Sfoglia per Autore
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models
1998-01-01 Pigini, Maria; Bousquet, P.; Brasili, L.; Carrieri, A.; Cavagna, R.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Leonetti, F.; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A.
Binding of Tracizolines to the Imidazoline Receptor. Role of Lipophilicity in Quantitative Structure-Activity Relationship Models.
1999-01-01 Pigini, Maria; Bousquet, P; Brasili, L; Carrieri, A; Dontenwill, M; Gentili, Francesco; Giannella, Mario; Leonetti, F; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A.
2-(2-Phenylcyclopropyl)imidazolines: Reversed Enantioselective Interaction at I1 and I2 Imidazoline Receptors
1999-01-01 Quaglia, Wilma; Bousquet, P.; Pigini, Maria; Carotti, A.; Carrieri, A.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Maranca, F.; Piergentili, Alessandro; Brasili, L.
Hyperphagic effect of novel compounds with high affinity for imidazoline I2 binding sites
2000-01-01 Polidori, Carlo; Gentili, Francesco; Pigini, Maria; Quaglia, Wilma; Panocka, I.; Massi, M.
Structure-activity relationship at alpha-adrenergic receptors within a series of imidazoline analogues of cirazoline
2000-01-01 Pigini, Maria; Quaglia, Wilma; Gentili, Francesco; Marucci, Gabriella; Cantalamessa, F.; Franchini, S.; Sorbi, C.; Brasili, L.
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes
2002-01-01 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C.
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives
2002-01-01 Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma
Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole
2002-01-01 Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria
14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry
2003-01-01 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Imidazoline binding sites (IBS) profile modulation: Key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues
2003-01-01 Gentili, Francesco; Bousquet, P.; Brasili, L.; Dontenwill, M.; Feldman, J.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine
2003-01-01 Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands
2004-01-01 Nicolotti, O.; Carotti, A.; Carrieri, A.; Pigini, Maria; Gentili, Francesco; Brasili, L.; Giannella, Mario; Quaglia, Wilma; Piergentili, Alessandro; Bousquet, P.; Dontenwill, M.
alpha(2)-Adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha2C-subtype
2004-01-01 Gentili, Francesco; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Vesprini, C.; Crassous, A.; Paris, H.; Carrieri, A.
Structure-activity relationships in 1,4-benzodioxan-related compounds. 8.(1) {2-[2-(4 chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha1D- and alpha1B-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation
2005-01-01 Quaglia, Wilma; Santoni, Giorgio; Pigini, Maria; Piergentili, Alessandro; Gentili, Francesco; Buccioni, Michela; Mosca, Michela; Lucciarini, Roberta; Amantini, Consuelo; Nabissi, Massimo; Ballarini, P; Poggesi, E; Leonardi, A; Ballarini, Patrizia
Rational design of new alpha(2)-adrenoreceptor agonists
2007-01-01 Gentili, Francesco; Cardinaletti, C.; Carrieri, A.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, Maria
16th Camerino-Noordwijkerhout Symposium - An Overview of Receptor Chemistry
2007-01-01 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Alpha(2)-Adrenoreceptors Profile Modulation. 3. (R)-(+)-m-Nitrobiphenyline, a New Efficient and alpha(2C)-Subtype Selective Agonist.
2007-01-01 Crassous, P. A.; Cardinaletti, C; Carrieri, A; Bruni, B; DI VAIRA, M; Gentili, Francesco; Ghelfi, F; Giannella, Mario; Paris, H; Piergentili, Alessandro; Quaglia, Wilma; Schaak, S; Vesprini, C; Pigini, Maria
Agonists and antagonists targeting the different alpha(2)-adrenoceptor subtypes
2007-01-01 Gentili, Francesco; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario
Solution-phase synthesis of ICG-001, a beta-turn peptidomimetic molecule inhibitor of beta-catenin-Tcf-mediated transcription
2007-01-01 Piergentili, Alessandro; DEL BELLO, Fabio; Gentili, Francesco; Giannella, Mario; Quaglia, Wilma; Vesprini, Christian; Thomas, R. J.; Robertson, G. M.
alpha(2)-adrenoreceptors profile modulation. 4. From antagonist, to agonist behavior
2008-01-01 Gentili, Francesco; Cardinaletti, C.; Vesprini, C.; Carrieri, A.; Ghelfi, F.; Farande, A.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Laurila, J. M.; Huhtinen, A.; Scheinin, M.; Pigini, Maria
| Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
|---|---|---|---|---|
| Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models | 1-gen-1998 | Pigini, Maria; Bousquet, P.; Brasili, L.; Carrieri, A.; Cavagna, R.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Leonetti, F.; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A. | Articolo | |
| Binding of Tracizolines to the Imidazoline Receptor. Role of Lipophilicity in Quantitative Structure-Activity Relationship Models. | 1-gen-1999 | Pigini, Maria; Bousquet, P; Brasili, L; Carrieri, A; Dontenwill, M; Gentili, Francesco; Giannella, Mario; Leonetti, F; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A. | Articolo | |
| 2-(2-Phenylcyclopropyl)imidazolines: Reversed Enantioselective Interaction at I1 and I2 Imidazoline Receptors | 1-gen-1999 | Quaglia, Wilma; Bousquet, P.; Pigini, Maria; Carotti, A.; Carrieri, A.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Maranca, F.; Piergentili, Alessandro; Brasili, L. | Articolo | |
| Hyperphagic effect of novel compounds with high affinity for imidazoline I2 binding sites | 1-gen-2000 | Polidori, Carlo; Gentili, Francesco; Pigini, Maria; Quaglia, Wilma; Panocka, I.; Massi, M. | Articolo | |
| Structure-activity relationship at alpha-adrenergic receptors within a series of imidazoline analogues of cirazoline | 1-gen-2000 | Pigini, Maria; Quaglia, Wilma; Gentili, Francesco; Marucci, Gabriella; Cantalamessa, F.; Franchini, S.; Sorbi, C.; Brasili, L. | Articolo | |
| Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes | 1-gen-2002 | Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C. | Articolo | |
| Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives | 1-gen-2002 | Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma | Articolo | |
| Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole | 1-gen-2002 | Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria | Articolo | |
| 14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry | 1-gen-2003 | Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | ORGANIZZAZIONE DI EVENTI | |
| Imidazoline binding sites (IBS) profile modulation: Key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues | 1-gen-2003 | Gentili, Francesco; Bousquet, P.; Brasili, L.; Dontenwill, M.; Feldman, J.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | Articolo | |
| Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine | 1-gen-2003 | Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario | Articolo | |
| Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands | 1-gen-2004 | Nicolotti, O.; Carotti, A.; Carrieri, A.; Pigini, Maria; Gentili, Francesco; Brasili, L.; Giannella, Mario; Quaglia, Wilma; Piergentili, Alessandro; Bousquet, P.; Dontenwill, M. | Articolo | |
| alpha(2)-Adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha2C-subtype | 1-gen-2004 | Gentili, Francesco; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Vesprini, C.; Crassous, A.; Paris, H.; Carrieri, A. | Articolo | |
| Structure-activity relationships in 1,4-benzodioxan-related compounds. 8.(1) {2-[2-(4 chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha1D- and alpha1B-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation | 1-gen-2005 | Quaglia, Wilma; Santoni, Giorgio; Pigini, Maria; Piergentili, Alessandro; Gentili, Francesco; Buccioni, Michela; Mosca, Michela; Lucciarini, Roberta; Amantini, Consuelo; Nabissi, Massimo; Ballarini, P; Poggesi, E; Leonardi, A; Ballarini, Patrizia | Articolo | |
| Rational design of new alpha(2)-adrenoreceptor agonists | 1-gen-2007 | Gentili, Francesco; Cardinaletti, C.; Carrieri, A.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, Maria | Articolo | |
| 16th Camerino-Noordwijkerhout Symposium - An Overview of Receptor Chemistry | 1-gen-2007 | Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | ORGANIZZAZIONE DI EVENTI | |
| Alpha(2)-Adrenoreceptors Profile Modulation. 3. (R)-(+)-m-Nitrobiphenyline, a New Efficient and alpha(2C)-Subtype Selective Agonist. | 1-gen-2007 | Crassous, P. A.; Cardinaletti, C; Carrieri, A; Bruni, B; DI VAIRA, M; Gentili, Francesco; Ghelfi, F; Giannella, Mario; Paris, H; Piergentili, Alessandro; Quaglia, Wilma; Schaak, S; Vesprini, C; Pigini, Maria | Articolo | |
| Agonists and antagonists targeting the different alpha(2)-adrenoceptor subtypes | 1-gen-2007 | Gentili, Francesco; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario | Articolo | |
| Solution-phase synthesis of ICG-001, a beta-turn peptidomimetic molecule inhibitor of beta-catenin-Tcf-mediated transcription | 1-gen-2007 | Piergentili, Alessandro; DEL BELLO, Fabio; Gentili, Francesco; Giannella, Mario; Quaglia, Wilma; Vesprini, Christian; Thomas, R. J.; Robertson, G. M. | Articolo | |
| alpha(2)-adrenoreceptors profile modulation. 4. From antagonist, to agonist behavior | 1-gen-2008 | Gentili, Francesco; Cardinaletti, C.; Vesprini, C.; Carrieri, A.; Ghelfi, F.; Farande, A.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Laurila, J. M.; Huhtinen, A.; Scheinin, M.; Pigini, Maria | Articolo |
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