Sfoglia per Autore
1,4-Dioxane ring as a promising template of novel 5-HT1A full agonists
2008-01-01 Giannella, Mario; DEL BELLO, Fabio; A., Farande; A., Leonardi; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
alpha(2)-adrenoreceptors profile modulation. 4. From antagonist, to agonist behavior
2008-01-01 Gentili, Francesco; Cardinaletti, C.; Vesprini, C.; Carrieri, A.; Ghelfi, F.; Farande, A.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Laurila, J. M.; Huhtinen, A.; Scheinin, M.; Pigini, Maria
Structure-activity relationships in 1,4-benzodioxan-related compounds. 9.From 1,4-benzodioxan to 1,4-dioxane ring as a promising template of novel alpha(1D)-adrenoreceptor antagonists, 5-HT1A full agonists, and cytotoxic agents.
2008-01-01 Quaglia, Wilma; Piergentili, Alessandro; DEL BELLO, Fabio; Farande, YOGITA ANIKET; Giannella, Mario; Pigini, Maria; Rafaiani, Giovanni; Carrieri, A; Amantini, Consuelo; Lucciarini, R; Santoni, Giorgio; Poggesi, E; Leonardi, A.
Novel ligands rationally designed for characterizing I2-imidazoline binding sites nature and functions
2008-01-01 Gentili, Francesco; Cardinaletti, Claudia; Vesprini, C.; Ghelfi, Francesca; Farande, ANIKET VIJAYKUMAR; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Mattioli, Laura; Perfumi, Marina Cecilia; Hudson, A.; Pigini, Maria
Rapid novel divergent synthesis and muscarinic agonist profile of all four optical isomers of N,N,N-trimethyl(6-methyl-1,4-dioxan-2-yl)methanaminium iodide.
2008-01-01 Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Buccioni, Michela; Nesi, M; Matucci, R.
Potent muscarinic antagonists bearing 1,4-dioxane scaffold
2009-01-01 DEL BELLO, Fabio; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; R., Matucci; M., Nesi
Enantiomers of 6,6-diphenyl-1,4-dioxane derivatives to highlight stereochemical requirements for selective alpha1D-AR and 5- HT1A receptor recognition
2009-01-01 Y. A., Farande; DEL BELLO, Fabio; Giannella, Mario; A., Leonardi; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Might adrenergic α2C-agonist/α2A-antagonist become a novel therapeutic multitarget tool for morphine chronic treatment of pain?
2009-01-01 Cardinaletti, Claudia; Mattioli, Laura; Ghelfi, Francesca; Giannella, Mario; Perfumi, Marina Cecilia; Nasuti, Cinzia Carla; DEL BELLO, Fabio; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
Molecular determinants in the binding of novel 1,4-benzodioxan-related α1D-adrenergic receptor antagonists: a computational study
2009-01-01 A., Carrieri; Quaglia, Wilma; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; A., Leonardi; F., Fanelli
Properly substituted 1,4-dioxane nucleus favours the selective M3 muscarinic receptor activation
2009-01-01 Piergentili, Alessandro; Quaglia, Wilma; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Barocelli, E.; Bertoni, S.; Matucci, R.; Nesi, M.; Bruni, B.; DI VAIRA, M.
Might Adrenergic alpha2C-agonists/alpha2A-antagonists become novel therapeutic tools for pain treatment with morphine?
2009-01-01 Cardinaletti, Claudia; Mattioli, Laura; Ghelfi, Francesca; DEL BELLO, Fabio; Giannella, Mario; Bruzzone, A.; Paris, H.; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
28th Camerino-Cyprus-Noordwijkerhout Symposium - Trekking through Receptor Chemistry
2010-01-01 Ambrosini, Dario; Angeli, Piero; DEL BELLO, Fabio; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Copresence of 1,4-dioxane and quinuclidine nuclei in the design of novel muscarinic antagonists
2010-01-01 DEL BELLO, Fabio; A., Farande; Y., Farande; Giannella, Mario; Pigini, Maria; Piergentili, Alessandro; Quaglia, Wilma; M., Nesi; R., Matucci
Novel α1-adrenoreceptor antagonists related to openphendioxan: biological evaluation and α1d computational study
2010-01-01 A., Carrieri; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; A., Leonardi; F., Fanelli; Quaglia, Wilma
Aminopyrimidines as inhibitors of the Wnt signalling pathway
2010-01-01 DEL BELLO, Fabio; A., Farande; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; A., Mencini; R., Thomas; M., Varrone; T., Benicchi; G., Benedetti; A., De Robertis; S., Valensin
Enantioselective interactions to improve adrenergic α2C-agonism/α2A-antagonism
2010-01-01 DEL BELLO, Fabio; Mattioli, Laura; A., Farande; Ghelfi, Francesca; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Perfumi, Marina Cecilia; R., Thomas; C., Marchioro; M., Dal Cin; Pigini, Maria
Novel muscarinic antagonists designed on the 1,4-dioxane scaffold
2010-01-01 DEL BELLO, Fabio; A., Farande; Giannella, Mario; Pigini, Maria; Piergentili, Alessandro; Quaglia, Wilma; M., Nesi; R., Matucci
Structure-activity relationships in 1,4-benzodioxan-related compounds. 10. Novel alpha1-adrenoreceptor antagonists related to openphendioxan: synthesis, biological evaluation, and alpha1d computational study
2010-01-01 Carrieri, A.; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Leonardi, A.; Fanelli, F.; Quaglia, Wilma
Fruitful Adrenergic alpha(2C)-Agonism/alpha(2A)-Antagonism Combination to Prevent and Contrast Morphine Tolerance and Dependence
2010-01-01 DEL BELLO, Fabio; Mattioli, Laura; Ghelfi, Francesca; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Cardinaletti, Claudia; Perfumi, Marina Cecilia; Thomas, R. J.; Zanelli, U.; Marchioro, C.; DAL CIN, M.; Pigini, Maria
Novel Highly Potent and Selective σ1 Receptor Antagonists Related to Spipethiane
2010-01-01 Piergentili, Alessandro; Amantini, Consuelo; DEL BELLO, Fabio; Giannella, Mario; Mattioli, Laura; Maura, Palmery; Perfumi, Marina Cecilia; Pigini, Maria; Santoni, Giorgio; Paolo, Tucci; Margherita, Zotti; Quaglia, Wilma
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
1,4-Dioxane ring as a promising template of novel 5-HT1A full agonists | 1-gen-2008 | Giannella, Mario; DEL BELLO, Fabio; A., Farande; A., Leonardi; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | Poster atto convegno su rivista | |
alpha(2)-adrenoreceptors profile modulation. 4. From antagonist, to agonist behavior | 1-gen-2008 | Gentili, Francesco; Cardinaletti, C.; Vesprini, C.; Carrieri, A.; Ghelfi, F.; Farande, A.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Laurila, J. M.; Huhtinen, A.; Scheinin, M.; Pigini, Maria | Articolo | |
Structure-activity relationships in 1,4-benzodioxan-related compounds. 9.From 1,4-benzodioxan to 1,4-dioxane ring as a promising template of novel alpha(1D)-adrenoreceptor antagonists, 5-HT1A full agonists, and cytotoxic agents. | 1-gen-2008 | Quaglia, Wilma; Piergentili, Alessandro; DEL BELLO, Fabio; Farande, YOGITA ANIKET; Giannella, Mario; Pigini, Maria; Rafaiani, Giovanni; Carrieri, A; Amantini, Consuelo; Lucciarini, R; Santoni, Giorgio; Poggesi, E; Leonardi, A. | Articolo | |
Novel ligands rationally designed for characterizing I2-imidazoline binding sites nature and functions | 1-gen-2008 | Gentili, Francesco; Cardinaletti, Claudia; Vesprini, C.; Ghelfi, Francesca; Farande, ANIKET VIJAYKUMAR; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Mattioli, Laura; Perfumi, Marina Cecilia; Hudson, A.; Pigini, Maria | Articolo | |
Rapid novel divergent synthesis and muscarinic agonist profile of all four optical isomers of N,N,N-trimethyl(6-methyl-1,4-dioxan-2-yl)methanaminium iodide. | 1-gen-2008 | Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Buccioni, Michela; Nesi, M; Matucci, R. | Articolo | |
Potent muscarinic antagonists bearing 1,4-dioxane scaffold | 1-gen-2009 | DEL BELLO, Fabio; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; R., Matucci; M., Nesi | Poster atto convegno su volume | |
Enantiomers of 6,6-diphenyl-1,4-dioxane derivatives to highlight stereochemical requirements for selective alpha1D-AR and 5- HT1A receptor recognition | 1-gen-2009 | Y. A., Farande; DEL BELLO, Fabio; Giannella, Mario; A., Leonardi; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | Poster atto convegno su volume | |
Might adrenergic α2C-agonist/α2A-antagonist become a novel therapeutic multitarget tool for morphine chronic treatment of pain? | 1-gen-2009 | Cardinaletti, Claudia; Mattioli, Laura; Ghelfi, Francesca; Giannella, Mario; Perfumi, Marina Cecilia; Nasuti, Cinzia Carla; DEL BELLO, Fabio; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | Poster atto convegno su volume | |
Molecular determinants in the binding of novel 1,4-benzodioxan-related α1D-adrenergic receptor antagonists: a computational study | 1-gen-2009 | A., Carrieri; Quaglia, Wilma; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; A., Leonardi; F., Fanelli | Poster atto convegno su volume | |
Properly substituted 1,4-dioxane nucleus favours the selective M3 muscarinic receptor activation | 1-gen-2009 | Piergentili, Alessandro; Quaglia, Wilma; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Barocelli, E.; Bertoni, S.; Matucci, R.; Nesi, M.; Bruni, B.; DI VAIRA, M. | Articolo | |
Might Adrenergic alpha2C-agonists/alpha2A-antagonists become novel therapeutic tools for pain treatment with morphine? | 1-gen-2009 | Cardinaletti, Claudia; Mattioli, Laura; Ghelfi, Francesca; DEL BELLO, Fabio; Giannella, Mario; Bruzzone, A.; Paris, H.; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | Articolo | |
28th Camerino-Cyprus-Noordwijkerhout Symposium - Trekking through Receptor Chemistry | 1-gen-2010 | Ambrosini, Dario; Angeli, Piero; DEL BELLO, Fabio; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | ORGANIZZAZIONE DI EVENTI | |
Copresence of 1,4-dioxane and quinuclidine nuclei in the design of novel muscarinic antagonists | 1-gen-2010 | DEL BELLO, Fabio; A., Farande; Y., Farande; Giannella, Mario; Pigini, Maria; Piergentili, Alessandro; Quaglia, Wilma; M., Nesi; R., Matucci | Poster atto convegno su rivista | |
Novel α1-adrenoreceptor antagonists related to openphendioxan: biological evaluation and α1d computational study | 1-gen-2010 | A., Carrieri; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; A., Leonardi; F., Fanelli; Quaglia, Wilma | Contributo in atto di convegno su volume | |
Aminopyrimidines as inhibitors of the Wnt signalling pathway | 1-gen-2010 | DEL BELLO, Fabio; A., Farande; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; A., Mencini; R., Thomas; M., Varrone; T., Benicchi; G., Benedetti; A., De Robertis; S., Valensin | Poster atto convegno su volume | |
Enantioselective interactions to improve adrenergic α2C-agonism/α2A-antagonism | 1-gen-2010 | DEL BELLO, Fabio; Mattioli, Laura; A., Farande; Ghelfi, Francesca; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Perfumi, Marina Cecilia; R., Thomas; C., Marchioro; M., Dal Cin; Pigini, Maria | Poster atto convegno su volume | |
Novel muscarinic antagonists designed on the 1,4-dioxane scaffold | 1-gen-2010 | DEL BELLO, Fabio; A., Farande; Giannella, Mario; Pigini, Maria; Piergentili, Alessandro; Quaglia, Wilma; M., Nesi; R., Matucci | Poster atto convegno su volume | |
Structure-activity relationships in 1,4-benzodioxan-related compounds. 10. Novel alpha1-adrenoreceptor antagonists related to openphendioxan: synthesis, biological evaluation, and alpha1d computational study | 1-gen-2010 | Carrieri, A.; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Leonardi, A.; Fanelli, F.; Quaglia, Wilma | Articolo | |
Fruitful Adrenergic alpha(2C)-Agonism/alpha(2A)-Antagonism Combination to Prevent and Contrast Morphine Tolerance and Dependence | 1-gen-2010 | DEL BELLO, Fabio; Mattioli, Laura; Ghelfi, Francesca; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Cardinaletti, Claudia; Perfumi, Marina Cecilia; Thomas, R. J.; Zanelli, U.; Marchioro, C.; DAL CIN, M.; Pigini, Maria | Articolo | |
Novel Highly Potent and Selective σ1 Receptor Antagonists Related to Spipethiane | 1-gen-2010 | Piergentili, Alessandro; Amantini, Consuelo; DEL BELLO, Fabio; Giannella, Mario; Mattioli, Laura; Maura, Palmery; Perfumi, Marina Cecilia; Pigini, Maria; Santoni, Giorgio; Paolo, Tucci; Margherita, Zotti; Quaglia, Wilma | Articolo |
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