Sfoglia per Autore
Novel Highly Potent and Selective σ1 Receptor Antagonists Related to Spipethiane
2010-01-01 Piergentili, Alessandro; Amantini, Consuelo; DEL BELLO, Fabio; Giannella, Mario; Mattioli, Laura; Maura, Palmery; Perfumi, Marina Cecilia; Pigini, Maria; Santoni, Giorgio; Paolo, Tucci; Margherita, Zotti; Quaglia, Wilma
Structure-activity relationships in 1,4-benzodioxan-related compounds. 10. Novel alpha1-adrenoreceptor antagonists related to openphendioxan: synthesis, biological evaluation, and alpha1d computational study
2010-01-01 Carrieri, A.; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Leonardi, A.; Fanelli, F.; Quaglia, Wilma
Fruitful Adrenergic alpha(2C)-Agonism/alpha(2A)-Antagonism Combination to Prevent and Contrast Morphine Tolerance and Dependence
2010-01-01 DEL BELLO, Fabio; Mattioli, Laura; Ghelfi, Francesca; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Cardinaletti, Claudia; Perfumi, Marina Cecilia; Thomas, R. J.; Zanelli, U.; Marchioro, C.; DAL CIN, M.; Pigini, Maria
From benzodioxane to 1,4-dioxane scaffold in the design of 5-HT1A serotoninergic full agonists from α1-adrenergic antagonists
2011-01-01 DEL BELLO, Fabio; Y. A., Farande; A., Bonifazi; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Allyphenyline analogues potentially useful in the management of chronic pain and opioid addiction.
2011-01-01 E., Diamanti; DEL BELLO, Fabio; Giannella, Mario; V., Mammoli; Piergentili, Alessandro; Quaglia, Wilma; A., Carrieri; G., Carbonara; G., Fracchiolla; Pigini, Maria
Hybrid molecules from xanomeline and 77-LH-28-1 as potential novel M1 muscarinic agonists
2011-01-01 Piergentili, Alessandro; A., Bonifazi; M., Cancellieri; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Quaglia, Wilma; C., Castaldo; M., Pollastrini; M., Nesi; Rosanna, Matucci
Alpha2C-adrenoceptor modulators: a patent review
2011-01-01 Quaglia, Wilma; DEL BELLO, Fabio; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria
Might Allyphenyline and Cyclomethyline Become Profitable Multifunctional Tools in the Opioid Addiction Management?
2012-01-01 DEL BELLO, Fabio
Design and synthesis of novel imidazoline derivatives potentially targeting dopamine receptors
2012-01-01 DEL BELLO, Fabio; Giannella, Mario; V., Mammoli; Piergentili, Alessandro; Quaglia, Wilma
Imidazoline nucleus as a biologically versatile scaffold
2012-01-01 DEL BELLO, Fabio; V., Mammoli; A., Bonifazi; E., Diamanti; Giannella, Mario; A. L., Hudson; Mattioli, Laura; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
Low doses of allyphenyline and cyclomethyline, effective against morphine dependence, elicit an antidepressant-like effect
2012-01-01 DEL BELLO, Fabio; Diamanti, E.; Giannella, Mario; Mammoli, V.; Marchioro, C.; Mattioli, Laura; Titomanlio, F.; Piergentili, Alessandro; Quaglia, Wilma; Benedetti, G; Varrone, M.; Pigini, Maria
Might the observed alpha2A-adrenoreceptor agonism or antagonism of allyphenyline analogues be ascribed to different molecular conformations?
2012-01-01 Diamanti, E; DEL BELLO, Fabio; Carbonara, G; Carrieri, A; Fracchiolla, G; Giannella, Mario; Mammoli, V; Piergentili, Alessandro; Pohjanoksa, K; Quaglia, Wilma; Scheinin, M; Pigini, Maria
1,4-Dioxane, a Suitable Scaffold for the Development of Novel M3 Muscarinic Receptor Antagonists
2012-01-01 DEL BELLO, Fabio; Barocelli, E.; Bertoni, S.; Bonifazi, A.; Camalli, M.; Campi, G.; Giannella, Mario; Matucci, R.; Nesi, M.; Pigini, Maria; Quaglia, Wilma; Piergentili, Alessandro
Favourable involvement of α2A-adrenoreceptor antagonism in the I₂-imidazoline binding sites-mediated morphine analgesia enhancement.
2012-01-01 Mammoli, Valerio; Bonifazi, Alessandro; DEL BELLO, Fabio; Diamanti, Eleonora; Giannella, Mario; Hudson, Al; Mattioli, Laura; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Titomanlio, Federica; Pigini, Maria
Effects of imidazoline I2 receptor ligands on acute nociception in rats
2012-01-01 Cristal, Sampson; Yanan, Zhang; DEL BELLO, Fabio; Jun Xu, Li
31st Camerino-Cyprus-Noordwijkerhout Symposium - Receptor Chemistry Skyline
2013-01-01 Angeli, Piero; DEL BELLO, Fabio; Pigini, Maria; Giannella, Mario; Giorgioni, Gianfabio; Quaglia, Wilma; Piergentili, Alessandro; Giardina', Dario
31st Camerino-Cyprus-Noordwijkerhout Symposium - Receptor Chemistry Skyline
2013-01-01 Angeli, Piero; DEL BELLO, Fabio; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
NOVEL BIVALENT LIGANDS OF XANOMELINE AND 77-LH-28-1 AS POTENTIAL M1 MUSCARINIC AGONISTS
2013-01-01 Bonifazi, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Mammoli, Valerio; Pigini, Maria; Piergentili, Alessandro; Quaglia, Wilma; Hideaki, Yano; Sergi, Ferré; Marta, Nesi; Rosanna, Matucci
1,4-DIOXANE NUCLEUS AS A SUITABLE SCAFFOLD FOR NOVEL D2-LIKE RECEPTOR LIGANDS
2013-01-01 Bonifazi, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Thomas M., Keck; Amy H., Newman
MORPHINE TOLERANCE MODULATION INDUCED BY alpha2-ADRENERGIC OR/AND I2 IMIDAZOLINE BINDING SITES LIGANDS
2013-01-01 DEL BELLO, Fabio; Giannella, Mario; Mammoli, Valerio; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria; Laura, Mennuni; Flora, Ferrari; Gianfranco, Caselli; Marco, Lanza
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Novel Highly Potent and Selective σ1 Receptor Antagonists Related to Spipethiane | 1-gen-2010 | Piergentili, Alessandro; Amantini, Consuelo; DEL BELLO, Fabio; Giannella, Mario; Mattioli, Laura; Maura, Palmery; Perfumi, Marina Cecilia; Pigini, Maria; Santoni, Giorgio; Paolo, Tucci; Margherita, Zotti; Quaglia, Wilma | Articolo | |
Structure-activity relationships in 1,4-benzodioxan-related compounds. 10. Novel alpha1-adrenoreceptor antagonists related to openphendioxan: synthesis, biological evaluation, and alpha1d computational study | 1-gen-2010 | Carrieri, A.; Piergentili, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Leonardi, A.; Fanelli, F.; Quaglia, Wilma | Articolo | |
Fruitful Adrenergic alpha(2C)-Agonism/alpha(2A)-Antagonism Combination to Prevent and Contrast Morphine Tolerance and Dependence | 1-gen-2010 | DEL BELLO, Fabio; Mattioli, Laura; Ghelfi, Francesca; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Cardinaletti, Claudia; Perfumi, Marina Cecilia; Thomas, R. J.; Zanelli, U.; Marchioro, C.; DAL CIN, M.; Pigini, Maria | Articolo | |
From benzodioxane to 1,4-dioxane scaffold in the design of 5-HT1A serotoninergic full agonists from α1-adrenergic antagonists | 1-gen-2011 | DEL BELLO, Fabio; Y. A., Farande; A., Bonifazi; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | Contributo in atto di convegno su volume | |
Allyphenyline analogues potentially useful in the management of chronic pain and opioid addiction. | 1-gen-2011 | E., Diamanti; DEL BELLO, Fabio; Giannella, Mario; V., Mammoli; Piergentili, Alessandro; Quaglia, Wilma; A., Carrieri; G., Carbonara; G., Fracchiolla; Pigini, Maria | Poster atto convegno su volume | |
Hybrid molecules from xanomeline and 77-LH-28-1 as potential novel M1 muscarinic agonists | 1-gen-2011 | Piergentili, Alessandro; A., Bonifazi; M., Cancellieri; DEL BELLO, Fabio; Giannella, Mario; Pigini, Maria; Quaglia, Wilma; C., Castaldo; M., Pollastrini; M., Nesi; Rosanna, Matucci | Poster atto convegno su volume | |
Alpha2C-adrenoceptor modulators: a patent review | 1-gen-2011 | Quaglia, Wilma; DEL BELLO, Fabio; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria | Articolo | |
Might Allyphenyline and Cyclomethyline Become Profitable Multifunctional Tools in the Opioid Addiction Management? | 1-gen-2012 | DEL BELLO, Fabio | Contributo in atto di convegno su volume | |
Design and synthesis of novel imidazoline derivatives potentially targeting dopamine receptors | 1-gen-2012 | DEL BELLO, Fabio; Giannella, Mario; V., Mammoli; Piergentili, Alessandro; Quaglia, Wilma | Poster atto convegno su volume | |
Imidazoline nucleus as a biologically versatile scaffold | 1-gen-2012 | DEL BELLO, Fabio; V., Mammoli; A., Bonifazi; E., Diamanti; Giannella, Mario; A. L., Hudson; Mattioli, Laura; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | Contributo in atto di convegno su volume | |
Low doses of allyphenyline and cyclomethyline, effective against morphine dependence, elicit an antidepressant-like effect | 1-gen-2012 | DEL BELLO, Fabio; Diamanti, E.; Giannella, Mario; Mammoli, V.; Marchioro, C.; Mattioli, Laura; Titomanlio, F.; Piergentili, Alessandro; Quaglia, Wilma; Benedetti, G; Varrone, M.; Pigini, Maria | Articolo | |
Might the observed alpha2A-adrenoreceptor agonism or antagonism of allyphenyline analogues be ascribed to different molecular conformations? | 1-gen-2012 | Diamanti, E; DEL BELLO, Fabio; Carbonara, G; Carrieri, A; Fracchiolla, G; Giannella, Mario; Mammoli, V; Piergentili, Alessandro; Pohjanoksa, K; Quaglia, Wilma; Scheinin, M; Pigini, Maria | Articolo | |
1,4-Dioxane, a Suitable Scaffold for the Development of Novel M3 Muscarinic Receptor Antagonists | 1-gen-2012 | DEL BELLO, Fabio; Barocelli, E.; Bertoni, S.; Bonifazi, A.; Camalli, M.; Campi, G.; Giannella, Mario; Matucci, R.; Nesi, M.; Pigini, Maria; Quaglia, Wilma; Piergentili, Alessandro | Articolo | |
Favourable involvement of α2A-adrenoreceptor antagonism in the I₂-imidazoline binding sites-mediated morphine analgesia enhancement. | 1-gen-2012 | Mammoli, Valerio; Bonifazi, Alessandro; DEL BELLO, Fabio; Diamanti, Eleonora; Giannella, Mario; Hudson, Al; Mattioli, Laura; Perfumi, Marina Cecilia; Piergentili, Alessandro; Quaglia, Wilma; Titomanlio, Federica; Pigini, Maria | Articolo | |
Effects of imidazoline I2 receptor ligands on acute nociception in rats | 1-gen-2012 | Cristal, Sampson; Yanan, Zhang; DEL BELLO, Fabio; Jun Xu, Li | Articolo | |
31st Camerino-Cyprus-Noordwijkerhout Symposium - Receptor Chemistry Skyline | 1-gen-2013 | Angeli, Piero; DEL BELLO, Fabio; Pigini, Maria; Giannella, Mario; Giorgioni, Gianfabio; Quaglia, Wilma; Piergentili, Alessandro; Giardina', Dario | ORGANIZZAZIONE DI EVENTI | |
31st Camerino-Cyprus-Noordwijkerhout Symposium - Receptor Chemistry Skyline | 1-gen-2013 | Angeli, Piero; DEL BELLO, Fabio; Giannella, Mario; Giardina', Dario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | Cura di atti, volumi e cataloghi | |
NOVEL BIVALENT LIGANDS OF XANOMELINE AND 77-LH-28-1 AS POTENTIAL M1 MUSCARINIC AGONISTS | 1-gen-2013 | Bonifazi, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Mammoli, Valerio; Pigini, Maria; Piergentili, Alessandro; Quaglia, Wilma; Hideaki, Yano; Sergi, Ferré; Marta, Nesi; Rosanna, Matucci | Poster atto convegno su volume | |
1,4-DIOXANE NUCLEUS AS A SUITABLE SCAFFOLD FOR NOVEL D2-LIKE RECEPTOR LIGANDS | 1-gen-2013 | Bonifazi, Alessandro; DEL BELLO, Fabio; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Thomas M., Keck; Amy H., Newman | Poster atto convegno su volume | |
MORPHINE TOLERANCE MODULATION INDUCED BY alpha2-ADRENERGIC OR/AND I2 IMIDAZOLINE BINDING SITES LIGANDS | 1-gen-2013 | DEL BELLO, Fabio; Giannella, Mario; Mammoli, Valerio; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria; Laura, Mennuni; Flora, Ferrari; Gianfranco, Caselli; Marco, Lanza | Poster atto convegno su volume |
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