Sfoglia per Autore
Synthesis and alpha1-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin
2007-01-01 Sagratini, Gianni; Angeli, Piero; Buccioni, Michela; Gulini, Ugo; Marucci, Gabriella; Melchiorre, C; Leonardi, A; Poggesi, E; Giardina', Dario
Dioxane and Oxathiane Nuclei: Suitable Substructures for Muscarinic Agonists
2007-01-01 Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Bruni, B; Buccioni, Michela; Carrieri, A; Ciattini, S.
Synthesis, affinity profile, and functional activity of muscarinic antagonists with a 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine structure
2007-01-01 Dei, S.; Bellucci, C.; Buccioni, Michela; Ferraroni, M.; Guandalini, L.; Manetti, D.; Martini, E.; Marucci, Gabriella; Matucci, R.; Nesi, M.; Romanelli, M. N.; Scapecchi, S.; Teodori, E.
Muscarinic antagonists with multiple stereocenters: Synthesis, affinity profile and functional activity of isomeric 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl) pyrrolidine sulfoxide derivatives
2008-01-01 Dei, S.; Bellucci, C.; Buccioni, Michela; Ferraroni, M.; Guandalini, L.; Manetti, D.; Marucci, Gabriella; Matucci, R.; Nesi, M.; Romanelli, M. N.; Scapecchi, S.; Teodori, E.
Synthesis and pharmacological characterization of chiral pyrrolidinylfuran derivatives: The discovery of new functionally selective muscarinic agonists
2008-01-01 Scapecchi, S.; Nesi, M.; Matucci, R.; Bellucci, C.; Buccioni, Michela; Dei, S.; Guandalini, L.; Manetti, D.; Martini, E.; Marucci, Gabriella; Romanelli, M. N.; Teodori, E.; Cirilli, R.
Levels of polychlorinated biphenyls in fish and shellfish from the Adriatic Sea
2008-01-01 Sagratini, Gianni; Buccioni, Michela; Ciccarelli, C.; Conti, Paolo; Cristalli, Gloria; Giardina', Dario; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Vittori, Sauro
In vitro metabolism studies of new adenosine A(2A) receptor antagonists
2008-01-01 Marucci, Gabriella; Finaurini, S; Buccioni, Michela; Lammi, C; Kandhavelu, M; Volpini, Rosaria; Ricciutelli, Massimo; Angeli, Piero; Commandeur, Jnm; Cristalli, Gloria
Synthesis and pharmacological profile of a series of 1-substituted-2-carbonyl derivatives of diphenidol: novel M4 muscarinic receptor antagonists
2008-01-01 Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Fazio, N; Marucci, Gabriella; Recanatini, M; Spampanato, S.
Rapid novel divergent synthesis and muscarinic agonist profile of all four optical isomers of N,N,N-trimethyl(6-methyl-1,4-dioxan-2-yl)methanaminium iodide.
2008-01-01 Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Buccioni, Michela; Nesi, M; Matucci, R.
(2,2-Diphenyl-[1,3]oxathiolan-5-ylmethyl)-(3-phenyl-propyl)-amine: a Potent and Selective 5-HT1A Receptor Agonist
2009-01-01 Franchini, S.; Tait, A.; Prandi, A.; Sorbi, C.; Gallesi, R.; Buccioni, Michela; Marucci, Gabriella; DE STEFANI, C.; Cilia, A.; Brasili, L.
“Third Joint Italian-German Purine Club Meeting - Purinergic Receptors: New Frontiers for Novel Therapies”
2009-01-01 Cristalli, Gloria; Buccioni, Michela; Cappellacci, Loredana; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Petrelli, Riccardo; Volpini, Rosaria
8-Bromo-9-alkyl adenine derivatives as tools for developing new adenosine A(2A) and A(2B) receptors ligands
2009-01-01 Lambertucci, Catia; Antonini, Ippolito; Buccioni, Michela; DAL BEN, Diego; Kachare, Dd; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Synthesis and biological evaluation of 2-alkynyl-N6-methyl-5'-N-methylcarboxamidoadenosine derivatives as potent and highly selective agonists for the human adenosine A(3) receptor
2009-01-01 Volpini, Rosaria; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Marucci, Gabriella; Ramadori, At; Klotz, K. N.; Cristalli, Gloria
Existence of snoRNA, microRNA, piRNA characteristics in a novel non-coding RNA: x-ncRNA and its biological implication in Homo sapiens
2009-01-01 Kandhavelu, M; Lammi, C; Buccioni, Michela; DAL BEN, Diego; Volpini, Rosaria; Marucci, Gabriella
Identification of alpha(1)-adrenoceptor subtypes involved in contraction of young CD rat epididymal vas deferens
2009-01-01 Buccioni, Michela; Kandhavelu, M; Angeli, Piero; Cristalli, Gloria; DAL BEN, Diego; Giardinà, D; Lambertucci, Catia; Lammi, C; Volpini, Rosaria; Marucci, Gabriella
Molecular modeling studies on the human neuropeptide S receptor and its antagonists.
2010-01-01 DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria
Synthesis and α(1)-adrenoceptor antagonist activity of tamsulosin analogues
2010-01-01 Sagratini, Gianni; Angeli, Piero; Buccioni, Michela; Gulini, U; Marucci, Gabriella; Melchiorre, C; Poggesi, E; Giardinà, D.
1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: Structure-affinity/activity relationship at α1-adrenoceptor subtypes and at 5-HT1A receptors.
2010-01-01 Franchini, S; Prandi, A; Baraldi, A; Sorbi, C; Tait, A; Buccioni, Michela; Marucci, Gabriella; Cilia, A; Pirona, L; Fossa, P; Cichero, E; Brasili, L.
Identification of putative guanosine receptor in rat brain
2010-01-01 Lammi, C; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria
Human adenosine A3 receptor as selective target of new 2-aralkynyl-N6-methyl-MECA derivatives
2010-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Ramadori, At; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Synthesis and alpha1-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin | 1-gen-2007 | Sagratini, Gianni; Angeli, Piero; Buccioni, Michela; Gulini, Ugo; Marucci, Gabriella; Melchiorre, C; Leonardi, A; Poggesi, E; Giardina', Dario | Articolo | |
Dioxane and Oxathiane Nuclei: Suitable Substructures for Muscarinic Agonists | 1-gen-2007 | Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Bruni, B; Buccioni, Michela; Carrieri, A; Ciattini, S. | Articolo | |
Synthesis, affinity profile, and functional activity of muscarinic antagonists with a 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine structure | 1-gen-2007 | Dei, S.; Bellucci, C.; Buccioni, Michela; Ferraroni, M.; Guandalini, L.; Manetti, D.; Martini, E.; Marucci, Gabriella; Matucci, R.; Nesi, M.; Romanelli, M. N.; Scapecchi, S.; Teodori, E. | Articolo | |
Muscarinic antagonists with multiple stereocenters: Synthesis, affinity profile and functional activity of isomeric 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl) pyrrolidine sulfoxide derivatives | 1-gen-2008 | Dei, S.; Bellucci, C.; Buccioni, Michela; Ferraroni, M.; Guandalini, L.; Manetti, D.; Marucci, Gabriella; Matucci, R.; Nesi, M.; Romanelli, M. N.; Scapecchi, S.; Teodori, E. | Articolo | |
Synthesis and pharmacological characterization of chiral pyrrolidinylfuran derivatives: The discovery of new functionally selective muscarinic agonists | 1-gen-2008 | Scapecchi, S.; Nesi, M.; Matucci, R.; Bellucci, C.; Buccioni, Michela; Dei, S.; Guandalini, L.; Manetti, D.; Martini, E.; Marucci, Gabriella; Romanelli, M. N.; Teodori, E.; Cirilli, R. | Articolo | |
Levels of polychlorinated biphenyls in fish and shellfish from the Adriatic Sea | 1-gen-2008 | Sagratini, Gianni; Buccioni, Michela; Ciccarelli, C.; Conti, Paolo; Cristalli, Gloria; Giardina', Dario; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Vittori, Sauro | Articolo | |
In vitro metabolism studies of new adenosine A(2A) receptor antagonists | 1-gen-2008 | Marucci, Gabriella; Finaurini, S; Buccioni, Michela; Lammi, C; Kandhavelu, M; Volpini, Rosaria; Ricciutelli, Massimo; Angeli, Piero; Commandeur, Jnm; Cristalli, Gloria | Articolo | |
Synthesis and pharmacological profile of a series of 1-substituted-2-carbonyl derivatives of diphenidol: novel M4 muscarinic receptor antagonists | 1-gen-2008 | Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Fazio, N; Marucci, Gabriella; Recanatini, M; Spampanato, S. | Articolo | |
Rapid novel divergent synthesis and muscarinic agonist profile of all four optical isomers of N,N,N-trimethyl(6-methyl-1,4-dioxan-2-yl)methanaminium iodide. | 1-gen-2008 | Piergentili, Alessandro; Quaglia, Wilma; Giannella, Mario; DEL BELLO, Fabio; Buccioni, Michela; Nesi, M; Matucci, R. | Articolo | |
(2,2-Diphenyl-[1,3]oxathiolan-5-ylmethyl)-(3-phenyl-propyl)-amine: a Potent and Selective 5-HT1A Receptor Agonist | 1-gen-2009 | Franchini, S.; Tait, A.; Prandi, A.; Sorbi, C.; Gallesi, R.; Buccioni, Michela; Marucci, Gabriella; DE STEFANI, C.; Cilia, A.; Brasili, L. | Articolo | |
“Third Joint Italian-German Purine Club Meeting - Purinergic Receptors: New Frontiers for Novel Therapies” | 1-gen-2009 | Cristalli, Gloria; Buccioni, Michela; Cappellacci, Loredana; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Petrelli, Riccardo; Volpini, Rosaria | ORGANIZZAZIONE DI EVENTI | |
8-Bromo-9-alkyl adenine derivatives as tools for developing new adenosine A(2A) and A(2B) receptors ligands | 1-gen-2009 | Lambertucci, Catia; Antonini, Ippolito; Buccioni, Michela; DAL BEN, Diego; Kachare, Dd; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Synthesis and biological evaluation of 2-alkynyl-N6-methyl-5'-N-methylcarboxamidoadenosine derivatives as potent and highly selective agonists for the human adenosine A(3) receptor | 1-gen-2009 | Volpini, Rosaria; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Marucci, Gabriella; Ramadori, At; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Existence of snoRNA, microRNA, piRNA characteristics in a novel non-coding RNA: x-ncRNA and its biological implication in Homo sapiens | 1-gen-2009 | Kandhavelu, M; Lammi, C; Buccioni, Michela; DAL BEN, Diego; Volpini, Rosaria; Marucci, Gabriella | Articolo | |
Identification of alpha(1)-adrenoceptor subtypes involved in contraction of young CD rat epididymal vas deferens | 1-gen-2009 | Buccioni, Michela; Kandhavelu, M; Angeli, Piero; Cristalli, Gloria; DAL BEN, Diego; Giardinà, D; Lambertucci, Catia; Lammi, C; Volpini, Rosaria; Marucci, Gabriella | Articolo | |
Molecular modeling studies on the human neuropeptide S receptor and its antagonists. | 1-gen-2010 | DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Vittori, Sauro; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Synthesis and α(1)-adrenoceptor antagonist activity of tamsulosin analogues | 1-gen-2010 | Sagratini, Gianni; Angeli, Piero; Buccioni, Michela; Gulini, U; Marucci, Gabriella; Melchiorre, C; Poggesi, E; Giardinà, D. | Articolo | |
1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: Structure-affinity/activity relationship at α1-adrenoceptor subtypes and at 5-HT1A receptors. | 1-gen-2010 | Franchini, S; Prandi, A; Baraldi, A; Sorbi, C; Tait, A; Buccioni, Michela; Marucci, Gabriella; Cilia, A; Pirona, L; Fossa, P; Cichero, E; Brasili, L. | Articolo | |
Identification of putative guanosine receptor in rat brain | 1-gen-2010 | Lammi, C; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Volpini, Rosaria; Cristalli, Gloria | Abstract atto convegno su rivista | |
Human adenosine A3 receptor as selective target of new 2-aralkynyl-N6-methyl-MECA derivatives | 1-gen-2010 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Ramadori, At; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Abstract atto convegno su rivista |
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