Sfoglia per Autore
Identification of alpha(1)-adrenoceptor subtypes involved in contraction of young CD rat epididymal vas deferens
2009-01-01 Buccioni, Michela; Kandhavelu, M; Angeli, Piero; Cristalli, Gloria; DAL BEN, Diego; Giardinà, D; Lambertucci, Catia; Lammi, C; Volpini, Rosaria; Marucci, Gabriella
8-Bromo-9-alkyl adenine derivatives as tools for developing new adenosine A(2A) and A(2B) receptors ligands
2009-01-01 Lambertucci, Catia; Antonini, Ippolito; Buccioni, Michela; DAL BEN, Diego; Kachare, Dd; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Novel potent and highly selective human A(3) adenosine receptor antagonists belonging to the 4-amido-2-arylpyrazolo[3,4-c]quinoline series: Molecular docking analysis and pharmacological studies
2009-01-01 Colotta, V.; Capelli, F.; Lenzi, O.; Catarzi, D.; Varano, F.; Poli, D.; Vincenzi, F.; Varani, K.; Borea, P. A.; DAL BEN, Diego; Volpini, Rosaria; Cristalli, Gloria; Filacchioni, G.
Synthesis and biological evaluation of 2-alkynyl-N6-methyl-5'-N-methylcarboxamidoadenosine derivatives as potent and highly selective agonists for the human adenosine A(3) receptor
2009-01-01 Volpini, Rosaria; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Marucci, Gabriella; Ramadori, At; Klotz, K. N.; Cristalli, Gloria
Substituted adenine derivatives as novel P2X3 receptor ligands
2010-01-01 Panmand, Ds; DAL BEN, Diego; Giacobbe, D; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Nistri, A; Cristalli, Gloria
Molecular modeling studies on the human neuropeptide S receptor and its antagonists.
2010-01-01 DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria
Molecular modeling study on potent and selective adenosine A3 receptor agonists.
2010-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria
New substituted MECA derivatives as potent and selective agonists for the human adenosine A3 receptor
2010-01-01 Lambertucci, Catia; DAL BEN, Diego; Lammi, C; Marucci, Gabriella; Ramadori, At; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Identification of putative guanosine receptor in rat brain
2010-01-01 Lammi, C; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria
Human adenosine A3 receptor as selective target of new 2-aralkynyl-N6-methyl-MECA derivatives
2010-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Ramadori, At; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
GTP-Eu binding assay optimization for the adenosine A3 receptor ligands screening
2010-01-01 Buccioni, Michela; DAL BEN, Diego; Giacobbe, D; Lammi, C; Marucci, Gabriella; Panmand, Ds; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Adenosine receptor modeling: what does the A2A crystal structure tell us?
2010-01-01 DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria
New 9-methyl-8-(4-hydroxyphenyl)adenine derivatives as A(1) adenosine receptor antagonists
2011-01-01 Lambertucci, Catia; Buccioni, Michela; Cacciarri, B; DAL BEN, Diego; Federico, S; Klotz, K. N.; Marucci, Gabriella; Volpini, Rosaria; Spalluto, G; Cristalli, Gloria
Comparison and optimization of transient transfection methods at human astrocytoma cell line 1321N1
2011-01-01 Marucci, Gabriella; Lammi, C; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Amantini, Consuelo; Santoni, Giorgio; Kandhavelu, M; Abbracchio, Mp; Lecca, D; Volpini, Rosaria; Cristalli, Gloria
The importance of alkynyl chain presence for the activity of adenine nucleosides/nucleotides on purinergic receptors
2011-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria
Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17
2011-01-01 Buccioni, Michela; Marucci, Gabriella; DAL BEN, Diego; Giacobbe, Dania; Lambertucci, Catia; Soverchia, Laura; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria
Synthesis, structure-affinity relationships and molecular modeling studies of novel pyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists
2011-01-01 Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Squarcialupi, L; Filacchioni, G; Varani, K; Vincenzi, F; Borea, Pa; DAL BEN, Diego; Lambertucci, Catia; Cristalli, Gloria
Neuropeptide S Receptor: recent updates on non-peptide antagonist discovery
2011-01-01 DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria
Evidence for the existence of a specific G protein-coupled receptor activated by guanosine
2011-01-01 Volpini, Rosaria; Marucci, Gabriella; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Mishra, Cr; Thomas, Ajiroghene; Cristalli, Gloria
GPR17 ligands: synthesis and characterization of new potent agonists
2012-01-01 Volpini, Rosaria; Buccioni, Michela; Ceruti, S; DAL BEN, Diego; Daniele, S; Lambertucci, Catia; Lecca, D; Marucci, Gabriella; Trincavelli, Ml; Martini, C; Abbracchio, Mp; Cristalli, Gloria
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Identification of alpha(1)-adrenoceptor subtypes involved in contraction of young CD rat epididymal vas deferens | 1-gen-2009 | Buccioni, Michela; Kandhavelu, M; Angeli, Piero; Cristalli, Gloria; DAL BEN, Diego; Giardinà, D; Lambertucci, Catia; Lammi, C; Volpini, Rosaria; Marucci, Gabriella | Articolo | |
8-Bromo-9-alkyl adenine derivatives as tools for developing new adenosine A(2A) and A(2B) receptors ligands | 1-gen-2009 | Lambertucci, Catia; Antonini, Ippolito; Buccioni, Michela; DAL BEN, Diego; Kachare, Dd; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Novel potent and highly selective human A(3) adenosine receptor antagonists belonging to the 4-amido-2-arylpyrazolo[3,4-c]quinoline series: Molecular docking analysis and pharmacological studies | 1-gen-2009 | Colotta, V.; Capelli, F.; Lenzi, O.; Catarzi, D.; Varano, F.; Poli, D.; Vincenzi, F.; Varani, K.; Borea, P. A.; DAL BEN, Diego; Volpini, Rosaria; Cristalli, Gloria; Filacchioni, G. | Articolo | |
Synthesis and biological evaluation of 2-alkynyl-N6-methyl-5'-N-methylcarboxamidoadenosine derivatives as potent and highly selective agonists for the human adenosine A(3) receptor | 1-gen-2009 | Volpini, Rosaria; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Marucci, Gabriella; Ramadori, At; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Substituted adenine derivatives as novel P2X3 receptor ligands | 1-gen-2010 | Panmand, Ds; DAL BEN, Diego; Giacobbe, D; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Nistri, A; Cristalli, Gloria | Abstract atto convegno su rivista | |
Molecular modeling studies on the human neuropeptide S receptor and its antagonists. | 1-gen-2010 | DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Molecular modeling study on potent and selective adenosine A3 receptor agonists. | 1-gen-2010 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
New substituted MECA derivatives as potent and selective agonists for the human adenosine A3 receptor | 1-gen-2010 | Lambertucci, Catia; DAL BEN, Diego; Lammi, C; Marucci, Gabriella; Ramadori, At; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Abstract atto convegno su rivista | |
Identification of putative guanosine receptor in rat brain | 1-gen-2010 | Lammi, C; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria | Abstract atto convegno su rivista | |
Human adenosine A3 receptor as selective target of new 2-aralkynyl-N6-methyl-MECA derivatives | 1-gen-2010 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Ramadori, At; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Abstract atto convegno su rivista | |
GTP-Eu binding assay optimization for the adenosine A3 receptor ligands screening | 1-gen-2010 | Buccioni, Michela; DAL BEN, Diego; Giacobbe, D; Lammi, C; Marucci, Gabriella; Panmand, Ds; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Abstract atto convegno su rivista | |
Adenosine receptor modeling: what does the A2A crystal structure tell us? | 1-gen-2010 | DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
New 9-methyl-8-(4-hydroxyphenyl)adenine derivatives as A(1) adenosine receptor antagonists | 1-gen-2011 | Lambertucci, Catia; Buccioni, Michela; Cacciarri, B; DAL BEN, Diego; Federico, S; Klotz, K. N.; Marucci, Gabriella; Volpini, Rosaria; Spalluto, G; Cristalli, Gloria | Articolo | |
Comparison and optimization of transient transfection methods at human astrocytoma cell line 1321N1 | 1-gen-2011 | Marucci, Gabriella; Lammi, C; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Amantini, Consuelo; Santoni, Giorgio; Kandhavelu, M; Abbracchio, Mp; Lecca, D; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
The importance of alkynyl chain presence for the activity of adenine nucleosides/nucleotides on purinergic receptors | 1-gen-2011 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17 | 1-gen-2011 | Buccioni, Michela; Marucci, Gabriella; DAL BEN, Diego; Giacobbe, Dania; Lambertucci, Catia; Soverchia, Laura; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Synthesis, structure-affinity relationships and molecular modeling studies of novel pyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists | 1-gen-2011 | Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Squarcialupi, L; Filacchioni, G; Varani, K; Vincenzi, F; Borea, Pa; DAL BEN, Diego; Lambertucci, Catia; Cristalli, Gloria | Articolo | |
Neuropeptide S Receptor: recent updates on non-peptide antagonist discovery | 1-gen-2011 | DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Evidence for the existence of a specific G protein-coupled receptor activated by guanosine | 1-gen-2011 | Volpini, Rosaria; Marucci, Gabriella; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Mishra, Cr; Thomas, Ajiroghene; Cristalli, Gloria | Articolo | |
GPR17 ligands: synthesis and characterization of new potent agonists | 1-gen-2012 | Volpini, Rosaria; Buccioni, Michela; Ceruti, S; DAL BEN, Diego; Daniele, S; Lambertucci, Catia; Lecca, D; Marucci, Gabriella; Trincavelli, Ml; Martini, C; Abbracchio, Mp; Cristalli, Gloria | Abstract atto convegno su rivista |
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