Sfoglia per Autore
Synthesis and dopamine receptor affinities of 6-amino-5,6,7,8-tetrahydroquinoline derivatives
1989-01-01 Claudi, Francesco; Cingolani, Gian Mario; Giorgioni, Gianfabio; F., Cattabeni; M., Cimino; M., DI LUCA
Synthesis and Pharmacological Characterization of 2-(4-Chloro-3-hydroxyphenyl)ethylamine and N,N-dialkyl Derivatives as Dopamine Receptor Ligands
1992-01-01 Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; M. P., Abbracchio; A. M., Paoletti; W., Balduini
Structure-Activity Relationships of N-n-Propyl-2-(4-fluoro-3-hydroxyphenyl)ethylamine Derivatives as Dopamine Receptor Ligands
1992-01-01 Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; F., Reno'; W., Balduini
Synthesis and Evaluation of N-n-Propyl-N-(2-phenylethyl)-2-(3-fluoro-4- hydroxyphenyl)ethylamine Derivatives as Dopamine Receptor Ligands
1992-01-01 Claudi, Francesco; Cingolani, Gian Mario; A., DI STEFANO; Giorgioni, Gianfabio; A., Cagnotto; M., Skorupska
A Comparative Behavioural Analysis in Rats of the D2 Agonist RU 24213 and Two New Structurally Similar Compounds
1993-01-01 F., Ferrari; Claudi, Francesco; Giorgioni, Gianfabio; D., Giuliani
Synthesis and Dopamine Receptor Binding of 4-(2-Aminoethyl)-1H-pyrazole and Its N,N- Dialkyl Derivatives
1993-01-01 Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; A., Cagnotto; M., Skorupska
Synthesis and Evaluation of 2-(5-Methoxythiophen-3- yl)ethylamines as Potential Dopamine Agonists
1994-01-01 Cardellini, Mario; Cingolani, Gian Mario; Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; Cantalamessa, Franco; A., Cagnotto; M., Skorupska
Activity of N-(2-Phenylethyl)-N-n-Propyl-2-(3-Hydroxyphenyl)ethylamine Derivatives as Dopamine Receptor Ligands
1994-01-01 Claudi, Francesco; Cardellini, Mario; A., DI STEFANO; Giorgioni, Gianfabio; Cantalamessa, Franco; F., Reno'; W., Balduini
New 2- pyridylethylamines with dopaminergic activity: synthesis and radioligand binding evaluation
1995-01-01 Claudi, Francesco; Giorgioni, Gianfabio; Cardellini, Mario; Amenta, Francesco; Polidori, Carlo
New Systems for the Specific Delivery and Sustained Release of Dopamine to the Brain
1996-01-01 V., Carelli; F., Liberatore; L., Scipione; M., Impicciatore; E., Barocelli; Cardellini, Mario; Giorgioni, Gianfabio
Synthesis, resolution and preliminary evaluation of trans-2-amino-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes and related derivatives as dopamine receptor ligands
1996-01-01 Claudi, Francesco; Cingolani, Gm; DI STEFANO, A; Giorgioni, Gianfabio; Amenta, Francesco; Barili, Paolo; Ferrari, F; Giuliani, D.
A de novo design probe of a dopamine receptor ligand based on a theoretical approach
1996-01-01 M., Baginski; Claudi, Francesco; Giorgioni, Gianfabio; J. A., Fontenla; E., Rosa; Cardellini, Mario
3-[2-[4-(4-Fluorobenzoyl)piperidin-1-yl]ethyl]-5,6,7,8-tetrahydro-4(3H)quinazolinones: serotonin 5-HT2A receptor antagonists endowed with potent, central action
1997-01-01 Claudi, Francesco; Giorgioni, Gianfabio; Scoccia, L; Ciccocioppo, Roberto; Panocka, I; Massi, Maurizio
Simplified analogues of Ritanserin and their affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors
1998-01-01 Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Marucci, Gabriella; DI STEFANO, A.; Gessi, S.; Siniscalchi, A.; Borea, P. A.
4-(4-Fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2c serotonin receptors
1999-01-01 Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Accorroni, Beatrice; Marucci, Gabriella; Gessi, S; Siniscalchi, A; Borea, Pa
Synthesis of L-(+)-3-(3-hydroxy-4-pivaloyloxybenzyl)-2,5-diketomorpholine as potential prodrug of L-Dopa
2000-01-01 Cingolani, Gian Mario; DI STEFANO, A.; Mosciatti, B.; Napolitani, F.; Giorgioni, Gianfabio; Ricciutelli, Massimo; Claudi, Francesco
Binding and preliminary evaluation of 5-hydroxy- and 10-hydroxy-2,3,12,12a-tetrahydro-1H-[1]benzoxepino[2,3,4-ij]isoquinoles as dopamine receptor ligands
2000-01-01 Claudi, Francesco; DI STEFANO, A.; Napolitani, F.; Cingolani, Gian Mario; Giorgioni, Gianfabio; Fontenla, J. A.; Montenegro, G. Y.; Rivas, M. E.; Rosa, E.; Michelotto, B.; Orlando, G.; Brunetti, L.
Synthesis and Preliminary Pharmacological Evaluation of 5-Hydroxy- and 5,6-Dihydroxy-1,2,3,7,12,12a-hexahydrobenzo [5,6]cyclohepta[1,2,3-ij]isoquinoline Derivatives as Dopamine Receptor Ligands
2001-01-01 Cingolani, Gian Mario; DI STEFANO, A.; Napolitani, F.; Mosciatti, B.; Giorgioni, Gianfabio; Cinone, N.; Brunetti, L.; Luisi, G.; Michelotto, B.; Orlando, G.; Costa, B.; Lucacchini, A.; Martini, C.; Claudi, Francesco
Dimeric L-Dopa Derivatives as Potential Prodrugs
2001-01-01 DI STEFANO, A.; Mosciatti, B.; Cingolani, Gian Mario; Giorgioni, Gianfabio; Ricciutelli, Massimo; Cacciatore, I.; Sozio, P.; Claudi, Francesco
Synthesis and Biological Evaluation of GABA Derivatives Able to Cross the Blood -Brain Barrier in Rats
2003-01-01 Carelli, V; Liberatore, F; Scipione, L; Giorgioni, Gianfabio; DI STEFANO, A; Impicciatore, M; Ballabeni, V; Calcina, F; Magnanini, F; Barocelli, E.
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Synthesis and dopamine receptor affinities of 6-amino-5,6,7,8-tetrahydroquinoline derivatives | 1-gen-1989 | Claudi, Francesco; Cingolani, Gian Mario; Giorgioni, Gianfabio; F., Cattabeni; M., Cimino; M., DI LUCA | Articolo | |
Synthesis and Pharmacological Characterization of 2-(4-Chloro-3-hydroxyphenyl)ethylamine and N,N-dialkyl Derivatives as Dopamine Receptor Ligands | 1-gen-1992 | Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; M. P., Abbracchio; A. M., Paoletti; W., Balduini | Articolo | |
Structure-Activity Relationships of N-n-Propyl-2-(4-fluoro-3-hydroxyphenyl)ethylamine Derivatives as Dopamine Receptor Ligands | 1-gen-1992 | Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; F., Reno'; W., Balduini | Articolo | |
Synthesis and Evaluation of N-n-Propyl-N-(2-phenylethyl)-2-(3-fluoro-4- hydroxyphenyl)ethylamine Derivatives as Dopamine Receptor Ligands | 1-gen-1992 | Claudi, Francesco; Cingolani, Gian Mario; A., DI STEFANO; Giorgioni, Gianfabio; A., Cagnotto; M., Skorupska | Articolo | |
A Comparative Behavioural Analysis in Rats of the D2 Agonist RU 24213 and Two New Structurally Similar Compounds | 1-gen-1993 | F., Ferrari; Claudi, Francesco; Giorgioni, Gianfabio; D., Giuliani | Articolo | |
Synthesis and Dopamine Receptor Binding of 4-(2-Aminoethyl)-1H-pyrazole and Its N,N- Dialkyl Derivatives | 1-gen-1993 | Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; A., Cagnotto; M., Skorupska | Articolo | |
Synthesis and Evaluation of 2-(5-Methoxythiophen-3- yl)ethylamines as Potential Dopamine Agonists | 1-gen-1994 | Cardellini, Mario; Cingolani, Gian Mario; Claudi, Francesco; Giorgioni, Gianfabio; A., DI STEFANO; Cantalamessa, Franco; A., Cagnotto; M., Skorupska | Articolo | |
Activity of N-(2-Phenylethyl)-N-n-Propyl-2-(3-Hydroxyphenyl)ethylamine Derivatives as Dopamine Receptor Ligands | 1-gen-1994 | Claudi, Francesco; Cardellini, Mario; A., DI STEFANO; Giorgioni, Gianfabio; Cantalamessa, Franco; F., Reno'; W., Balduini | Articolo | |
New 2- pyridylethylamines with dopaminergic activity: synthesis and radioligand binding evaluation | 1-gen-1995 | Claudi, Francesco; Giorgioni, Gianfabio; Cardellini, Mario; Amenta, Francesco; Polidori, Carlo | Articolo | |
New Systems for the Specific Delivery and Sustained Release of Dopamine to the Brain | 1-gen-1996 | V., Carelli; F., Liberatore; L., Scipione; M., Impicciatore; E., Barocelli; Cardellini, Mario; Giorgioni, Gianfabio | Articolo | |
Synthesis, resolution and preliminary evaluation of trans-2-amino-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes and related derivatives as dopamine receptor ligands | 1-gen-1996 | Claudi, Francesco; Cingolani, Gm; DI STEFANO, A; Giorgioni, Gianfabio; Amenta, Francesco; Barili, Paolo; Ferrari, F; Giuliani, D. | Articolo | |
A de novo design probe of a dopamine receptor ligand based on a theoretical approach | 1-gen-1996 | M., Baginski; Claudi, Francesco; Giorgioni, Gianfabio; J. A., Fontenla; E., Rosa; Cardellini, Mario | Articolo | |
3-[2-[4-(4-Fluorobenzoyl)piperidin-1-yl]ethyl]-5,6,7,8-tetrahydro-4(3H)quinazolinones: serotonin 5-HT2A receptor antagonists endowed with potent, central action | 1-gen-1997 | Claudi, Francesco; Giorgioni, Gianfabio; Scoccia, L; Ciccocioppo, Roberto; Panocka, I; Massi, Maurizio | Articolo | |
Simplified analogues of Ritanserin and their affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors | 1-gen-1998 | Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Marucci, Gabriella; DI STEFANO, A.; Gessi, S.; Siniscalchi, A.; Borea, P. A. | Articolo | |
4-(4-Fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2c serotonin receptors | 1-gen-1999 | Claudi, Francesco; Scoccia, Loredana; Giorgioni, Gianfabio; Accorroni, Beatrice; Marucci, Gabriella; Gessi, S; Siniscalchi, A; Borea, Pa | Articolo | |
Synthesis of L-(+)-3-(3-hydroxy-4-pivaloyloxybenzyl)-2,5-diketomorpholine as potential prodrug of L-Dopa | 1-gen-2000 | Cingolani, Gian Mario; DI STEFANO, A.; Mosciatti, B.; Napolitani, F.; Giorgioni, Gianfabio; Ricciutelli, Massimo; Claudi, Francesco | Articolo | |
Binding and preliminary evaluation of 5-hydroxy- and 10-hydroxy-2,3,12,12a-tetrahydro-1H-[1]benzoxepino[2,3,4-ij]isoquinoles as dopamine receptor ligands | 1-gen-2000 | Claudi, Francesco; DI STEFANO, A.; Napolitani, F.; Cingolani, Gian Mario; Giorgioni, Gianfabio; Fontenla, J. A.; Montenegro, G. Y.; Rivas, M. E.; Rosa, E.; Michelotto, B.; Orlando, G.; Brunetti, L. | Articolo | |
Synthesis and Preliminary Pharmacological Evaluation of 5-Hydroxy- and 5,6-Dihydroxy-1,2,3,7,12,12a-hexahydrobenzo [5,6]cyclohepta[1,2,3-ij]isoquinoline Derivatives as Dopamine Receptor Ligands | 1-gen-2001 | Cingolani, Gian Mario; DI STEFANO, A.; Napolitani, F.; Mosciatti, B.; Giorgioni, Gianfabio; Cinone, N.; Brunetti, L.; Luisi, G.; Michelotto, B.; Orlando, G.; Costa, B.; Lucacchini, A.; Martini, C.; Claudi, Francesco | Articolo | |
Dimeric L-Dopa Derivatives as Potential Prodrugs | 1-gen-2001 | DI STEFANO, A.; Mosciatti, B.; Cingolani, Gian Mario; Giorgioni, Gianfabio; Ricciutelli, Massimo; Cacciatore, I.; Sozio, P.; Claudi, Francesco | Articolo | |
Synthesis and Biological Evaluation of GABA Derivatives Able to Cross the Blood -Brain Barrier in Rats | 1-gen-2003 | Carelli, V; Liberatore, F; Scipione, L; Giorgioni, Gianfabio; DI STEFANO, A; Impicciatore, M; Ballabeni, V; Calcina, F; Magnanini, F; Barocelli, E. | Articolo |
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