Sfoglia "1.1 Articolo" per Titolo
1'-Benzyl-3,4-dihydrospiro[2H-1-benzothiopyran-2,4'-piperidine] (Spipethiane), a potent and highly selective sigma1 lingand
1998-01-01 Quaglia, Wilma; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Brasili, L.; DI TORO, R.; Rossetti, R.; Spampinato, S.; Melchiorre, C.
1,2,4-Benzothiadiazine derivatives as alpha1 and 5-HT1A receptor ligands
2005-01-01 Tait, A; Luppi, A; Franchini, S; Preziosi, E; Parenti, C; Buccioni, Michela; Marucci, Gabriella; Leonardi, A; Poggesi, E; Brasili, L.
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies
2015-01-01 Daniela, Catarzi; Flavia, Varano; Daniela, Poli; Lucia, Squarcialupi; Marco, Betti; Letizia, Trincavelli; Claudia, Martini; DAL BEN, Diego; Thomas, Ajiroghene; Volpini, Rosaria; Vittoria, Colotta
The 1,2,4-Triazolo[4,3-a]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the A2A Receptor Subtype
2017-01-01 Falsini, Matteo; Squarcialupi, Lucia; Catarzi, Daniela; Varano, Flavia; Betti, Marco; DAL BEN, Diego; Marucci, Gabriella; Buccioni, Michela; Volpini, Rosaria; De Vita, Teresa; Cavalli, Andrea; Colotta, Vittoria
1,2-Asymmetric Induction in the TiCl4 Mediated Alkylation of alfa-Methyl-beta-Silyloxy Ketones with Grignard Reagents
1997-01-01 Bartoli, G.; Bosco, M.; Marcantoni, Enrico; Sambri, L.
“1,3 Oxathiolane Muscarinic Ligands Modified at the Cationic Head”.
1994-01-01 Teodori, E; Dei, S; Romanelli, M. N.; Scapecchi, S; Gualtieri, F; Angeli, Piero; Marucci, Gabriella; Matucci, R.
1,3-Dinitro Alkanes: An Emerging Class of Bidentate Compounds
2014-01-01 Ballini, Roberto; Gabrielli, Serena; Palmieri, Alessandro
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity
2019-01-01 Franchini, Silvia; Sorbi, Claudia; Linciano, Pasquale; Carnevale, Gianluca; Tait, Annalisa; Ronsisvalle, Simone; Buccioni, Michela; Del Bello, Fabio; Cilia, Antonio; Pirona, Lorenza; Denora, Nunzio; Maria Iacobazzi, Rosa; Brasili, Livio
1,3-Dioxolane-based ligands as a novel class of alpha(1)-adrenoceptor antagonists
2003-01-01 Brasili, L.; Sorbi, C.; Franchini, S.; Manicardi, M.; Angeli, Piero; Marucci, Gabriella; Leonardi, A.; Poggesi, E.
1,3-Dioxolane-based ligands as rigid analogues of Naftopidil: structure-affinity/activity relationships at alpha1 and 5-HT1A receptors.
2009-01-01 Sorbi, C.; Franchini, S.; Tait, A.; Prandi, A.; Gallesi, R.; Angeli, Piero; Marucci, Gabriella; Pirona, L.; Poggesi, E.; Brasili, L.
1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: Structure-affinity/activity relationship at α1-adrenoceptor subtypes and at 5-HT1A receptors.
2010-01-01 Franchini, S; Prandi, A; Baraldi, A; Sorbi, C; Tait, A; Buccioni, Michela; Marucci, Gabriella; Cilia, A; Pirona, L; Fossa, P; Cichero, E; Brasili, L.
1,3-Dioxolanes from carbonyl compounds over zeolite HSZ-360 as a reusable heterogeneous catalyst
1998-01-01 Ballini, Roberto; Bosica, Giovanna
1,4-Dioxane, a Suitable Scaffold for the Development of Novel M3 Muscarinic Receptor Antagonists
2012-01-01 DEL BELLO, Fabio; Barocelli, E.; Bertoni, S.; Bonifazi, A.; Camalli, M.; Campi, G.; Giannella, Mario; Matucci, R.; Nesi, M.; Pigini, Maria; Quaglia, Wilma; Piergentili, Alessandro
1-[3-(4-Butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1) as a Model for the Rational Design of a Novel Class of Brain Penetrant Ligands with High Affinity and Selectivity for Dopamine D4 Receptor
2018-01-01 Del Bello, Fabio; Bonifazi, Alessandro; Giorgioni, Gianfabio; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Petrelli, Riccardo; Piergentili, Alessandro; Fontana, Stefano; Mammoli, Valerio; Yano, Hideaki; Matucci, Rosanna; Vistoli, Giulio; Quaglia, Wilma
1-Alkoxyamino-2-nitro as Key Building Blocks for a Chemo- and Diastereoselective Synthesis of a New Type of polyfunctionalized N-Alkoxypiperidine
2010-01-01 M. A., Lopez Garcia; I., Maya; J. G., Fernandez Bolagnos; Ballini, Roberto; Bosica, Giovanna
1-Nitroicosane as the Key Building Block for the First Synthesis of Triacontan-11-ol, A New Fatty Alcohol Isolated from Argemone mexicana
2005-01-01 Ballini, Roberto; Fiorini, Dennis; Palmieri, Alessandro
(1-Phenyl-3-methyl-4-acetylpyrazolon-5-ato)rhodium(I) complexes, synthesis, structural and spectroscopical characterization: reactivity of diolefin- and dicarbonyl-rhodium complexes toward N-, P- and O-donors.
1998-01-01 Pettinari, Claudio; F., Accorroni; Cingolani, Augusto; Marchetti, Fabio; A., Cassetta; L., Barba
10 domande a Cristiano Toraldo di Francia
2018-01-01 Romagni, Ludovico; Emili, Anna Rita
10 DOMANDE A FRANCO PURINI
2018-01-01 Romagni, Ludovico; Emili, Anna Rita
10 DOMANDE A PAOLO DESIDERI
2018-01-01 Romagni, Ludovico; Emili, Anna Rita
| Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
|---|---|---|---|---|
| 1'-Benzyl-3,4-dihydrospiro[2H-1-benzothiopyran-2,4'-piperidine] (Spipethiane), a potent and highly selective sigma1 lingand | 1-gen-1998 | Quaglia, Wilma; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Brasili, L.; DI TORO, R.; Rossetti, R.; Spampinato, S.; Melchiorre, C. | Articolo | |
| 1,2,4-Benzothiadiazine derivatives as alpha1 and 5-HT1A receptor ligands | 1-gen-2005 | Tait, A; Luppi, A; Franchini, S; Preziosi, E; Parenti, C; Buccioni, Michela; Marucci, Gabriella; Leonardi, A; Poggesi, E; Brasili, L. | Articolo | |
| 1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies | 1-gen-2015 | Daniela, Catarzi; Flavia, Varano; Daniela, Poli; Lucia, Squarcialupi; Marco, Betti; Letizia, Trincavelli; Claudia, Martini; DAL BEN, Diego; Thomas, Ajiroghene; Volpini, Rosaria; Vittoria, Colotta | Articolo | |
| The 1,2,4-Triazolo[4,3-a]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the A2A Receptor Subtype | 1-gen-2017 | Falsini, Matteo; Squarcialupi, Lucia; Catarzi, Daniela; Varano, Flavia; Betti, Marco; DAL BEN, Diego; Marucci, Gabriella; Buccioni, Michela; Volpini, Rosaria; De Vita, Teresa; Cavalli, Andrea; Colotta, Vittoria | Articolo | |
| 1,2-Asymmetric Induction in the TiCl4 Mediated Alkylation of alfa-Methyl-beta-Silyloxy Ketones with Grignard Reagents | 1-gen-1997 | Bartoli, G.; Bosco, M.; Marcantoni, Enrico; Sambri, L. | Articolo | |
| “1,3 Oxathiolane Muscarinic Ligands Modified at the Cationic Head”. | 1-gen-1994 | Teodori, E; Dei, S; Romanelli, M. N.; Scapecchi, S; Gualtieri, F; Angeli, Piero; Marucci, Gabriella; Matucci, R. | Articolo | |
| 1,3-Dinitro Alkanes: An Emerging Class of Bidentate Compounds | 1-gen-2014 | Ballini, Roberto; Gabrielli, Serena; Palmieri, Alessandro | Articolo | |
| 1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity | 1-gen-2019 | Franchini, Silvia; Sorbi, Claudia; Linciano, Pasquale; Carnevale, Gianluca; Tait, Annalisa; Ronsisvalle, Simone; Buccioni, Michela; Del Bello, Fabio; Cilia, Antonio; Pirona, Lorenza; Denora, Nunzio; Maria Iacobazzi, Rosa; Brasili, Livio | Articolo | |
| 1,3-Dioxolane-based ligands as a novel class of alpha(1)-adrenoceptor antagonists | 1-gen-2003 | Brasili, L.; Sorbi, C.; Franchini, S.; Manicardi, M.; Angeli, Piero; Marucci, Gabriella; Leonardi, A.; Poggesi, E. | Articolo | |
| 1,3-Dioxolane-based ligands as rigid analogues of Naftopidil: structure-affinity/activity relationships at alpha1 and 5-HT1A receptors. | 1-gen-2009 | Sorbi, C.; Franchini, S.; Tait, A.; Prandi, A.; Gallesi, R.; Angeli, Piero; Marucci, Gabriella; Pirona, L.; Poggesi, E.; Brasili, L. | Articolo | |
| 1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: Structure-affinity/activity relationship at α1-adrenoceptor subtypes and at 5-HT1A receptors. | 1-gen-2010 | Franchini, S; Prandi, A; Baraldi, A; Sorbi, C; Tait, A; Buccioni, Michela; Marucci, Gabriella; Cilia, A; Pirona, L; Fossa, P; Cichero, E; Brasili, L. | Articolo | |
| 1,3-Dioxolanes from carbonyl compounds over zeolite HSZ-360 as a reusable heterogeneous catalyst | 1-gen-1998 | Ballini, Roberto; Bosica, Giovanna | Articolo | |
| 1,4-Dioxane, a Suitable Scaffold for the Development of Novel M3 Muscarinic Receptor Antagonists | 1-gen-2012 | DEL BELLO, Fabio; Barocelli, E.; Bertoni, S.; Bonifazi, A.; Camalli, M.; Campi, G.; Giannella, Mario; Matucci, R.; Nesi, M.; Pigini, Maria; Quaglia, Wilma; Piergentili, Alessandro | Articolo | |
| 1-[3-(4-Butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1) as a Model for the Rational Design of a Novel Class of Brain Penetrant Ligands with High Affinity and Selectivity for Dopamine D4 Receptor | 1-gen-2018 | Del Bello, Fabio; Bonifazi, Alessandro; Giorgioni, Gianfabio; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Petrelli, Riccardo; Piergentili, Alessandro; Fontana, Stefano; Mammoli, Valerio; Yano, Hideaki; Matucci, Rosanna; Vistoli, Giulio; Quaglia, Wilma | Articolo | |
| 1-Alkoxyamino-2-nitro as Key Building Blocks for a Chemo- and Diastereoselective Synthesis of a New Type of polyfunctionalized N-Alkoxypiperidine | 1-gen-2010 | M. A., Lopez Garcia; I., Maya; J. G., Fernandez Bolagnos; Ballini, Roberto; Bosica, Giovanna | Articolo | |
| 1-Nitroicosane as the Key Building Block for the First Synthesis of Triacontan-11-ol, A New Fatty Alcohol Isolated from Argemone mexicana | 1-gen-2005 | Ballini, Roberto; Fiorini, Dennis; Palmieri, Alessandro | Articolo | |
| (1-Phenyl-3-methyl-4-acetylpyrazolon-5-ato)rhodium(I) complexes, synthesis, structural and spectroscopical characterization: reactivity of diolefin- and dicarbonyl-rhodium complexes toward N-, P- and O-donors. | 1-gen-1998 | Pettinari, Claudio; F., Accorroni; Cingolani, Augusto; Marchetti, Fabio; A., Cassetta; L., Barba | Articolo | |
| 10 domande a Cristiano Toraldo di Francia | 1-gen-2018 | Romagni, Ludovico; Emili, Anna Rita | Articolo | |
| 10 DOMANDE A FRANCO PURINI | 1-gen-2018 | Romagni, Ludovico; Emili, Anna Rita | Articolo | |
| 10 DOMANDE A PAOLO DESIDERI | 1-gen-2018 | Romagni, Ludovico; Emili, Anna Rita | Articolo |
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