Sfoglia per Autore
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario
Synthesis and Enzymatic Evaluation of NAD Mimics as Nicotinamide Adenine Dinucleotide Kinase (NADK) Inhibitors
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Krzysztof, Felczak; Vita, Patrizia; Torquati, Ilaria; Palmarisa, Franchetti; Michele Di, Stefano; Giulio, Magni; Mario, Grifantini; Krzysztof W., Pankiewicz
Synthesis and biological activity of novel N6-substituted and 2,N6-disubstituted adenine ribo- and 3'-C-methyl-ribonucleosides as antitumor agents
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Franchetti, Palmarisa; Vita, Patrizia; Kusumanchi, P; Kumar, M; Jayaram, H. N.; Zhou, B; Yen, Y; Grifantini, Mario
Synthesis and biological evaluation of (methylene)bisphosphonate derivatives of 2’-C-methyl-, and 3’-C-methyl-adenosine
2012-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Palmarisa, Franchetti; Torquati, Ilaria; Matthew O., Barrett; Kendal T., Harden; Mario, Grifantini
Design, synthesis and biological evaluation of novel inhibitors of NAD kinase
2012-01-01 Torquati, Ilaria; Vita, Patrizia; Petrelli, Riccardo; Di Stefano, M; Cappellacci, Loredana
PROBING BINDING REQUIREMENTS OF NAD KINASE WITH MODIFIED NAD ANALOGUES
2012-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krzysztof, Felczak; Palmarisa, Franchetti; Mario, Grifantini; Michele Di, Stefano; Giulio, Magni; Krzysztof W., Pankiewicz; Cappellacci, Loredana
Bisphosphonate Derivatives of 2’-C-Methyl-, and 3’-C-Methyl-Adenosine as Ligands at P2Y1 and P2Y2 Receptors
2012-01-01 Petrelli, Riccardo; Vita, Patrizia; Franchetti, P; Torquati, Ilaria; Barrett, O. M.; Harden, Kt; Grifantini, M; Cappellacci, Loredana
ADP- and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 receptor ligands
2012-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Jacobson, Ka; Barrett, Mo; Franklin, D; Harden, Kt; Franchetti, Palmarisa; Grifantini, Mario
5’-CHLORO-5’-DEOXY-N6-SUBSTITUTED ADENOSINE DERIVATIVES: SYNTHESIS, ADENOSINE RECEPTOR AFFINITY AND ANTINOCICEPTIVE ACTIVITY
2013-01-01 Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Luongo; K. N., Klotz; S., Kachler; F., Guida; M., De Chiaro; S., Maione; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana
NOVEL 2-SUBSTITUTED 2’/3’-C-METHYL-ADENOSINE DERIVATIVES: SYNTHESIS AND BIOLOGICAL EVALUATION AGAINST TRYPANOSOMA BRUCEI
2013-01-01 Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Boccoli; A., Hofer; M., Vodnala; P., Franchetti; M., Grifantini; Cappellacci, Loredana
Novel Inhibitors of Inosine Monophosphate Dehydrogenase in Patent Literature of the Last Decade
2013-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krysztof, Felczak; Daniel J., Wilson; Franchetti, Palmarisa; Cappellacci, Loredana
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE
2013-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; L., Luongo; F., Guida; M., De Chiaro; K. N., Klotz; S., Kachler; P., Franchetti; S., Maione; M., Grifantini; Cappellacci, Loredana
From the covalent linkage of drugs to novel inhibitors of ribonucleotide reductase: synthesis and biological evaluation of valproic esters of 3'-C-methyladenosine
2014-01-01 Petrelli, Riccardo; Maria, Meli; Vita, Patrizia; Torquati, Ilaria; Arianna, Ferro; Munender, Vodnala; Natale, D’Alessandro; Manlio, Tolomeo; DEL BELLO, Fabio; Praveen, Kusumanchi; Palmarisa, Franchetti; Mario, Grifantini; Hiremagalur N., Jayaram; Anders, Hofer; Cappellacci, Loredana
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE
2014-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Livio, Luongo; Francesca, Guida; Maria De, Chiaro; Karl Norbert, Klotz; Sonja, Kachler; Palmarisa, Franchetti; Sabatino, Maione; Mario, Grifantini; Cappellacci, Loredana
5’-deoxy-5’-N-pyrazolyl-N6-substituded adenosine derivates as A1 adenosine receptor agonists: synthesis and antinociception in mice
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Sonja, Kachler; Vita, Patrizia; Scortichini, Mirko; Antonio, Lavecchia; Sabatino, Maione; Karl Nornert, Klotz; Cappellacci, Loredana
Structure-Based Design, Synthesis and in vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists
2018-01-01 Petrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; DEL BELLO, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario | Poster atto convegno su volume | |
Synthesis and Enzymatic Evaluation of NAD Mimics as Nicotinamide Adenine Dinucleotide Kinase (NADK) Inhibitors | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Krzysztof, Felczak; Vita, Patrizia; Torquati, Ilaria; Palmarisa, Franchetti; Michele Di, Stefano; Giulio, Magni; Mario, Grifantini; Krzysztof W., Pankiewicz | Poster atto convegno su volume | |
Synthesis and biological activity of novel N6-substituted and 2,N6-disubstituted adenine ribo- and 3'-C-methyl-ribonucleosides as antitumor agents | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Franchetti, Palmarisa; Vita, Patrizia; Kusumanchi, P; Kumar, M; Jayaram, H. N.; Zhou, B; Yen, Y; Grifantini, Mario | Articolo | |
Synthesis and biological evaluation of (methylene)bisphosphonate derivatives of 2’-C-methyl-, and 3’-C-methyl-adenosine | 1-gen-2012 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Palmarisa, Franchetti; Torquati, Ilaria; Matthew O., Barrett; Kendal T., Harden; Mario, Grifantini | Poster atto convegno su volume | |
Design, synthesis and biological evaluation of novel inhibitors of NAD kinase | 1-gen-2012 | Torquati, Ilaria; Vita, Patrizia; Petrelli, Riccardo; Di Stefano, M; Cappellacci, Loredana | Contributo in atto di convegno su volume | |
PROBING BINDING REQUIREMENTS OF NAD KINASE WITH MODIFIED NAD ANALOGUES | 1-gen-2012 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krzysztof, Felczak; Palmarisa, Franchetti; Mario, Grifantini; Michele Di, Stefano; Giulio, Magni; Krzysztof W., Pankiewicz; Cappellacci, Loredana | Poster atto convegno su volume | |
Bisphosphonate Derivatives of 2’-C-Methyl-, and 3’-C-Methyl-Adenosine as Ligands at P2Y1 and P2Y2 Receptors | 1-gen-2012 | Petrelli, Riccardo; Vita, Patrizia; Franchetti, P; Torquati, Ilaria; Barrett, O. M.; Harden, Kt; Grifantini, M; Cappellacci, Loredana | Poster atto convegno su volume | |
ADP- and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 receptor ligands | 1-gen-2012 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Jacobson, Ka; Barrett, Mo; Franklin, D; Harden, Kt; Franchetti, Palmarisa; Grifantini, Mario | Contributo in atto di convegno su rivista | |
5’-CHLORO-5’-DEOXY-N6-SUBSTITUTED ADENOSINE DERIVATIVES: SYNTHESIS, ADENOSINE RECEPTOR AFFINITY AND ANTINOCICEPTIVE ACTIVITY | 1-gen-2013 | Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Luongo; K. N., Klotz; S., Kachler; F., Guida; M., De Chiaro; S., Maione; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana | Poster atto convegno su volume | |
NOVEL 2-SUBSTITUTED 2’/3’-C-METHYL-ADENOSINE DERIVATIVES: SYNTHESIS AND BIOLOGICAL EVALUATION AGAINST TRYPANOSOMA BRUCEI | 1-gen-2013 | Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Boccoli; A., Hofer; M., Vodnala; P., Franchetti; M., Grifantini; Cappellacci, Loredana | Poster atto convegno su volume | |
Novel Inhibitors of Inosine Monophosphate Dehydrogenase in Patent Literature of the Last Decade | 1-gen-2013 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krysztof, Felczak; Daniel J., Wilson; Franchetti, Palmarisa; Cappellacci, Loredana | Articolo | |
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE | 1-gen-2013 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; L., Luongo; F., Guida; M., De Chiaro; K. N., Klotz; S., Kachler; P., Franchetti; S., Maione; M., Grifantini; Cappellacci, Loredana | Poster atto convegno su volume | |
From the covalent linkage of drugs to novel inhibitors of ribonucleotide reductase: synthesis and biological evaluation of valproic esters of 3'-C-methyladenosine | 1-gen-2014 | Petrelli, Riccardo; Maria, Meli; Vita, Patrizia; Torquati, Ilaria; Arianna, Ferro; Munender, Vodnala; Natale, D’Alessandro; Manlio, Tolomeo; DEL BELLO, Fabio; Praveen, Kusumanchi; Palmarisa, Franchetti; Mario, Grifantini; Hiremagalur N., Jayaram; Anders, Hofer; Cappellacci, Loredana | Articolo | |
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE | 1-gen-2014 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Livio, Luongo; Francesca, Guida; Maria De, Chiaro; Karl Norbert, Klotz; Sonja, Kachler; Palmarisa, Franchetti; Sabatino, Maione; Mario, Grifantini; Cappellacci, Loredana | Poster atto convegno su rivista | |
5’-deoxy-5’-N-pyrazolyl-N6-substituded adenosine derivates as A1 adenosine receptor agonists: synthesis and antinociception in mice | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Sonja, Kachler; Vita, Patrizia; Scortichini, Mirko; Antonio, Lavecchia; Sabatino, Maione; Karl Nornert, Klotz; Cappellacci, Loredana | Poster atto convegno su volume | |
Structure-Based Design, Synthesis and in vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists | 1-gen-2018 | Petrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; DEL BELLO, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana | Articolo |
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