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Titolo Data di pubblicazione Autore(i) Tipo File
Coupling of I-1 Imidazoline Receptors to the cAMP Pathway: Studies with a Highly Selective Ligand, Benazoline 1-gen-2000 Greney, H.; Ronde, P.; Magnier, C.; Maranca, F.; Rascente, C.; Quaglia, Wilma; Giannella, Mario; Pigini, Maria; Brasili, L.; Lugnier, C.; Bousquet, P.; Dontenwill, M. Articolo
Homoazanicotine: A structure-affinity study for nicotinic acetylcholine (nACh) receptor binding 1-gen-2002 Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A. Articolo
Deoxamuscaroneoxime Devatives as useful Muscarinic Aginist to Explore the Muscarinic Subsite: Demox, Amodulator of Orthosteric and Allosteric Site at Cardiac Muscarinic M2 Receptors. 1-gen-2002 Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Piergentili, Alessandro; Giannella, Mario; Quaglia, Wilma; Pigini, Maria; Cantalamessa, Franco; Nasuti, Cinzia Carla; Novi, F; Maggio, R; Quasem, A. R.; Spampinato, S. Articolo
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives 1-gen-2002 Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes 1-gen-2002 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C. Articolo
Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole 1-gen-2002 Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria Articolo
Binding of nicotine and homoazanicotine analogues at neuronal nicotinic acetylcholinergic (nACh) receptors 1-gen-2003 Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A. Articolo
Imidazoline binding sites (IBS) profile modulation: Key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues 1-gen-2003 Gentili, Francesco; Bousquet, P.; Brasili, L.; Dontenwill, M.; Feldman, J.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria Articolo
Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine 1-gen-2003 Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario Articolo
14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry 1-gen-2003 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma ORGANIZZAZIONE DI EVENTI
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands 1-gen-2004 Nicolotti, O.; Carotti, A.; Carrieri, A.; Pigini, Maria; Gentili, Francesco; Brasili, L.; Giannella, Mario; Quaglia, Wilma; Piergentili, Alessandro; Bousquet, P.; Dontenwill, M. Articolo
alpha(2)-Adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha2C-subtype 1-gen-2004 Gentili, Francesco; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Vesprini, C.; Crassous, A.; Paris, H.; Carrieri, A. Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 8.(1) {2-[2-(4 chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha1D- and alpha1B-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation 1-gen-2005 Quaglia, Wilma; Santoni, Giorgio; Pigini, Maria; Piergentili, Alessandro; Gentili, Francesco; Buccioni, Michela; Mosca, Michela; Lucciarini, Roberta; Amantini, Consuelo; Nabissi, Massimo; Ballarini, P; Poggesi, E; Leonardi, A; Ballarini, Patrizia Articolo
Solution-phase synthesis of ICG-001, a beta-turn peptidomimetic molecule inhibitor of beta-catenin-Tcf-mediated transcription 1-gen-2007 Piergentili, Alessandro; DEL BELLO, Fabio; Gentili, Francesco; Giannella, Mario; Quaglia, Wilma; Vesprini, Christian; Thomas, R. J.; Robertson, G. M. Articolo
Dioxane and Oxathiane Nuclei: Suitable Substructures for Muscarinic Agonists 1-gen-2007 Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Bruni, B; Buccioni, Michela; Carrieri, A; Ciattini, S. Articolo
Agonists and antagonists targeting the different alpha(2)-adrenoceptor subtypes 1-gen-2007 Gentili, Francesco; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario Articolo
Rational design of new alpha(2)-adrenoreceptor agonists 1-gen-2007 Gentili, Francesco; Cardinaletti, C.; Carrieri, A.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, Maria Articolo
Alpha(2)-Adrenoreceptors Profile Modulation. 3. (R)-(+)-m-Nitrobiphenyline, a New Efficient and alpha(2C)-Subtype Selective Agonist. 1-gen-2007 Crassous, P. A.; Cardinaletti, C; Carrieri, A; Bruni, B; DI VAIRA, M; Gentili, Francesco; Ghelfi, F; Giannella, Mario; Paris, H; Piergentili, Alessandro; Quaglia, Wilma; Schaak, S; Vesprini, C; Pigini, Maria Articolo
16th Camerino-Noordwijkerhout Symposium - An Overview of Receptor Chemistry 1-gen-2007 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma ORGANIZZAZIONE DI EVENTI
1,4-Dioxane ring as a promising template of novel 5-HT1A full agonists 1-gen-2008 Giannella, Mario; DEL BELLO, Fabio; A., Farande; A., Leonardi; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma Poster atto convegno su rivista
Mostrati risultati da 21 a 40 di 106
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