Sfoglia per Autore
2- And 8- alkynyladenosines: conformational studies and docking to human adenosine A(3) receptor can explain their different biological behavior
2003-01-01 Costanzi, S; Lambertucci, Catia; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria
9-ethyladenine derivatives as adenosine receptor antagonists: 2- and 8-substitution results in distinct selectivities
2003-01-01 Klotz, K. N.; Kachler, S; Lambertucci, Catia; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria
2-phenylhydroxypropynyladenosine derivatives as high potent agonists at A(2B) adenosine receptor subtype
2003-01-01 Lambertucci, Catia; Volpini, Rosaria; Costanzi, S; Taffi, S; Vittori, Sauro; Cristalli, Gloria
Purine and deazapurine nucleosides: synthetic approaches, molecular modeling and biological activity
2003-01-01 Cristalli, Gloria; ., COSTANZI S; Lambertucci, Catia; Taffi, S; Vittori, Sauro; Volpini, Rosaria
A(2B) adenosine receptor agonists: synthesis and biological evaluation of 2-phenylhydroxypropynyladenosine and NECA derivatives
2004-01-01 Vittori, Sauro; Costanzi, S; Lambertucci, Catia; Portino, Fr; Taffi, S; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Adenosine receptor agonists:synthesis and binding affinity of 2-(aryl)alkylthioadenosine derivatives
2004-01-01 Volpini, Rosaria; Costanzi, S; Lambertucci, Catia; Portino, Fr; Taffi, S; Vittori, Sauro; Zablocki, Ja; Klotz, K. N.; Cristalli, Gloria
Ring opening reactions: synthesis of AICAR analogs as potential antimetabolite agents
2005-01-01 Costanzi, S; Lambertucci, Catia; Portino, Fr; Volpini, Rosaria; Vittori, Sauro; Cristalli, Gloria
2- And 8-alkynyl-9-ethyladenines: Synthesis and biological activity at human and rat adenosines receptors
2005-01-01 Volpini, Rosaria; Costanzi, S; Lambertucci, Catia; Vittori, Sauro; Martini, C; Trincavelli, Ml; Klotz, K. N.; Cristalli, Gloria
Effects of 5 '-phosphate derivatives of 2-hexynyl adenosine and 2-phenylethynyl adenosine on responses of human platelets mediated by P2Y receptors
2005-01-01 Cristalli, Gloria; Podda, G; Costanzi, S; Lambertucci, Catia; Lecchi, A; Vittori, Sauro; Volpini, Rosaria; Zighetti, M; Cattaneo, M.
A3 adenosine receptors: synthesis and biological evaluation of new potent and selective ligands
2005-01-01 Volpini, R.; Lambertucci, C.; Taffi, Sara; Vittori, S.; Klotz, K. -N.; Cristalli, G.
GPCRs as therapeutic targets: a view on adenosine receptors structure and functions, and molecular modeling support
2005-01-01 DAL BEN, Diego; Lambertucci, Catia; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria
2-substituted 5 '-N-methylcarboxamidoadenosine (MECA) derivatives as A(3) adenosine receptor ligands
2005-01-01 Vittori, Sauro; Volpini, Rosaria; Lambertucci, Catia; Taffi, S; Klotz, K. N.; Cristalli, Gloria
Solid phase synthesis and antiprotozoal evaluation of di- and trisubstituted 5 '-carboxamidoadenosine analogues
2006-01-01 Rodenko, B; Detz, Rj; Pinas, Va; Lambertucci, Catia; Brun, R; Wanner, Mj; Koomen, Gj
Antiviral properties of deazaadenine nucleoside derivatives
2006-01-01 Vittori, Sauro; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria
Molecular modeling study of 2-phenylethynyladenosine (PEAdo) derivatives as highly selective A3 adenosine receptor ligands
2006-01-01 DAL BEN, Diego; Lambertucci, Catia; Taffi, S; Vittori, Sauro; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
New 2,6,9-trisubstituted adenines as adenosine receptor antagonists: a preliminary SAR profile
2007-01-01 Lambertucci, Catia; Cristalli, Gloria; DAL BEN, Diego; Kachare, Dd; Bolcato, C; Klotz, K. N.; Spalluto, G; Volpini, Rosaria
Synthesis and stability studies of 2 ',3 ',5 '-tri-O-acetyl-2-amino(-N-6-cyclopentyl)-1-deazaadenosines
2007-01-01 Vittori, Sauro; Mishra, Rc; DAL BEN, Diego; Kachare, D; Lambertucci, Catia; Volpini, Rosaria; Cristalli, Gloria
N6-methoxy-2-alkynyladenosine derivatives as highly potent and selective ligands at the human A(3) adenosine receptor
2007-01-01 Volpini, Rosaria; DAL BEN, Diego; Lambertucci, Catia; Taffi, S; Vittori, Sauro; Klotz, K. N.; Cristalli, Gloria
Synthesis and evaluation of hexitol nucleoside congeners as ambiguous nucleosides
2007-01-01 Lambertucci, Catia; Schepers, G; Cristalli, Gloria; Herdewijn, P; VAN AERSCHOT, A.
Highlights on the development of A(2A) adenosine receptor agonists and antagonists
2007-01-01 Cristalli, Gloria; Cacciari, B; DAL BEN, Diego; Lambertucci, Catia; Moro, S; Spalluto, G; Volpini, Rosaria
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
2- And 8- alkynyladenosines: conformational studies and docking to human adenosine A(3) receptor can explain their different biological behavior | 1-gen-2003 | Costanzi, S; Lambertucci, Catia; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
9-ethyladenine derivatives as adenosine receptor antagonists: 2- and 8-substitution results in distinct selectivities | 1-gen-2003 | Klotz, K. N.; Kachler, S; Lambertucci, Catia; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
2-phenylhydroxypropynyladenosine derivatives as high potent agonists at A(2B) adenosine receptor subtype | 1-gen-2003 | Lambertucci, Catia; Volpini, Rosaria; Costanzi, S; Taffi, S; Vittori, Sauro; Cristalli, Gloria | Articolo | |
Purine and deazapurine nucleosides: synthetic approaches, molecular modeling and biological activity | 1-gen-2003 | Cristalli, Gloria; ., COSTANZI S; Lambertucci, Catia; Taffi, S; Vittori, Sauro; Volpini, Rosaria | Articolo | |
A(2B) adenosine receptor agonists: synthesis and biological evaluation of 2-phenylhydroxypropynyladenosine and NECA derivatives | 1-gen-2004 | Vittori, Sauro; Costanzi, S; Lambertucci, Catia; Portino, Fr; Taffi, S; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Adenosine receptor agonists:synthesis and binding affinity of 2-(aryl)alkylthioadenosine derivatives | 1-gen-2004 | Volpini, Rosaria; Costanzi, S; Lambertucci, Catia; Portino, Fr; Taffi, S; Vittori, Sauro; Zablocki, Ja; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Ring opening reactions: synthesis of AICAR analogs as potential antimetabolite agents | 1-gen-2005 | Costanzi, S; Lambertucci, Catia; Portino, Fr; Volpini, Rosaria; Vittori, Sauro; Cristalli, Gloria | Articolo | |
2- And 8-alkynyl-9-ethyladenines: Synthesis and biological activity at human and rat adenosines receptors | 1-gen-2005 | Volpini, Rosaria; Costanzi, S; Lambertucci, Catia; Vittori, Sauro; Martini, C; Trincavelli, Ml; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Effects of 5 '-phosphate derivatives of 2-hexynyl adenosine and 2-phenylethynyl adenosine on responses of human platelets mediated by P2Y receptors | 1-gen-2005 | Cristalli, Gloria; Podda, G; Costanzi, S; Lambertucci, Catia; Lecchi, A; Vittori, Sauro; Volpini, Rosaria; Zighetti, M; Cattaneo, M. | Articolo | |
A3 adenosine receptors: synthesis and biological evaluation of new potent and selective ligands | 1-gen-2005 | Volpini, R.; Lambertucci, C.; Taffi, Sara; Vittori, S.; Klotz, K. -N.; Cristalli, G. | Contributo in atto di convegno su volume | |
GPCRs as therapeutic targets: a view on adenosine receptors structure and functions, and molecular modeling support | 1-gen-2005 | DAL BEN, Diego; Lambertucci, Catia; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
2-substituted 5 '-N-methylcarboxamidoadenosine (MECA) derivatives as A(3) adenosine receptor ligands | 1-gen-2005 | Vittori, Sauro; Volpini, Rosaria; Lambertucci, Catia; Taffi, S; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Solid phase synthesis and antiprotozoal evaluation of di- and trisubstituted 5 '-carboxamidoadenosine analogues | 1-gen-2006 | Rodenko, B; Detz, Rj; Pinas, Va; Lambertucci, Catia; Brun, R; Wanner, Mj; Koomen, Gj | Articolo | |
Antiviral properties of deazaadenine nucleoside derivatives | 1-gen-2006 | Vittori, Sauro; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Molecular modeling study of 2-phenylethynyladenosine (PEAdo) derivatives as highly selective A3 adenosine receptor ligands | 1-gen-2006 | DAL BEN, Diego; Lambertucci, Catia; Taffi, S; Vittori, Sauro; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Articolo | |
New 2,6,9-trisubstituted adenines as adenosine receptor antagonists: a preliminary SAR profile | 1-gen-2007 | Lambertucci, Catia; Cristalli, Gloria; DAL BEN, Diego; Kachare, Dd; Bolcato, C; Klotz, K. N.; Spalluto, G; Volpini, Rosaria | Articolo | |
Synthesis and stability studies of 2 ',3 ',5 '-tri-O-acetyl-2-amino(-N-6-cyclopentyl)-1-deazaadenosines | 1-gen-2007 | Vittori, Sauro; Mishra, Rc; DAL BEN, Diego; Kachare, D; Lambertucci, Catia; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
N6-methoxy-2-alkynyladenosine derivatives as highly potent and selective ligands at the human A(3) adenosine receptor | 1-gen-2007 | Volpini, Rosaria; DAL BEN, Diego; Lambertucci, Catia; Taffi, S; Vittori, Sauro; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Synthesis and evaluation of hexitol nucleoside congeners as ambiguous nucleosides | 1-gen-2007 | Lambertucci, Catia; Schepers, G; Cristalli, Gloria; Herdewijn, P; VAN AERSCHOT, A. | Articolo | |
Highlights on the development of A(2A) adenosine receptor agonists and antagonists | 1-gen-2007 | Cristalli, Gloria; Cacciari, B; DAL BEN, Diego; Lambertucci, Catia; Moro, S; Spalluto, G; Volpini, Rosaria | Articolo |
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