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Titolo Data di pubblicazione Autore(i) Tipo File
Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole 1-gen-2002 Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria Articolo
Structure-Activity Relatioships Among Novel Phenoxybenzamine-Related Beta-Chloroethylamines. 1-gen-2002 Giardina', Dario; Crucianelli, M; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Gulini, Ugo; Sagratini, Gianni; Melchiorre, C. Articolo
Deoxamuscaroneoxime Devatives as useful Muscarinic Aginist to Explore the Muscarinic Subsite: Demox, Amodulator of Orthosteric and Allosteric Site at Cardiac Muscarinic M2 Receptors. 1-gen-2002 Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Piergentili, Alessandro; Giannella, Mario; Quaglia, Wilma; Pigini, Maria; Cantalamessa, Franco; Nasuti, Cinzia Carla; Novi, F; Maggio, R; Quasem, A. R.; Spampinato, S. Articolo
Structure-Activity Relationships of Methoctramine-Related Polyamines as Muscular Nicotinic Receptor Noncompetitive Antagonists. 2. Role of Polymethylene Chain Lengths Separating Amine Functions and of Substituents on the Terminal Nitrogen Atoms. 1-gen-2002 Rosini, M.; Bixel, M. G.; Marucci, Gabriella; Budriesi, R.; Krauss, M.; Bolognesi, M. L.; Minarini, A.; Tumiatti, V.; Hucho, F.; Melchiorre, C. Articolo
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure 1-gen-2002 Bolognesi, M.; Bixel, M. G.; Marucci, Gabriella; Bartolini, M.; Krauss, M.; Angeli, Piero; Antonello, A.; Rosini, M.; Tumiatti, V.; Hucho, F.; Melchiorre, C. Articolo
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives 1-gen-2002 Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma Articolo
Medicinal chemistry and pharmacology of purinergic receptors 1-gen-2003 Cristalli, Gloria; Costanzi, S; Giorgioni, Gianfabio; Lambertucci, Catia; Marucci, Gabriella; Taffi, S; Vittori, Sauro; Volpini, Rosaria ORGANIZZAZIONE DI EVENTI
14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry 1-gen-2003 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma ORGANIZZAZIONE DI EVENTI
5HT2B receptor antagonists: a probe for spotting the pharmacophore 1-gen-2003 Claudi, F.; Giorgioni, Gianfabio; Accorroni, Beatrice; Di Stefano, A.; Marucci, Gabriella; Siniscalchi, A. Poster atto convegno su volume
Searching for cyclazosin analogues as alfa1B-adrenoceptor antagonists 1-gen-2003 Giardina', Dario; Polimanti, O.; Sagratini, Gianni; Angeli, Piero; Gulini, Ugo; Marucci, Gabriella; Melchiorre, C.; Poggesi, E.; Leonardi, A. Articolo
1,3-Dioxolane-based ligands as a novel class of alpha(1)-adrenoceptor antagonists 1-gen-2003 Brasili, L.; Sorbi, C.; Franchini, S.; Manicardi, M.; Angeli, Piero; Marucci, Gabriella; Leonardi, A.; Poggesi, E. Articolo
Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol 1-gen-2003 Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Cavalli, A; Marucci, Gabriella; Recanatini, M. Articolo
Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine 1-gen-2003 Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario Articolo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine 1-gen-2003 Tumiatti, V; Rosini, M.; Bartolini, M.; Cavalli, A.; Marucci, Gabriella; Andrisano, V.; Angeli, Piero; Banzi, R.; Minarini, A.; Recanatini, M.; Melchiorre, C. Articolo
Prazosin-Related Compounds. Effect of Transforming the Piperazinylquinazoline Moiety into an Aminomethyltetrahydroacridine System on the Affinity for alpha1-Adrenoceptors 1-gen-2003 Rosini, M; Antonello, A; Cavalli, A; Bolognesi, Ml; Minarini, A; Marucci, Gabriella; Poggesi, E; Leonardi, A; Melchiorre, C. Articolo
(+)-Cyclazosin derivatives as α1-adrenoceptor antagonists 1-gen-2004 Sagratini, Gianni; Buccioni, Michela; Gulini, U.; Marucci, Gabriella; Melchiorre, C.; Leonardi, A.; Testa, R.; Giardinà, D. Articolo
Molecular modulation of muscarinic antagonists. Synthesis and pharmacological profile of 2,2-diphenyl-2-ethylthioacetic and 3,3-diphenyl-3-ethylthiopropionic acid derivatives characterized by a dipeptide spacer. 1-gen-2004 S., Scapecchi; C., Martelli; Angeli, Piero; C., Bellucci; Buccioni, Michela; S., Dei; F., Gualtieri; Marucci, Gabriella; R., Matucci; M. N., Romanelli; E., Teodori Articolo
Molecular modulation of muscarinic antagonists. Synthesis and affinity profile of 2,2-diphenyl-2-ethylthio-acetic acid esters designed to probe the binding site cavity. 1-gen-2004 Scapecchi, S; Martini, E; Bellucci, C; Buccioni, Michela; Dei, S; Guandalini, L; Manetti, D; Martelli, C; Marucci, Gabriella; Matucci, R. Articolo
Polyamines may modulate both G protein-coupled receptors and G proteins. 1-gen-2004 Marucci, Gabriella; Novi, F; Banzi, R; Bolognesi, M. L.; Buccioni, Michela; Minarini, A; Rosini, M; Angeli, Piero; Maggio, R; Melchiorre, C. Articolo
Design, synthesis, and biological evaluation of prazosin-related derivatives as multipotent compounds 1-gen-2005 Antonello, A.; Hrelia, P.; Leonardi, A.; Marucci, Gabriella; Rosini, M.; Tarozzi, A.; Tumiatti, V.; Melchiorre, C. Articolo
Mostrati risultati da 41 a 60 di 170
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