Sfoglia per Autore
Chain-lengthened and imidazoline analogues of nicotine
2000-01-01 Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A.
Synthesis, molecular modeling, and pharmacological testing of bis-quinolinium cyclophanes: Potent, non-peptidic blockers of the apamin-sensitive Ca2+-activated K+ channel
2000-01-01 CAMPOS ROSA, J.; Galanakis, D.; Piergentili, Alessandro; Bhandari, K.; Ganellin, C. R.; Dunn, P. M.; Jenkinson, D. H.
Deoxamuscaroneoxime Devatives as useful Muscarinic Aginist to Explore the Muscarinic Subsite: Demox, Amodulator of Orthosteric and Allosteric Site at Cardiac Muscarinic M2 Receptors.
2002-01-01 Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Piergentili, Alessandro; Giannella, Mario; Quaglia, Wilma; Pigini, Maria; Cantalamessa, Franco; Nasuti, Cinzia Carla; Novi, F; Maggio, R; Quasem, A. R.; Spampinato, S.
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes
2002-01-01 Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C.
Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives
2002-01-01 Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma
Homoazanicotine: A structure-affinity study for nicotinic acetylcholine (nACh) receptor binding
2002-01-01 Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A.
Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole
2002-01-01 Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria
Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine
2003-01-01 Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario
14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry
2003-01-01 Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Imidazoline binding sites (IBS) profile modulation: Key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues
2003-01-01 Gentili, Francesco; Bousquet, P.; Brasili, L.; Dontenwill, M.; Feldman, J.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
Binding of nicotine and homoazanicotine analogues at neuronal nicotinic acetylcholinergic (nACh) receptors
2003-01-01 Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A.
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands
2004-01-01 Nicolotti, O.; Carotti, A.; Carrieri, A.; Pigini, Maria; Gentili, Francesco; Brasili, L.; Giannella, Mario; Quaglia, Wilma; Piergentili, Alessandro; Bousquet, P.; Dontenwill, M.
alpha(2)-Adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha2C-subtype
2004-01-01 Gentili, Francesco; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Vesprini, C.; Crassous, A.; Paris, H.; Carrieri, A.
Rational design of the new antihypertensive I1-receptor ligand 2-(2-Biphenyl-2-yl-1-methyl-ethyl)-4,5-dihydro-1H-imidazole
2005-01-01 Gentili, F.; Bousquet, P.; Carrieri, A.; Feldman, J.; Ghelfi, F.; Giannella, M.; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, M.
Synthesis and antimuscarinic activity of derivatives of 2-substituted-1,3-dioxolanes
2005-01-01 Marucci, Gabriella; Angeli, Piero; Brasili, L.; Giardina', Dario; Gulini, U.; Piergentili, Alessandro; Sagratini, Gianni; Franchini, S.
Structure-activity relationships in 1,4-benzodioxan-related compounds. 8.(1) {2-[2-(4 chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha1D- and alpha1B-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation
2005-01-01 Quaglia, Wilma; Santoni, Giorgio; Pigini, Maria; Piergentili, Alessandro; Gentili, Francesco; Buccioni, Michela; Mosca, Michela; Lucciarini, Roberta; Amantini, Consuelo; Nabissi, Massimo; Ballarini, P; Poggesi, E; Leonardi, A; Ballarini, Patrizia
Solution-phase synthesis of ICG-001, a beta-turn peptidomimetic molecule inhibitor of beta-catenin-Tcf-mediated transcription
2007-01-01 Piergentili, Alessandro; DEL BELLO, Fabio; Gentili, Francesco; Giannella, Mario; Quaglia, Wilma; Vesprini, Christian; Thomas, R. J.; Robertson, G. M.
Dioxane and Oxathiane Nuclei: Suitable Substructures for Muscarinic Agonists
2007-01-01 Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Bruni, B; Buccioni, Michela; Carrieri, A; Ciattini, S.
Alpha(2)-Adrenoreceptors Profile Modulation. 3. (R)-(+)-m-Nitrobiphenyline, a New Efficient and alpha(2C)-Subtype Selective Agonist.
2007-01-01 Crassous, P. A.; Cardinaletti, C; Carrieri, A; Bruni, B; DI VAIRA, M; Gentili, Francesco; Ghelfi, F; Giannella, Mario; Paris, H; Piergentili, Alessandro; Quaglia, Wilma; Schaak, S; Vesprini, C; Pigini, Maria
Rational design of new alpha(2)-adrenoreceptor agonists
2007-01-01 Gentili, Francesco; Cardinaletti, C.; Carrieri, A.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, Maria
| Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
|---|---|---|---|---|
| Chain-lengthened and imidazoline analogues of nicotine | 1-gen-2000 | Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A. | Articolo | |
| Synthesis, molecular modeling, and pharmacological testing of bis-quinolinium cyclophanes: Potent, non-peptidic blockers of the apamin-sensitive Ca2+-activated K+ channel | 1-gen-2000 | CAMPOS ROSA, J.; Galanakis, D.; Piergentili, Alessandro; Bhandari, K.; Ganellin, C. R.; Dunn, P. M.; Jenkinson, D. H. | Articolo | |
| Deoxamuscaroneoxime Devatives as useful Muscarinic Aginist to Explore the Muscarinic Subsite: Demox, Amodulator of Orthosteric and Allosteric Site at Cardiac Muscarinic M2 Receptors. | 1-gen-2002 | Angeli, Piero; Marucci, Gabriella; Buccioni, Michela; Piergentili, Alessandro; Giannella, Mario; Quaglia, Wilma; Pigini, Maria; Cantalamessa, Franco; Nasuti, Cinzia Carla; Novi, F; Maggio, R; Quasem, A. R.; Spampinato, S. | Articolo | |
| Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes | 1-gen-2002 | Quaglia, Wilma; Pigini, Maria; Piergentili, Alessandro; Giannella, Mario; Gentili, Francesco; Marucci, Gabriella; Carrieri, A.; Carotti, A.; Poggesi, E.; Leonardi, A.; Melchiorre, C. | Articolo | |
| Design, synthesis and muscarinic activity of deoxamuscarine-related derivatives | 1-gen-2002 | Piergentili, Alessandro; Angeli, Piero; Gagliardi, Roberto; Gentili, Francesco; Giannella, Mario; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma | Articolo | |
| Homoazanicotine: A structure-affinity study for nicotinic acetylcholine (nACh) receptor binding | 1-gen-2002 | Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A. | Articolo | |
| Alpha(2)-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole | 1-gen-2002 | Gentili, Francesco; Bousquet, P.; Brasili, L.; Caretto, M.; Carrieri, A.; Dontenwill, M.; Giannella, Mario; Marucci, Gabriella; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Rascente, C.; Pigini, Maria | Articolo | |
| Muscarinic subtypes profile modulation within a series of new antagonists, bridged bicyclic derivatives of 2,2-diphenyl-[1,3]-dioxolan-4-ylmethyl-dimethylamine | 1-gen-2003 | Piergentili, Alessandro; Gentili, Francesco; Ghelfi, F.; Marucci, Gabriella; Pigini, Maria; Quaglia, Wilma; Giannella, Mario | Articolo | |
| 14th Camerino-Noordwijkerhout Symposium - Ongoing Progress in Receptor Chemistry | 1-gen-2003 | Angeli, Piero; Gentili, Francesco; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Gulini, Ugo; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | ORGANIZZAZIONE DI EVENTI | |
| Imidazoline binding sites (IBS) profile modulation: Key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues | 1-gen-2003 | Gentili, Francesco; Bousquet, P.; Brasili, L.; Dontenwill, M.; Feldman, J.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | Articolo | |
| Binding of nicotine and homoazanicotine analogues at neuronal nicotinic acetylcholinergic (nACh) receptors | 1-gen-2003 | Ferretti, G.; Dukat, M.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Damaj, M. I.; Martin, B. R.; Glennon, R. A. | Articolo | |
| Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands | 1-gen-2004 | Nicolotti, O.; Carotti, A.; Carrieri, A.; Pigini, Maria; Gentili, Francesco; Brasili, L.; Giannella, Mario; Quaglia, Wilma; Piergentili, Alessandro; Bousquet, P.; Dontenwill, M. | Articolo | |
| alpha(2)-Adrenoreceptors profile modulation. 2. Biphenyline analogues as tools for selective activation of the alpha2C-subtype | 1-gen-2004 | Gentili, Francesco; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Vesprini, C.; Crassous, A.; Paris, H.; Carrieri, A. | Articolo | |
| Rational design of the new antihypertensive I1-receptor ligand 2-(2-Biphenyl-2-yl-1-methyl-ethyl)-4,5-dihydro-1H-imidazole | 1-gen-2005 | Gentili, F.; Bousquet, P.; Carrieri, A.; Feldman, J.; Ghelfi, F.; Giannella, M.; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, M. | Articolo | |
| Synthesis and antimuscarinic activity of derivatives of 2-substituted-1,3-dioxolanes | 1-gen-2005 | Marucci, Gabriella; Angeli, Piero; Brasili, L.; Giardina', Dario; Gulini, U.; Piergentili, Alessandro; Sagratini, Gianni; Franchini, S. | Articolo | |
| Structure-activity relationships in 1,4-benzodioxan-related compounds. 8.(1) {2-[2-(4 chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha1D- and alpha1B-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation | 1-gen-2005 | Quaglia, Wilma; Santoni, Giorgio; Pigini, Maria; Piergentili, Alessandro; Gentili, Francesco; Buccioni, Michela; Mosca, Michela; Lucciarini, Roberta; Amantini, Consuelo; Nabissi, Massimo; Ballarini, P; Poggesi, E; Leonardi, A; Ballarini, Patrizia | Articolo | |
| Solution-phase synthesis of ICG-001, a beta-turn peptidomimetic molecule inhibitor of beta-catenin-Tcf-mediated transcription | 1-gen-2007 | Piergentili, Alessandro; DEL BELLO, Fabio; Gentili, Francesco; Giannella, Mario; Quaglia, Wilma; Vesprini, Christian; Thomas, R. J.; Robertson, G. M. | Articolo | |
| Dioxane and Oxathiane Nuclei: Suitable Substructures for Muscarinic Agonists | 1-gen-2007 | Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Bruni, B; Buccioni, Michela; Carrieri, A; Ciattini, S. | Articolo | |
| Alpha(2)-Adrenoreceptors Profile Modulation. 3. (R)-(+)-m-Nitrobiphenyline, a New Efficient and alpha(2C)-Subtype Selective Agonist. | 1-gen-2007 | Crassous, P. A.; Cardinaletti, C; Carrieri, A; Bruni, B; DI VAIRA, M; Gentili, Francesco; Ghelfi, F; Giannella, Mario; Paris, H; Piergentili, Alessandro; Quaglia, Wilma; Schaak, S; Vesprini, C; Pigini, Maria | Articolo | |
| Rational design of new alpha(2)-adrenoreceptor agonists | 1-gen-2007 | Gentili, Francesco; Cardinaletti, C.; Carrieri, A.; Ghelfi, F.; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Vesprini, C.; Pigini, Maria | Articolo |
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