Sfoglia per Autore
Synthesis and alpha-blocking activity of some analogues of idazoxan
1987-01-01 Pigini, Maria; Brasili, L.; Cassinelli, A.; Giardinà, D.; Gulini, U.; Quaglia, Wilma; Melchiorre, C.
Structure-activity relationships in 1,4-benzodioxan-related compounds. Investigation on the role of the dehydrodioxane ring on alpha1-adrenoreceptor blocking activity
1988-01-01 Pigini, Maria; Brasili, L.; Giannella, Mario; Giardinà, D.; Gulini, U.; Quaglia, Wilma; Melchiorre, C.
3-Phenyl analogues of 2-[[[2-(2,6-Dimethoxyphenoxyethyllamino]methyl]-1,4-benzodioxan (WB 4101) as highly selective alpha1-adrenoreceptor antagonists1
1990-01-01 Quaglia, Wilma; Pigini, Maria; Giannella, Mario; Melchiorre, C.
“Pharmacological Characterization of Muscarinic Receptor Subtypes in Rabbit Isolated Tissue Preparations”
1991-01-01 Angeli, Piero; Brasili, L; Cingolani, M. L.; Marucci, Gabriella; Pigini, Maria; Tonnini, M. C.
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 4. Effect of aryl and alkyl Substituents at Position 3 on α-adrenoreceptor blocking activity
1993-01-01 Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Melchiorre, C.
Synthesis and muscarinic properties of (1S*,3R*,5R*)-trimethyl(1-methyl-6-oxabicyclo[3.1.0]hex-3-yl)methyl ammonium iodide
1994-01-01 Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Rafaiani, Giovanni; Tayebati, Seyed Khosrow
Separation of alpha-adrenergic and imidazoline/guanidinium receptive sites (IGRS) activity in a series of imidazoline analogues of cirazoline
1995-01-01 Brasili, L.; Pigini, Maria; Marucci, Gabriella; Quaglia, Wilma; Malmusi, L.; Lanier, S. M.; Lanier, B.
Age-related Changes in the Density of Muscarinic Cholinergic M1 and M2 Receptor Subtypes in Pyramidal Neurons or the rat Hippocampus
1995-01-01 Amenta, Francesco; A., Liu; Giannella, Mario; Pigini, Maria; Tayebati, Seyed Khosrow; AND D., Zaccheo
Muscarinic Thioligands with Cyclopentane Nucleus
1996-01-01 Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow; Amenta, Francesco; Sabbatini, M.; Giannella, Mario
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 5. Effects of Modification of the side chain on alpha-adrenoreceptor blocking Activity
1996-01-01 Quaglia, Wilma; Giannella, Mario; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Tayebati, Seyed Khosrow; Melchiorre, C.
Discovery of Highly Selective Imidazoline Receptor Ligands
1996-01-01 L., Brasili; Pigini, Maria; R., Moriconi; A., Carotti; P., Bousquet; M., Dontenwill; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow
Synthesis, Absolute Configuration, and Biological Profile of the Enantiomers of trans-[2-(2,6-Dimethoxypheoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (Mephendioxan), a Potent Competitive alpha 1A-Adrenoreceptor Antagonist
1996-01-01 Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; A., Leonardi; C., Taddei; C., Melchiorre
Byciclic dioxolanes as potential antimuscarinic agents
1996-01-01 Piergentili, Alessandro; Angeli, Piero; Giannella, Mario; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow
Imidazoline receptors: Qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity
1997-01-01 Pigini, Maria; Bousquet, P; Carotti, A; Dontenwill, M; Giannella, Mario; Moriconi, R; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow; Brasili, L.
Use of frozen sections for the pharmacological characterization of compounds active on neurotransmitter receptors
1997-01-01 Tayebati, Seyed Khosrow; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Sabbatini, M.; Amenta, Francesco
Synthesis and Structure-Activity Relationship Studies in a Series of 2-Substituted 1,3-Dioxolanes Modified at the Cationic Head.
1997-01-01 Angeli, Piero; Cingolani, Augusto; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models
1998-01-01 Pigini, Maria; Bousquet, P.; Brasili, L.; Carrieri, A.; Cavagna, R.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Leonetti, F.; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A.
1'-Benzyl-3,4-dihydrospiro[2H-1-benzothiopyran-2,4'-piperidine] (Spipethiane), a potent and highly selective sigma1 lingand
1998-01-01 Quaglia, Wilma; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Brasili, L.; DI TORO, R.; Rossetti, R.; Spampinato, S.; Melchiorre, C.
Binding of Tracizolines to the Imidazoline Receptor. Role of Lipophilicity in Quantitative Structure-Activity Relationship Models.
1999-01-01 Pigini, Maria; Bousquet, P; Brasili, L; Carrieri, A; Dontenwill, M; Gentili, Francesco; Giannella, Mario; Leonetti, F; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A.
2-(2-Phenylcyclopropyl)imidazolines: Reversed Enantioselective Interaction at I1 and I2 Imidazoline Receptors
1999-01-01 Quaglia, Wilma; Bousquet, P.; Pigini, Maria; Carotti, A.; Carrieri, A.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Maranca, F.; Piergentili, Alessandro; Brasili, L.
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Synthesis and alpha-blocking activity of some analogues of idazoxan | 1-gen-1987 | Pigini, Maria; Brasili, L.; Cassinelli, A.; Giardinà, D.; Gulini, U.; Quaglia, Wilma; Melchiorre, C. | Articolo | |
Structure-activity relationships in 1,4-benzodioxan-related compounds. Investigation on the role of the dehydrodioxane ring on alpha1-adrenoreceptor blocking activity | 1-gen-1988 | Pigini, Maria; Brasili, L.; Giannella, Mario; Giardinà, D.; Gulini, U.; Quaglia, Wilma; Melchiorre, C. | Articolo | |
3-Phenyl analogues of 2-[[[2-(2,6-Dimethoxyphenoxyethyllamino]methyl]-1,4-benzodioxan (WB 4101) as highly selective alpha1-adrenoreceptor antagonists1 | 1-gen-1990 | Quaglia, Wilma; Pigini, Maria; Giannella, Mario; Melchiorre, C. | Articolo | |
“Pharmacological Characterization of Muscarinic Receptor Subtypes in Rabbit Isolated Tissue Preparations” | 1-gen-1991 | Angeli, Piero; Brasili, L; Cingolani, M. L.; Marucci, Gabriella; Pigini, Maria; Tonnini, M. C. | Articolo | |
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 4. Effect of aryl and alkyl Substituents at Position 3 on α-adrenoreceptor blocking activity | 1-gen-1993 | Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Melchiorre, C. | Articolo | |
Synthesis and muscarinic properties of (1S*,3R*,5R*)-trimethyl(1-methyl-6-oxabicyclo[3.1.0]hex-3-yl)methyl ammonium iodide | 1-gen-1994 | Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Rafaiani, Giovanni; Tayebati, Seyed Khosrow | Articolo | |
Separation of alpha-adrenergic and imidazoline/guanidinium receptive sites (IGRS) activity in a series of imidazoline analogues of cirazoline | 1-gen-1995 | Brasili, L.; Pigini, Maria; Marucci, Gabriella; Quaglia, Wilma; Malmusi, L.; Lanier, S. M.; Lanier, B. | Articolo | |
Age-related Changes in the Density of Muscarinic Cholinergic M1 and M2 Receptor Subtypes in Pyramidal Neurons or the rat Hippocampus | 1-gen-1995 | Amenta, Francesco; A., Liu; Giannella, Mario; Pigini, Maria; Tayebati, Seyed Khosrow; AND D., Zaccheo | Articolo | |
Muscarinic Thioligands with Cyclopentane Nucleus | 1-gen-1996 | Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow; Amenta, Francesco; Sabbatini, M.; Giannella, Mario | Articolo | |
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 5. Effects of Modification of the side chain on alpha-adrenoreceptor blocking Activity | 1-gen-1996 | Quaglia, Wilma; Giannella, Mario; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Tayebati, Seyed Khosrow; Melchiorre, C. | Articolo | |
Discovery of Highly Selective Imidazoline Receptor Ligands | 1-gen-1996 | L., Brasili; Pigini, Maria; R., Moriconi; A., Carotti; P., Bousquet; M., Dontenwill; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow | Capitolo di libro o voce di enciclopedia | |
Synthesis, Absolute Configuration, and Biological Profile of the Enantiomers of trans-[2-(2,6-Dimethoxypheoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (Mephendioxan), a Potent Competitive alpha 1A-Adrenoreceptor Antagonist | 1-gen-1996 | Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; A., Leonardi; C., Taddei; C., Melchiorre | Articolo | |
Byciclic dioxolanes as potential antimuscarinic agents | 1-gen-1996 | Piergentili, Alessandro; Angeli, Piero; Giannella, Mario; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow | Articolo | |
Imidazoline receptors: Qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity | 1-gen-1997 | Pigini, Maria; Bousquet, P; Carotti, A; Dontenwill, M; Giannella, Mario; Moriconi, R; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow; Brasili, L. | Articolo | |
Use of frozen sections for the pharmacological characterization of compounds active on neurotransmitter receptors | 1-gen-1997 | Tayebati, Seyed Khosrow; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Sabbatini, M.; Amenta, Francesco | Articolo | |
Synthesis and Structure-Activity Relationship Studies in a Series of 2-Substituted 1,3-Dioxolanes Modified at the Cationic Head. | 1-gen-1997 | Angeli, Piero; Cingolani, Augusto; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | Articolo | |
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models | 1-gen-1998 | Pigini, Maria; Bousquet, P.; Brasili, L.; Carrieri, A.; Cavagna, R.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Leonetti, F.; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A. | Articolo | |
1'-Benzyl-3,4-dihydrospiro[2H-1-benzothiopyran-2,4'-piperidine] (Spipethiane), a potent and highly selective sigma1 lingand | 1-gen-1998 | Quaglia, Wilma; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Brasili, L.; DI TORO, R.; Rossetti, R.; Spampinato, S.; Melchiorre, C. | Articolo | |
Binding of Tracizolines to the Imidazoline Receptor. Role of Lipophilicity in Quantitative Structure-Activity Relationship Models. | 1-gen-1999 | Pigini, Maria; Bousquet, P; Brasili, L; Carrieri, A; Dontenwill, M; Gentili, Francesco; Giannella, Mario; Leonetti, F; Piergentili, Alessandro; Quaglia, Wilma; Carotti, A. | Articolo | |
2-(2-Phenylcyclopropyl)imidazolines: Reversed Enantioselective Interaction at I1 and I2 Imidazoline Receptors | 1-gen-1999 | Quaglia, Wilma; Bousquet, P.; Pigini, Maria; Carotti, A.; Carrieri, A.; Dontenwill, M.; Gentili, Francesco; Giannella, Mario; Maranca, F.; Piergentili, Alessandro; Brasili, L. | Articolo |
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