, Gabriella; Recanatini, M. | Articolo | |
Structure-Activity Relationships in 1,4-Benzodioxan-Related Compounds. 6. Role of the Dioxane Unit on Selectivity for Alpha1-Adrenoreceptor Subtypes | 1-gen-1999 | Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Poggesi, E.; Leonardi, A.; Melchiorre, C. | Articolo | |
4-(4-Fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2c serotonin receptors | 1-gen-1999 | Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Accorroni, Beatrice; Marucci, Gabriella; Gessi, S; Siniscalchi, A; Borea, Pa | Articolo | |
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine | 1-gen-2000 | DE AMICI, M.; Dallanoce, C.; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; DE MICHELIS, C. | Articolo | |
Pharmacological profile of enantiomerically pure chiral muscarinic agonists - desoxymuscarines | 1-gen-2000 | DE AMICI, M; Dallanoce, C; DE MICHELI, C; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; Sparapassi, L. | Articolo | |
"[4-[[N-(3-Chlorophenyl)carbamoyl]-2-butynyl]-trimethylammonium (McN-A-343)-Related Compounds. Effect of the Butynyl Chain Inclusion into an Aromatic Unit of the Potency for Muscarinic Receptors | 1-gen-2000 | Tumiatti, V; Angeli, Piero; Andrisano, V; Bolognesi, Ml; Cavalli, A; Marucci, Gabriella; Minarini, A; Recanatini, M; Rosini, M; Melchiorre, C. | Articolo | |
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety | 1-gen-2000 | Melchiorre, C.; Angeli, Piero; Bolognesi, M. L.; Chiarini, A.; Giardinà, D.; Gulini, U.; Leonardi, A.; Marucci, Gabriella; Minarini, A.; Pigini, Maria; Quaglia, Wilma; Rosini, M.; Tumiatti, V. | Articolo | |
Structure-activity relationship at alpha-adrenergic receptors within a series of imidazoline analogues of cirazoline | 1-gen-2000 | Pigini, Maria; Quaglia, Wilma; Gentili, Francesco; Marucci, Gabriella; Cantalamessa, F.; Franchini, S.; Sorbi, C.; Brasili, L. | Articolo | |
Synthesis and α1-antagonist activity of derivatives of 4-chloro-5-{4-[2-(2-methoxyphenoxy)-ethyl]-1-piperazinyl}-3(2H)-pyridazinone | 1-gen-2000 | Strappaghetti, Giovannella; Barbaro, Roberta; Marucci, Gabriella | Articolo | |
Synthesis, Absolute Configuration and Antimuscarinic Activity of the Enantiomers of [1-(2,2-Diphenyl-[1,3]dioxolan-4-yl)-ethyl]-dimethyl-amine. | 1-gen-2001 | Gulini, Ugo; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Giardina', Dario; Antolini, L; Franchini, S; Sorbi, C; Brasili, L. | Articolo | |
Structure-Activity Relationships in 2,2-Diphenyl-2-ethylthioacetic Acid Esters: Unexpected Agonist Activity in a Series of Muscarinic Antagonists. | 1-gen-2001 | Scapecchi, S.; Marucci, Gabriella; Matucci, R.; Angeli, Piero; Bellucci, C.; Buccioni, Michela; Dei, S.; Gualtieri, F.; Manetti, D.; Romanelli, M. N.; Teodori, E. | Articolo | |
Analogues of Prazosin That Bear a Benextramine-Related Polyamine Backbone Exhibit Different Antagonism toward alpha1-Adrenoceptor Subtypes | 1-gen-2001 | Bolognesi, M. L.; Marucci, Gabriella; Angeli, Piero; Buccioni, Michela; Minarini, A.; Rosini, M.; Tumiatti, V.; Melchiorre, C. | Articolo | |
Structure-activity relationships among novel phenoxybenzamine-related beta-chloroethylamines | 1-gen-2002 | Giardina', Dario; Crucianelli, M.; Angeli, Piero; Buccioni, M.; Gulini, Ugo; Marucci, Gabriella; Sagratini, Gianni; Melchiorre, C. | Articolo | |
Structure-Activity Relatioships Among Novel Phenoxybenzamine-Related Beta-Chloroethylamines. | 1-gen-2002 | Giardina', Dario; Crucianelli, M; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Gulini, Ugo; Sagratini, Gianni; Melchiorre, C. | Articolo |
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