Sfoglia per Autore
STEREOSELECTIVE SYNTHESIS OF ISO-CARBOCYCLIC NUCLEOSIDE ANALOGUES AS POTENTIAL ANTIVIRAL DRUGS
2014-01-01 Torquati, Ilaria; Simon, Weising; Chris, Meier
5′-C-Ethyl-tetrazolyl-N6-Substituted Adenosine and 2-Chloro-adenosine Derivatives as Highly Potent Dual Acting A1 Adenosine Receptor Agonists and A3 Adenosine Receptor Antagonists
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Sonja, Kachler; Livio, Luongo; Sabatino, Maione; Palmarisa, Franchetti; Mario, Grifantini; Ettore, Novellino; Antonio, Lavecchia; Karl Norbert, Klotz; Cappellacci, Loredana
Design, Synthesis, and Anticancer Activity of Novel Pyridyl and Aryl Hydrazones
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Scortichini, Mirko; Grisogani, Federica; Angeloni, Yara; Girotti, Francesca; Brusseel, Marieke; Nabissi, Massimo; Santoni, Giorgio; Hofer, Anders; Ranjbarian, Farahnaz; Cappellacci, Loredana
5’-deoxy-5’-N-pyrazolyl-N6-substituded adenosine derivates as A1 adenosine receptor agonists: synthesis and antinociception in mice
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Sonja, Kachler; Vita, Patrizia; Scortichini, Mirko; Antonio, Lavecchia; Sabatino, Maione; Karl Nornert, Klotz; Cappellacci, Loredana
Novel N6/5’-Disubstituted Adenosine Derivatives As A1 Adenosine Receptor Agonists: Synthesis, Binding Assay And Antinociceptive Activity
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Luongo, Livio; Belardo, Carmela; Kachler, Sonja; Lavecchia, Antonio; Karl Norbert, Klotz; Maione, Sabatino; Cappellacci, Loredana
Synthesis and Biological Evaluations of Novel Arene Ru(II) Complexes of 4-acyl-5-pyrazolone-based Hydrazone Ligands
2015-01-01 Condello, Francesca; Palmucci, Jessica; Petrini, Agnese; Torquati, Ilaria; Petrelli, Riccardo; Cappellacci, Loredana; Hofer, Anders; Ranjbarian, Farahnaz; Pombeiro, A. J. L.; Lupidi, Giulio; Pettinari, Riccardo; Marchetti, Fabio; Pettinari, Claudio
c-di-GMP-based molecules as potent diguanylate cyclase (DGC) inhibitors
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Scortichini, Mirko; Rinaldo, Serena; Fernicola, Silvia; Giardina, Giorgio; Paiardini, Alessandro; Leoni, Livia; Rampioni, Giordano; Messina, Marco; Cutruzzolà, Francesca; Cappellacci, Loredana
4-acyl-5-pyrazolone-based hydrazones as novel anti-Trypanosoma brucei agents: structural design, synthesis and biological evaluation
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Scortichini, Mirko; DI GIOACCHINO, Valentina; Palumbo, Francesca; Bartelucci, Luca; Pettinari, Riccardo; Condello, Francesca; Pettinari, Claudio; Marchetti, Fabio; Hofer, Anders; Ranjbarian, Farahnaz; Cappellacci, Loredana
Allosteric control in the synthesis and sensing of cyclic-di-GMP
2015-01-01 Fernicola, Silvia; Rinaldo, Serena; Giardina, Giorgio; Brunotti, Paolo; Stelitano, Valentina; Paiardini, Alessandro; Petrelli, Riccardo; Torquati, Ilaria; Cappellacci, Loredana; Cutruzzolà, Francesca
Novel dual acting 5’-C-ethyl-tetrazolyl-N6-substituted adenosine derivatives: synthesis and biological evaluation
2015-01-01 Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Sonja, Kachler; Angeloni, Yara; Marieke, Brusseel; Antonio, Lavecchia; Sabatino, Maione; Karl Norbert, Klotz; Cappellacci, Loredana
Design, synthesis and biological evaluation of novel inhibitors of key enzymes in c-di-GMP metabolism as potential antibiofilm drugs
2015-03-20 Torquati, Ilaria
Exploring the Role of N6‐Substituents in Potent Dual Acting 5'‐C‐Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice
2017-01-01 Petrelli, Riccardo; Scortichini, Mirko; Kachler, Sonja; Boccella, Serena; Cerchia, Carmen; Torquati, Ilaria; DEL BELLO, Fabio; Salvemini, Daniela; Novellino, Ettore; Luongo, Livio; Maione, Sabatino; A Jacobson, Kenneth; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
STEREOSELECTIVE SYNTHESIS OF ISO-CARBOCYCLIC NUCLEOSIDE ANALOGUES AS POTENTIAL ANTIVIRAL DRUGS | 1-gen-2014 | Torquati, Ilaria; Simon, Weising; Chris, Meier | Poster atto convegno su volume | |
5′-C-Ethyl-tetrazolyl-N6-Substituted Adenosine and 2-Chloro-adenosine Derivatives as Highly Potent Dual Acting A1 Adenosine Receptor Agonists and A3 Adenosine Receptor Antagonists | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Sonja, Kachler; Livio, Luongo; Sabatino, Maione; Palmarisa, Franchetti; Mario, Grifantini; Ettore, Novellino; Antonio, Lavecchia; Karl Norbert, Klotz; Cappellacci, Loredana | Articolo | |
Design, Synthesis, and Anticancer Activity of Novel Pyridyl and Aryl Hydrazones | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Scortichini, Mirko; Grisogani, Federica; Angeloni, Yara; Girotti, Francesca; Brusseel, Marieke; Nabissi, Massimo; Santoni, Giorgio; Hofer, Anders; Ranjbarian, Farahnaz; Cappellacci, Loredana | Poster atto convegno su volume | |
5’-deoxy-5’-N-pyrazolyl-N6-substituded adenosine derivates as A1 adenosine receptor agonists: synthesis and antinociception in mice | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Sonja, Kachler; Vita, Patrizia; Scortichini, Mirko; Antonio, Lavecchia; Sabatino, Maione; Karl Nornert, Klotz; Cappellacci, Loredana | Poster atto convegno su volume | |
Novel N6/5’-Disubstituted Adenosine Derivatives As A1 Adenosine Receptor Agonists: Synthesis, Binding Assay And Antinociceptive Activity | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Luongo, Livio; Belardo, Carmela; Kachler, Sonja; Lavecchia, Antonio; Karl Norbert, Klotz; Maione, Sabatino; Cappellacci, Loredana | Poster atto convegno su volume | |
Synthesis and Biological Evaluations of Novel Arene Ru(II) Complexes of 4-acyl-5-pyrazolone-based Hydrazone Ligands | 1-gen-2015 | Condello, Francesca; Palmucci, Jessica; Petrini, Agnese; Torquati, Ilaria; Petrelli, Riccardo; Cappellacci, Loredana; Hofer, Anders; Ranjbarian, Farahnaz; Pombeiro, A. J. L.; Lupidi, Giulio; Pettinari, Riccardo; Marchetti, Fabio; Pettinari, Claudio | Poster atto convegno su volume | |
c-di-GMP-based molecules as potent diguanylate cyclase (DGC) inhibitors | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Scortichini, Mirko; Rinaldo, Serena; Fernicola, Silvia; Giardina, Giorgio; Paiardini, Alessandro; Leoni, Livia; Rampioni, Giordano; Messina, Marco; Cutruzzolà, Francesca; Cappellacci, Loredana | Poster atto convegno su volume | |
4-acyl-5-pyrazolone-based hydrazones as novel anti-Trypanosoma brucei agents: structural design, synthesis and biological evaluation | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Scortichini, Mirko; DI GIOACCHINO, Valentina; Palumbo, Francesca; Bartelucci, Luca; Pettinari, Riccardo; Condello, Francesca; Pettinari, Claudio; Marchetti, Fabio; Hofer, Anders; Ranjbarian, Farahnaz; Cappellacci, Loredana | Poster atto convegno su volume | |
Allosteric control in the synthesis and sensing of cyclic-di-GMP | 1-gen-2015 | Fernicola, Silvia; Rinaldo, Serena; Giardina, Giorgio; Brunotti, Paolo; Stelitano, Valentina; Paiardini, Alessandro; Petrelli, Riccardo; Torquati, Ilaria; Cappellacci, Loredana; Cutruzzolà, Francesca | Poster atto convegno su volume | |
Novel dual acting 5’-C-ethyl-tetrazolyl-N6-substituted adenosine derivatives: synthesis and biological evaluation | 1-gen-2015 | Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Sonja, Kachler; Angeloni, Yara; Marieke, Brusseel; Antonio, Lavecchia; Sabatino, Maione; Karl Norbert, Klotz; Cappellacci, Loredana | Poster atto convegno su volume | |
Design, synthesis and biological evaluation of novel inhibitors of key enzymes in c-di-GMP metabolism as potential antibiofilm drugs | 20-mar-2015 | Torquati, Ilaria | Doctoral Thesis | |
Exploring the Role of N6‐Substituents in Potent Dual Acting 5'‐C‐Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice | 1-gen-2017 | Petrelli, Riccardo; Scortichini, Mirko; Kachler, Sonja; Boccella, Serena; Cerchia, Carmen; Torquati, Ilaria; DEL BELLO, Fabio; Salvemini, Daniela; Novellino, Ettore; Luongo, Livio; Maione, Sabatino; A Jacobson, Kenneth; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana | Articolo |
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