Sfoglia per Autore
2'-C-Methyl analogs of selective adenosine receptors agonists: synthesis and binding studies
1996-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Costa, B; Martini, C; Lucacchini, A.
Preparation of purine and 8-azapurine derivatives for treatment of acquired immune deficiency syndrome.
1996-01-01 Grifantini, Mario; Franchetti, Palmarisa; Cappellacci, Loredana; La Colla, P; Loi, A. G.; Piras, G.
IMP Dehydrogenase as a target of antitumor and antiviral chemotherapy
1996-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario
Synthesis and IMP dehydrogenase (type I and type II) inhibitory activity of isosteric NAD analogs derived from thiophenfurin and furanfurin
1997-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; ABU SHEIKHA, G; Jayaram, Hn; Schneider, Bp; Sint, T; Gurudutt, Vv; Collart, Fr; Huberman, E; Grifantini, Mario
Synthesis and cytotoxic activity of selenophenfurin, a new inhibitor of IMP dehydrogenase
1997-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; ABU SHEIKHA, G; Jayaram, Hn; Gurudutt, Vv; Sint, T; Schneider, Bp; GOLDSTEIN BM PERRA, G; Poma, S; LA COLLA, P; Grifantini, Mario
Synthesis, structure, and antiproliferative activity of selenophenfurin, an IMP dehydrogenase inhibitor analogue of selenazofurin.
1997-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; ABU SHEIKHA, G; Jayaram, Hn; Gurudutt, Vv; Sint, T; Schneider, Bp; Jones, Wd; Goldstein, Bm; Perra, G; DE MONTIS, A; Loi, G; LA COLLA, P; Grifantini, Mario
Potent and selective inhibitors of human immunodeficiency virus protease structurally related to L-694,746.
1998-01-01 Franchetti, Palmarisa; Perlini, P; ABU SHEIKHA, G; Cappellacci, Loredana; Grifantini, Mario; Loi, Ag; DE MONTIS, A; Pani, A; Marongiu, Me; LA COLLA, P.
2'-C-Methyl analogues of selective adenosine receptor agonists: synthesis and binding studies.
1998-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Marchetti, S; Trincavelli, L; Martini, C; Mazzoni, Mr; Lucacchini, A; Grifantini, Mario
Isosteric Analogues of Nicotinamide Adenine Dinucleotide Derived from Furanfurin, Thiophenfurin, and Selenophenfurin as Mammalian Inosine Monophosphate dehydrogenase (Type I and II) Inhibitors
1998-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Perlini, P.; Jayaram, H. N.; Butler, A.; Schneider, B. P.; Collart, F. R.; Huberman, E.; Grifantini, Mario
Labelling of A1 and A3 adenosine receptors with the new selective A1 agonist 2'-Me-CCPA
1998-01-01 Amenta, Francesco; P., Barili; Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario
Structure-activity relationships of tiazofurin analogs: synthesis and computational studies of 4'-thio derivatives of thiophenfurin and furanfurin
1999-01-01 Franchetti, Palmarisa; Marchetti, S; Cappellacci, Loredana; Grifantini, Mario; Goldstein, Bm; Dukhan, D; Barascut, J. L.; Imbach, J. L.
Selective targeting to macrophages of a new homodinucleotide active aginst human immunodeficiency virus and herpes simplex virus
1999-01-01 Rossi, L; Serafini, S; Cappellacci, Loredana; Balestra, E; Brandi, G; Schiavano Giuditta, F; Franchetti, Palmarisa; Grifantini, Mario; Perno, C. F.; Magnani, M.
Red Blood cells as drug delivery system for antiviral nucleotide analogues
1999-01-01 Rossi, L.; Serafini, S.; Brandi, G.; Magnani, M.; Balestra, E.; Perno, C. F.; Cappellacci, Loredana; Franchetti, Palmarisa
Synthesis, Conformational Analysis, and Biological Activity of C-Thioribonucleosides Related to Tiazofurin
2000-01-01 Franchetti, Palmarisa; Marchetti, S.; Cappellacci, Loredana; Jayaram, H. N.; Yalowitz, J. A.; Goldstein, B. M.; Barascut, J. L.; Dukhan, D.; Imbach, J. L.; Grifantini, Mario
A new acyclic heterodinucleotide active against Human Immunodeficiency Virus and Herpes Simplex Virus
2000-01-01 Franchetti, Palmarisa; ABU SHEIKHA, G.; Cappellacci, Loredana; Marchetti, S.; Grifantini, Mario; Balestra, E.; Perno, C. F.; Benatti, U.; Brandi, G.; Rossi, L; Magnani, M.
C-Nucleoside Analogues of Furanfurin as Ligands to A(1) Adenosine Receptors
2000-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Marchetti, S.; Martini, C.; Costa, B.; Varani, K.; Borea, P. A.; Grifantini, Mario
Inhibition of human immunodeficency virus replication in macrophages by red blood cell-mediated delivery of a heterodinucleotide of azidothymidine and 9-(R)-2-(phosphonomethoxypropyl)adenine.
2001-01-01 Franchetti, Palmarisa; Rossi, L; Cappellacci, Loredana; Pasqualini, M; Grifantini, Mario; Balestra, E; Forbici, F; Perno, C. F.; Serafini, S; Magnani, M.
Erythrocyte-mediated delivery of a new homodinucleotide active against human immunodeficiency virus and herpes simplex virus
2001-01-01 Rossi, L; Serafini, S; Cappellacci, Loredana; Balestra, E; Brandi, G; Schiavano, G. F.; Franchetti, Palmarisa; Grifantini, Mario; Perno, C. F.; Magnani, M.
A new C-Nucleoside Analogue of Tiazofurin: Synthesis and Biological Evaluation of 2-beta-D-Ribofuranosylimidazole-4-carboxamide (Imidazofurin)
2001-01-01 Franchetti, Palmarisa; Marchetti, S.; Cappellacci, Loredana; Yalowitz, J. A.; Jayaram, H. N.; Goldstein, B. M.; Grifantini, Mario
Pharmacokinetic and antiretroviral activity in mice of oral [P1,P2-bis[2-(adenin-9-yl)ethoxymethyl]phosphonate], a prodrug of 9-(2-phosphonylmethoxyethyl)adenine
2002-01-01 Rossi, L.; Dominici, S.; Serafini, S.; Casabianca, A.; Cerasi, A.; Chiarantini, L.; Celeste, A. G.; Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Magnani, M.
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
2'-C-Methyl analogs of selective adenosine receptors agonists: synthesis and binding studies | 1-gen-1996 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Costa, B; Martini, C; Lucacchini, A. | Poster atto convegno su rivista | |
Preparation of purine and 8-azapurine derivatives for treatment of acquired immune deficiency syndrome. | 1-gen-1996 | Grifantini, Mario; Franchetti, Palmarisa; Cappellacci, Loredana; La Colla, P; Loi, A. G.; Piras, G. | 07 BREVETTO | |
IMP Dehydrogenase as a target of antitumor and antiviral chemotherapy | 1-gen-1996 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario | Articolo | |
Synthesis and IMP dehydrogenase (type I and type II) inhibitory activity of isosteric NAD analogs derived from thiophenfurin and furanfurin | 1-gen-1997 | Franchetti, Palmarisa; Cappellacci, Loredana; ABU SHEIKHA, G; Jayaram, Hn; Schneider, Bp; Sint, T; Gurudutt, Vv; Collart, Fr; Huberman, E; Grifantini, Mario | Articolo | |
Synthesis and cytotoxic activity of selenophenfurin, a new inhibitor of IMP dehydrogenase | 1-gen-1997 | Cappellacci, Loredana; Franchetti, Palmarisa; ABU SHEIKHA, G; Jayaram, Hn; Gurudutt, Vv; Sint, T; Schneider, Bp; GOLDSTEIN BM PERRA, G; Poma, S; LA COLLA, P; Grifantini, Mario | Articolo | |
Synthesis, structure, and antiproliferative activity of selenophenfurin, an IMP dehydrogenase inhibitor analogue of selenazofurin. | 1-gen-1997 | Franchetti, Palmarisa; Cappellacci, Loredana; ABU SHEIKHA, G; Jayaram, Hn; Gurudutt, Vv; Sint, T; Schneider, Bp; Jones, Wd; Goldstein, Bm; Perra, G; DE MONTIS, A; Loi, G; LA COLLA, P; Grifantini, Mario | Articolo | |
Potent and selective inhibitors of human immunodeficiency virus protease structurally related to L-694,746. | 1-gen-1998 | Franchetti, Palmarisa; Perlini, P; ABU SHEIKHA, G; Cappellacci, Loredana; Grifantini, Mario; Loi, Ag; DE MONTIS, A; Pani, A; Marongiu, Me; LA COLLA, P. | Articolo | |
2'-C-Methyl analogues of selective adenosine receptor agonists: synthesis and binding studies. | 1-gen-1998 | Franchetti, Palmarisa; Cappellacci, Loredana; Marchetti, S; Trincavelli, L; Martini, C; Mazzoni, Mr; Lucacchini, A; Grifantini, Mario | Articolo | |
Isosteric Analogues of Nicotinamide Adenine Dinucleotide Derived from Furanfurin, Thiophenfurin, and Selenophenfurin as Mammalian Inosine Monophosphate dehydrogenase (Type I and II) Inhibitors | 1-gen-1998 | Franchetti, Palmarisa; Cappellacci, Loredana; Perlini, P.; Jayaram, H. N.; Butler, A.; Schneider, B. P.; Collart, F. R.; Huberman, E.; Grifantini, Mario | Articolo | |
Labelling of A1 and A3 adenosine receptors with the new selective A1 agonist 2'-Me-CCPA | 1-gen-1998 | Amenta, Francesco; P., Barili; Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario | Poster atto convegno su rivista | |
Structure-activity relationships of tiazofurin analogs: synthesis and computational studies of 4'-thio derivatives of thiophenfurin and furanfurin | 1-gen-1999 | Franchetti, Palmarisa; Marchetti, S; Cappellacci, Loredana; Grifantini, Mario; Goldstein, Bm; Dukhan, D; Barascut, J. L.; Imbach, J. L. | Articolo | |
Selective targeting to macrophages of a new homodinucleotide active aginst human immunodeficiency virus and herpes simplex virus | 1-gen-1999 | Rossi, L; Serafini, S; Cappellacci, Loredana; Balestra, E; Brandi, G; Schiavano Giuditta, F; Franchetti, Palmarisa; Grifantini, Mario; Perno, C. F.; Magnani, M. | Poster atto convegno su rivista | |
Red Blood cells as drug delivery system for antiviral nucleotide analogues | 1-gen-1999 | Rossi, L.; Serafini, S.; Brandi, G.; Magnani, M.; Balestra, E.; Perno, C. F.; Cappellacci, Loredana; Franchetti, Palmarisa | Poster atto convegno su rivista | |
Synthesis, Conformational Analysis, and Biological Activity of C-Thioribonucleosides Related to Tiazofurin | 1-gen-2000 | Franchetti, Palmarisa; Marchetti, S.; Cappellacci, Loredana; Jayaram, H. N.; Yalowitz, J. A.; Goldstein, B. M.; Barascut, J. L.; Dukhan, D.; Imbach, J. L.; Grifantini, Mario | Articolo | |
A new acyclic heterodinucleotide active against Human Immunodeficiency Virus and Herpes Simplex Virus | 1-gen-2000 | Franchetti, Palmarisa; ABU SHEIKHA, G.; Cappellacci, Loredana; Marchetti, S.; Grifantini, Mario; Balestra, E.; Perno, C. F.; Benatti, U.; Brandi, G.; Rossi, L; Magnani, M. | Articolo | |
C-Nucleoside Analogues of Furanfurin as Ligands to A(1) Adenosine Receptors | 1-gen-2000 | Franchetti, Palmarisa; Cappellacci, Loredana; Marchetti, S.; Martini, C.; Costa, B.; Varani, K.; Borea, P. A.; Grifantini, Mario | Articolo | |
Inhibition of human immunodeficency virus replication in macrophages by red blood cell-mediated delivery of a heterodinucleotide of azidothymidine and 9-(R)-2-(phosphonomethoxypropyl)adenine. | 1-gen-2001 | Franchetti, Palmarisa; Rossi, L; Cappellacci, Loredana; Pasqualini, M; Grifantini, Mario; Balestra, E; Forbici, F; Perno, C. F.; Serafini, S; Magnani, M. | Articolo | |
Erythrocyte-mediated delivery of a new homodinucleotide active against human immunodeficiency virus and herpes simplex virus | 1-gen-2001 | Rossi, L; Serafini, S; Cappellacci, Loredana; Balestra, E; Brandi, G; Schiavano, G. F.; Franchetti, Palmarisa; Grifantini, Mario; Perno, C. F.; Magnani, M. | Articolo | |
A new C-Nucleoside Analogue of Tiazofurin: Synthesis and Biological Evaluation of 2-beta-D-Ribofuranosylimidazole-4-carboxamide (Imidazofurin) | 1-gen-2001 | Franchetti, Palmarisa; Marchetti, S.; Cappellacci, Loredana; Yalowitz, J. A.; Jayaram, H. N.; Goldstein, B. M.; Grifantini, Mario | Articolo | |
Pharmacokinetic and antiretroviral activity in mice of oral [P1,P2-bis[2-(adenin-9-yl)ethoxymethyl]phosphonate], a prodrug of 9-(2-phosphonylmethoxyethyl)adenine | 1-gen-2002 | Rossi, L.; Dominici, S.; Serafini, S.; Casabianca, A.; Cerasi, A.; Chiarantini, L.; Celeste, A. G.; Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Magnani, M. | Articolo |
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