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Mostrati risultati da 26.625 a 26.644 di 30.355
Titolo Data di pubblicazione Autore(i) Tipo File
Structure-Activity Relationships in 1,4-Benzodioxan-Related Compounds. 6. Role of the Dioxane Unit on Selectivity for Alpha1-Adrenoreceptor Subtypes 1-gen-1999 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Poggesi, E.; Leonardi, A.; Melchiorre, C. Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes 1-gen-2002 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C. Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 8.(1) {2-[2-(4 chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha1D- and alpha1B-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation 1-gen-2005 Quaglia, Wilma; Santoni, Giorgio; Pigini, Maria; Piergentili, Alessandro; Gentili, Francesco; Buccioni, Michela; Mosca, Michela; Lucciarini, Roberta; Amantini, Consuelo; Nabissi, Massimo; Ballarini, P; Poggesi, E; Leonardi, A; Ballarini, Patrizia Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 9. From 1,4-benzodioxane to 1,4-dioxane ring as a promising template of novel alpha1D-adrenoreceptor antagonists, 5-HT1A full agonists, and cytotoxic agents. 1-gen-2008 Quaglia, W; Piergentili, A; DEL BELLO, F; Farande, Y; Giannella, M; Pigini, M; Rafaiani, G; Carrieri, A; Amantini, C; Lucciarini, R; Santoni, Giorgio; Poggesi, E; Leonardi, A. Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. 9.From 1,4-benzodioxan to 1,4-dioxane ring as a promising template of novel alpha(1D)-adrenoreceptor antagonists, 5-HT1A full agonists, and cytotoxic agents. 1-gen-2008 Quaglia, Wilma; Piergentili, Alessandro; DEL BELLO, Fabio; Farande, YOGITA ANIKET; Giannella, Mario; Pigini, Maria; Rafaiani, Giovanni; Carrieri, A; Amantini, Consuelo; Lucciarini, R; Santoni, Giorgio; Poggesi, E; Leonardi, A. Articolo
Structure-activity relationships in 1,4-benzodioxan-related compounds. Investigation on the role of the dehydrodioxane ring on alpha1-adrenoreceptor blocking activity 1-gen-1988 Pigini, Maria; Brasili, L.; Giannella, Mario; Giardinà, D.; Gulini, U.; Quaglia, Wilma; Melchiorre, C. Articolo
Structure-Activity Relationships in 2,2-Diphenyl-2-ethylthioacetic Acid Esters: Unexpected Agonist Activity in a Series of Muscarinic Antagonists. 1-gen-2001 Scapecchi, S.; Marucci, Gabriella; Matucci, R.; Angeli, Piero; Bellucci, C.; Buccioni, Michela; Dei, S.; Gualtieri, F.; Manetti, D.; Romanelli, M. N.; Teodori, E. Articolo
Structure-activity relationships in prazosin-related compounds. Effect of replacing a piperazine ring with an alkanediamine moiety on alpha1- adrenoreceptorblocking activity. 1-gen-1989 Giardinà, D.; Brasili, L.; Gregori, M.; Massi, M.; Picchio, M. T.; Quaglia, Wilma; Melchiorre, C. Articolo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine 1-gen-2003 Tumiatti, V; Rosini, M.; Bartolini, M.; Cavalli, A.; Marucci, Gabriella; Andrisano, V.; Angeli, Piero; Banzi, R.; Minarini, A.; Recanatini, M.; Melchiorre, C. Articolo
Structure-activity relationships of adenine and deazaadenine derivatives as ligands for adenine receptors, a new purinergic receptor family 1-gen-2009 Borrmann, T; Abdelrahman, A; Volpini, Rosaria; Lambertucci, Catia; Alksnis, E; Gorzalka, S; Knospe, M; Schiedel, Ac; Cristalli, Gloria; Mueller, Ce Articolo
Structure-activity relationships of adenosine deaminase inhibitors 1-gen-1999 Vittori, Sauro; Camaioni, E; Costanzi, S; Volpini, Rosaria; Lupidi, Giulio; Cristalli, Gloria Articolo
Structure-activity relationships of bisphosphate nucleotide derivatives as P2Y(1) receptor antagonists and partial agonists 1-gen-1999 Nandanan, Erathodiyil; Camaioni, Emidio; Jang, Soo Yeon; Kim, Yong Chul; Cristalli, Gloria; Herdewijn, Piet; Secrist III, John A.; Tiwari, Kamal N.; Mohanram, Arvind; Harden, T. Kendall; Boyer, José L.; Jacobson, Kenneth A. Articolo
Structure-Activity Relationships of Methoctramine-Related Polyamines as Muscular Nicotinic Receptor Noncompetitive Antagonists. 2. Role of Polymethylene Chain Lengths Separating Amine Functions and of Substituents on the Terminal Nitrogen Atoms. 1-gen-2002 Rosini, M.; Bixel, M. G.; Marucci, Gabriella; Budriesi, R.; Krauss, M.; Bolognesi, M. L.; Minarini, A.; Tumiatti, V.; Hucho, F.; Melchiorre, C. Articolo
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure 1-gen-2002 Bolognesi, M.; Bixel, M. G.; Marucci, Gabriella; Bartolini, M.; Krauss, M.; Angeli, Piero; Antonello, A.; Rosini, M.; Tumiatti, V.; Hucho, F.; Melchiorre, C. Articolo
Structure-activity relationships of tiazofurin analogs: synthesis and computational studies of 4'-thio derivatives of thiophenfurin and furanfurin 1-gen-1999 Franchetti, Palmarisa; Marchetti, S; Cappellacci, Loredana; Grifantini, Mario; Goldstein, Bm; Dukhan, D; Barascut, J. L.; Imbach, J. L. Articolo
Structure-Activity Relatioships Among Novel Phenoxybenzamine-Related Beta-Chloroethylamines. 1-gen-2002 Giardina', Dario; Crucianelli, M; Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Gulini, Ugo; Sagratini, Gianni; Melchiorre, C. Articolo
Structure-affinity relathionships of 5'-carbamoyl- and 5'-thionocarbamoyl derivatives of the A1 selective adenosine receptor agonist 2'-MeCCPA as partial A1 agonists 1-gen-2005 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; B., Costa; C., Martini; A., Lavecchia; Kn, Klotz; Grifantini, Mario Poster atto convegno su rivista
Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α<alpha>1 and 5-HT1A receptors 1-gen-2014 Franchini, Silvia; Battisti, Umberto M; Baraldi, Annamaria; Prandi, Adolfo; Fossa, Paola; Cichero, Elena; Tait, Annalisa; Sorbi, Claudia; Marucci, Gabriella; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio Articolo
Structure-Based Design, Synthesis and in vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists 1-gen-2018 Petrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; DEL BELLO, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana Articolo
Structure-Based Optimization of Coumarin hA3 Adenosine Receptor Antagonists 1-gen-2020 Matos, M. J.; Vilar, S.; Vazquez-Rodriguez, S.; Kachler, S.; Klotz, K. -N.; Buccioni, M.; Delogu, G.; Santana, L.; Uriarte, E.; Borges, F. Articolo
Mostrati risultati da 26.625 a 26.644 di 30.355
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