Sfoglia per Autore
Early evaluation of a new 2,2'-bipyridyl derivative with potential inhibitory activity on the ribocleotide reductase enzyme
1990-01-01 G., Nocentini; E., Marconi; Franchetti, Palmarisa; Cappellacci, Loredana; A., Barzi
Synthesis and evaluation of anti-HIV-1 and antitumor activity of 2',3'-didehydro-2',3'-dideoxy-3-deazaadenosine, 2',3'-dideoxy-3-deazaadenosine and some 2',3'-dideoxy-3-deazaadenosine 5'-dialkyl phosphates
1991-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Cristalli, Gloria; Grifantini, Mario; Pani, A; LA COLLA, P; Nocentini, G.
Synthesis of 3-deazaclitocine [2-amino-3-nitro-4-(beta-D-ribofuranosylamino)pyridine] as cytotoxic agent
1991-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Cristalli, Gloria; Grifantini, Mario; Vittori, Sauro
Synthesis and antiviral evaluation of 1-deaza-8-aza- and 3-deaza-8-aza-purine nucleosides
1992-01-01 P., La Colla; Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; L., Messini; Me, Marongiu; A., Pani
8-Aza analogues of deaza purine nucleosides. Synthesis and biological evaluation of 8-aza-1-deazaadenosine and 2'-deoxy-8-aza-1-deazaadenosine
1992-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Lupidi, Giulio; Nocentini, G; Barzi, A.
A new facile synthesis and antiviral activity of oxazofurin
1993-01-01 Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; Grifantini, Mario; Guarracino, P; Marongiu, Me; Piras, G; LA COLLA, P.
Synthesis and in vivo antiviral activity of 8-aza-analogues of potent antiviral agents 9-[2-phosphonomethoxy)ethyl]adenine (PMEA) and 9-[2-phosphonomethoxy)ethyl]guanine (PMEG)
1993-01-01 Franchetti, Palmarisa; G., Abu Sheikha; Cappellacci, Loredana; L., Messini; Grifantini, Mario; Me, Marongiu; P., Guarracino; P., La Colla
8-Aza derivatives of 3-deazapurine nucleosides. Synthesis and in vitro evaluation of antiviral and antitumor activity
1993-01-01 Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; Grifantini, Mario; Nocentini, G; Guarracino, P; Marongiu, Me; LA COLLA, P.
Synthesis and evaluation of the anti-HIV activity of aza and deaza analogues of IsoddA and their phosphates as prodrugs.
1994-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Messini, L; ABU SHEIKHA, G; Loi, Ag; Tramontano, E; DE MONTIS, A; Spiga, Mg; LA COLLA, P.
8-Aza-1-deaza purine nucleosides as antiviral agents.
1994-01-01 Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; ABU SHEIKHA, G; Grifantini, Mario; Guarracino, P; DE MONTIS, A; Loi, Ag; Marongiu, Me; LA COLLA, P.
C-Glycosyl bond conformation in oxazofurin: crystallographic and computational studies of the oxazole analogue of tiazofurin.
1994-01-01 Goldstein, Bm; Li, H; Hallows, Wh; Langs, Da; Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario
8-Aza-analogues of PMEA and PMEG: synthesis and in vitro anti-HIV activity.
1994-01-01 Franchetti, Palmarisa; ABU SHEIKHA, G; Cappellacci, Loredana; Messini, L; Grifantini, Mario; Loi, Ag; DE MONTIS, A; Spiga, M; LA COLLA, P.
8-Azaxanthine derivatives as antagonists of adenosine receptors.
1994-01-01 Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; Grifantini, Mario; Lucacchini, A; Martini, C; Senatore, G.
Synthesis and anti-HIV activity of isonucleosides and acyclic nucleotides related to clitocine
1994-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; G., Abu Sheikha; Grifantini, Mario; L., Messini; Ag, Loi; A., De Montis; Mg, Spiga; P., La Colla
Synthesis and antiviral activity of 8-aza analogs of chiral [2-(Phosphono-methoxy)propyl]guanines.
1995-01-01 Franchetti, Palmarisa; ABU SHEIKHA, G; Cappellacci, Loredana; Grifantini, Mario; DE MONTIS, A; Piras, G; Loi, Ag; LA COLLA, P.
Tiazofurin analogs as selective agonists of A1 adenosine receptors
1995-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Senatore, G; Martini, C; Lucacchini, A.
Synthesis, antitumor activity and crystallographic studies of analogues of tiazofurin
1995-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; ABU SHEIKHA, G; Nocentini, G; Moraca, R; Goldstein, Bm
Furanfurin and Thiophenfurin: Two Novel Tiazofurin Analogues. Synthesis, Structure, Antitumor Activity and Interactions with IMP Dehydrogenase
1995-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Barzi, A.; G. NOCENTINI, G.; Yang, H.; O'Connor, A.; Jayaram, H. N.; Carrell, C.; Goldstein, B. M.
Acyclic nucleotides related to clitocine: synthesis and anti-HIV activity
1995-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; ABU SHEIKHA, G; Grifantini, Mario; Loi, Ag; DE MONTIS, A; Spiga, Mg; LA COLLA, P.
2'-C-Methyl analogs of selective adenosine receptors agonists: synthesis and binding studies
1996-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Costa, B; Martini, C; Lucacchini, A.
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Early evaluation of a new 2,2'-bipyridyl derivative with potential inhibitory activity on the ribocleotide reductase enzyme | 1-gen-1990 | G., Nocentini; E., Marconi; Franchetti, Palmarisa; Cappellacci, Loredana; A., Barzi | Poster atto convegno su rivista | |
Synthesis and evaluation of anti-HIV-1 and antitumor activity of 2',3'-didehydro-2',3'-dideoxy-3-deazaadenosine, 2',3'-dideoxy-3-deazaadenosine and some 2',3'-dideoxy-3-deazaadenosine 5'-dialkyl phosphates | 1-gen-1991 | Franchetti, Palmarisa; Cappellacci, Loredana; Cristalli, Gloria; Grifantini, Mario; Pani, A; LA COLLA, P; Nocentini, G. | Articolo | |
Synthesis of 3-deazaclitocine [2-amino-3-nitro-4-(beta-D-ribofuranosylamino)pyridine] as cytotoxic agent | 1-gen-1991 | Franchetti, Palmarisa; Cappellacci, Loredana; Cristalli, Gloria; Grifantini, Mario; Vittori, Sauro | Articolo | |
Synthesis and antiviral evaluation of 1-deaza-8-aza- and 3-deaza-8-aza-purine nucleosides | 1-gen-1992 | P., La Colla; Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; L., Messini; Me, Marongiu; A., Pani | Poster atto convegno su rivista | |
8-Aza analogues of deaza purine nucleosides. Synthesis and biological evaluation of 8-aza-1-deazaadenosine and 2'-deoxy-8-aza-1-deazaadenosine | 1-gen-1992 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Lupidi, Giulio; Nocentini, G; Barzi, A. | Articolo | |
A new facile synthesis and antiviral activity of oxazofurin | 1-gen-1993 | Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; Grifantini, Mario; Guarracino, P; Marongiu, Me; Piras, G; LA COLLA, P. | Articolo | |
Synthesis and in vivo antiviral activity of 8-aza-analogues of potent antiviral agents 9-[2-phosphonomethoxy)ethyl]adenine (PMEA) and 9-[2-phosphonomethoxy)ethyl]guanine (PMEG) | 1-gen-1993 | Franchetti, Palmarisa; G., Abu Sheikha; Cappellacci, Loredana; L., Messini; Grifantini, Mario; Me, Marongiu; P., Guarracino; P., La Colla | Poster atto convegno su rivista | |
8-Aza derivatives of 3-deazapurine nucleosides. Synthesis and in vitro evaluation of antiviral and antitumor activity | 1-gen-1993 | Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; Grifantini, Mario; Nocentini, G; Guarracino, P; Marongiu, Me; LA COLLA, P. | Articolo | |
Synthesis and evaluation of the anti-HIV activity of aza and deaza analogues of IsoddA and their phosphates as prodrugs. | 1-gen-1994 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Messini, L; ABU SHEIKHA, G; Loi, Ag; Tramontano, E; DE MONTIS, A; Spiga, Mg; LA COLLA, P. | Articolo | |
8-Aza-1-deaza purine nucleosides as antiviral agents. | 1-gen-1994 | Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; ABU SHEIKHA, G; Grifantini, Mario; Guarracino, P; DE MONTIS, A; Loi, Ag; Marongiu, Me; LA COLLA, P. | Articolo | |
C-Glycosyl bond conformation in oxazofurin: crystallographic and computational studies of the oxazole analogue of tiazofurin. | 1-gen-1994 | Goldstein, Bm; Li, H; Hallows, Wh; Langs, Da; Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario | Articolo | |
8-Aza-analogues of PMEA and PMEG: synthesis and in vitro anti-HIV activity. | 1-gen-1994 | Franchetti, Palmarisa; ABU SHEIKHA, G; Cappellacci, Loredana; Messini, L; Grifantini, Mario; Loi, Ag; DE MONTIS, A; Spiga, M; LA COLLA, P. | Articolo | |
8-Azaxanthine derivatives as antagonists of adenosine receptors. | 1-gen-1994 | Franchetti, Palmarisa; Messini, L; Cappellacci, Loredana; Grifantini, Mario; Lucacchini, A; Martini, C; Senatore, G. | Articolo | |
Synthesis and anti-HIV activity of isonucleosides and acyclic nucleotides related to clitocine | 1-gen-1994 | Franchetti, Palmarisa; Cappellacci, Loredana; G., Abu Sheikha; Grifantini, Mario; L., Messini; Ag, Loi; A., De Montis; Mg, Spiga; P., La Colla | Poster atto convegno su rivista | |
Synthesis and antiviral activity of 8-aza analogs of chiral [2-(Phosphono-methoxy)propyl]guanines. | 1-gen-1995 | Franchetti, Palmarisa; ABU SHEIKHA, G; Cappellacci, Loredana; Grifantini, Mario; DE MONTIS, A; Piras, G; Loi, Ag; LA COLLA, P. | Articolo | |
Tiazofurin analogs as selective agonists of A1 adenosine receptors | 1-gen-1995 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Senatore, G; Martini, C; Lucacchini, A. | Articolo | |
Synthesis, antitumor activity and crystallographic studies of analogues of tiazofurin | 1-gen-1995 | Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; ABU SHEIKHA, G; Nocentini, G; Moraca, R; Goldstein, Bm | Articolo | |
Furanfurin and Thiophenfurin: Two Novel Tiazofurin Analogues. Synthesis, Structure, Antitumor Activity and Interactions with IMP Dehydrogenase | 1-gen-1995 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Barzi, A.; G. NOCENTINI, G.; Yang, H.; O'Connor, A.; Jayaram, H. N.; Carrell, C.; Goldstein, B. M. | Articolo | |
Acyclic nucleotides related to clitocine: synthesis and anti-HIV activity | 1-gen-1995 | Franchetti, Palmarisa; Cappellacci, Loredana; ABU SHEIKHA, G; Grifantini, Mario; Loi, Ag; DE MONTIS, A; Spiga, Mg; LA COLLA, P. | Articolo | |
2'-C-Methyl analogs of selective adenosine receptors agonists: synthesis and binding studies | 1-gen-1996 | Franchetti, Palmarisa; Cappellacci, Loredana; Grifantini, Mario; Costa, B; Martini, C; Lucacchini, A. | Poster atto convegno su rivista |
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