Sfoglia per Autore
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine
2000-01-01 DE AMICI, M.; Dallanoce, C.; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; DE MICHELIS, C.
Pharmacological profile of enantiomerically pure chiral muscarinic agonists - desoxymuscarines
2000-01-01 DE AMICI, M; Dallanoce, C; DE MICHELI, C; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; Sparapassi, L.
"[4-[[N-(3-Chlorophenyl)carbamoyl]-2-butynyl]-trimethylammonium (McN-A-343)-Related Compounds. Effect of the Butynyl Chain Inclusion into an Aromatic Unit of the Potency for Muscarinic Receptors
2000-01-01 Tumiatti, V; Angeli, Piero; Andrisano, V; Bolognesi, Ml; Cavalli, A; Marucci, Gabriella; Minarini, A; Recanatini, M; Rosini, M; Melchiorre, C.
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety
2000-01-01 Melchiorre, C.; Angeli, Piero; Bolognesi, M. L.; Chiarini, A.; Giardinà, D.; Gulini, U.; Leonardi, A.; Marucci, Gabriella; Minarini, A.; Pigini, Maria; Quaglia, Wilma; Rosini, M.; Tumiatti, V.
Receptors in neurodegenerative diseases, muscarinic cholinergic receptors
2000-01-01 Angeli, Piero
Synthesis, Absolute Configuration and Antimuscarinic Activity of the Enantiomers of [1-(2,2-Diphenyl-[1,3]dioxolan-4-yl)-ethyl]-dimethyl-amine.
2001-01-01 Gulini, Ugo; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Giardina', Dario; Antolini, L; Franchini, S; Sorbi, C; Brasili, L.
Analogues of Prazosin That Bear a Benextramine-Related Polyamine Backbone Exhibit Different Antagonism toward alpha1-Adrenoceptor Subtypes
2001-01-01 Bolognesi, M. L.; Marucci, Gabriella; Angeli, Piero; Buccioni, Michela; Minarini, A.; Rosini, M.; Tumiatti, V.; Melchiorre, C.
Structure-Activity Relationships in 2,2-Diphenyl-2-ethylthioacetic Acid Esters: Unexpected Agonist Activity in a Series of Muscarinic Antagonists.
2001-01-01 Scapecchi, S.; Marucci, Gabriella; Matucci, R.; Angeli, Piero; Bellucci, C.; Buccioni, Michela; Dei, S.; Gualtieri, F.; Manetti, D.; Romanelli, M. N.; Teodori, E.
Structure-activity relationships among novel phenoxybenzamine-related beta-chloroethylamines
2002-01-01 Giardina', Dario; Crucianelli, M.; Angeli, Piero; Buccioni, M.; Gulini, Ugo; Marucci, Gabriella; Sagratini, Gianni; Melchiorre, C.
Structure-Activity Relatioships Among Novel Phenoxybenzamine-Related Beta-Chloroethylamines.
2002-01-01 Giardina', Dario; Crucianelli, M; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Gulini, Ugo; Sagratini, Gianni; Melchiorre, C.
Deoxamuscaroneoxime Devatives as useful Muscarinic Aginist to Explore the Muscarinic Subsite: Demox, Amodulator of Orthosteric and Allosteric Site at Cardiac Muscarinic M2 Receptors.
2002-01-01 Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Piergentili, Alessandro; Giannella, Mario; Quaglia, Wilma; Pigini, Maria; Cantalamessa, Franco; Nasuti, Cinzia Carla; Novi, F; Maggio, R; Quasem, A. R.; Spampinato, S.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure
2002-01-01 Bolognesi, M.; Bixel, M. G.; Marucci, Gabriella; Bartolini, M.; Krauss, M.; Angeli, Piero; Antonello, A.; Rosini, M.; Tumiatti, V.; Hucho, F.; Melchiorre, C.
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives
2002-01-01 Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma
Searching for cyclazosin analogues as alfa1B-adrenoceptor antagonists
2003-01-01 Giardina', Dario; Polimanti, O.; Sagratini, Gianni; Angeli, Piero; Gulini, Ugo; Marucci, Gabriella; Melchiorre, C.; Poggesi, E.; Leonardi, A.
1,3-Dioxolane-based ligands as a novel class of alpha(1)-adrenoceptor antagonists
2003-01-01 Brasili, L.; Sorbi, C.; Franchini, S.; Manicardi, M.; Angeli, Piero; Marucci, Gabriella; Leonardi, A.; Poggesi, E.
Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol
2003-01-01 Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Cavalli, A; Marucci, Gabriella; Recanatini, M.
14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry
2003-01-01 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine
2003-01-01 Tumiatti, V; Rosini, M.; Bartolini, M.; Cavalli, A.; Marucci, Gabriella; Andrisano, V.; Angeli, Piero; Banzi, R.; Minarini, A.; Recanatini, M.; Melchiorre, C.
Modulation of receptors and G-proteins
2004-01-01 Angeli, Piero
Molecular modulation of muscarinic antagonists. Synthesis and pharmacological profile of 2,2-diphenyl-2-ethylthioacetic and 3,3-diphenyl-3-ethylthiopropionic acid derivatives characterized by a dipeptide spacer.
2004-01-01 S., Scapecchi; C., Martelli; Angeli, Piero; C., Bellucci; Buccioni, Michela; S., Dei; F., Gualtieri; Marucci, Gabriella; R., Matucci; M. N., Romanelli; E., Teodori
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine | 1-gen-2000 | DE AMICI, M.; Dallanoce, C.; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; DE MICHELIS, C. | Articolo | |
Pharmacological profile of enantiomerically pure chiral muscarinic agonists - desoxymuscarines | 1-gen-2000 | DE AMICI, M; Dallanoce, C; DE MICHELI, C; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; Sparapassi, L. | Articolo | |
"[4-[[N-(3-Chlorophenyl)carbamoyl]-2-butynyl]-trimethylammonium (McN-A-343)-Related Compounds. Effect of the Butynyl Chain Inclusion into an Aromatic Unit of the Potency for Muscarinic Receptors | 1-gen-2000 | Tumiatti, V; Angeli, Piero; Andrisano, V; Bolognesi, Ml; Cavalli, A; Marucci, Gabriella; Minarini, A; Recanatini, M; Rosini, M; Melchiorre, C. | Articolo | |
Alpha 1-adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety | 1-gen-2000 | Melchiorre, C.; Angeli, Piero; Bolognesi, M. L.; Chiarini, A.; Giardinà, D.; Gulini, U.; Leonardi, A.; Marucci, Gabriella; Minarini, A.; Pigini, Maria; Quaglia, Wilma; Rosini, M.; Tumiatti, V. | Articolo | |
Receptors in neurodegenerative diseases, muscarinic cholinergic receptors | 1-gen-2000 | Angeli, Piero | Articolo | |
Synthesis, Absolute Configuration and Antimuscarinic Activity of the Enantiomers of [1-(2,2-Diphenyl-[1,3]dioxolan-4-yl)-ethyl]-dimethyl-amine. | 1-gen-2001 | Gulini, Ugo; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Giardina', Dario; Antolini, L; Franchini, S; Sorbi, C; Brasili, L. | Articolo | |
Analogues of Prazosin That Bear a Benextramine-Related Polyamine Backbone Exhibit Different Antagonism toward alpha1-Adrenoceptor Subtypes | 1-gen-2001 | Bolognesi, M. L.; Marucci, Gabriella; Angeli, Piero; Buccioni, Michela; Minarini, A.; Rosini, M.; Tumiatti, V.; Melchiorre, C. | Articolo | |
Structure-Activity Relationships in 2,2-Diphenyl-2-ethylthioacetic Acid Esters: Unexpected Agonist Activity in a Series of Muscarinic Antagonists. | 1-gen-2001 | Scapecchi, S.; Marucci, Gabriella; Matucci, R.; Angeli, Piero; Bellucci, C.; Buccioni, Michela; Dei, S.; Gualtieri, F.; Manetti, D.; Romanelli, M. N.; Teodori, E. | Articolo | |
Structure-activity relationships among novel phenoxybenzamine-related beta-chloroethylamines | 1-gen-2002 | Giardina', Dario; Crucianelli, M.; Angeli, Piero; Buccioni, M.; Gulini, Ugo; Marucci, Gabriella; Sagratini, Gianni; Melchiorre, C. | Articolo | |
Structure-Activity Relatioships Among Novel Phenoxybenzamine-Related Beta-Chloroethylamines. | 1-gen-2002 | Giardina', Dario; Crucianelli, M; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Gulini, Ugo; Sagratini, Gianni; Melchiorre, C. | Articolo | |
Deoxamuscaroneoxime Devatives as useful Muscarinic Aginist to Explore the Muscarinic Subsite: Demox, Amodulator of Orthosteric and Allosteric Site at Cardiac Muscarinic M2 Receptors. | 1-gen-2002 | Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Piergentili, Alessandro; Giannella, Mario; Quaglia, Wilma; Pigini, Maria; Cantalamessa, Franco; Nasuti, Cinzia Carla; Novi, F; Maggio, R; Quasem, A. R.; Spampinato, S. | Articolo | |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure | 1-gen-2002 | Bolognesi, M.; Bixel, M. G.; Marucci, Gabriella; Bartolini, M.; Krauss, M.; Angeli, Piero; Antonello, A.; Rosini, M.; Tumiatti, V.; Hucho, F.; Melchiorre, C. | Articolo | |
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives | 1-gen-2002 | Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma | Articolo | |
Searching for cyclazosin analogues as alfa1B-adrenoceptor antagonists | 1-gen-2003 | Giardina', Dario; Polimanti, O.; Sagratini, Gianni; Angeli, Piero; Gulini, Ugo; Marucci, Gabriella; Melchiorre, C.; Poggesi, E.; Leonardi, A. | Articolo | |
1,3-Dioxolane-based ligands as a novel class of alpha(1)-adrenoceptor antagonists | 1-gen-2003 | Brasili, L.; Sorbi, C.; Franchini, S.; Manicardi, M.; Angeli, Piero; Marucci, Gabriella; Leonardi, A.; Poggesi, E. | Articolo | |
Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol | 1-gen-2003 | Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Cavalli, A; Marucci, Gabriella; Recanatini, M. | Articolo | |
14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry | 1-gen-2003 | Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | ORGANIZZAZIONE DI EVENTI | |
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine | 1-gen-2003 | Tumiatti, V; Rosini, M.; Bartolini, M.; Cavalli, A.; Marucci, Gabriella; Andrisano, V.; Angeli, Piero; Banzi, R.; Minarini, A.; Recanatini, M.; Melchiorre, C. | Articolo | |
Modulation of receptors and G-proteins | 1-gen-2004 | Angeli, Piero | Articolo | |
Molecular modulation of muscarinic antagonists. Synthesis and pharmacological profile of 2,2-diphenyl-2-ethylthioacetic and 3,3-diphenyl-3-ethylthiopropionic acid derivatives characterized by a dipeptide spacer. | 1-gen-2004 | S., Scapecchi; C., Martelli; Angeli, Piero; C., Bellucci; Buccioni, Michela; S., Dei; F., Gualtieri; Marucci, Gabriella; R., Matucci; M. N., Romanelli; E., Teodori | Articolo |
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