Sfoglia per Autore
“Enantiomers of 8-(tert-butylamino-2-hydroxypropoxy) 3,4-dihydro-3-oxo-2H-(1,4) Benzothiazine: Racemic Resolution, Chiral Synthesis and Biological Activity“.
1990-01-01 Schiaffella, F; Fringuelli, R; Cecchetti, V; Fravolini, A; Angeli, Piero; Marucci, Gabriella
Determination of Muscarinic Agonist Potencies at M1 and M2 Muscarinic Receptors in a Modified Pithed rat Preparation
1990-01-01 Angeli, Piero; Brasili, L; Cantalamessa, Franco; Marucci, Gabriella; Wess, J.
“Pharmacological Characterization of Muscarinic Receptor Subtypes in Rabbit Isolated Tissue Preparations”
1991-01-01 Angeli, Piero; Brasili, L; Cingolani, M. L.; Marucci, Gabriella; Pigini, Maria; Tonnini, M. C.
“Methoctramine-Related Polymethylene Tetraamines”. 4(1)-Chirality Effect on M2 Muscarinic Receptor Blocking Activity.
1991-01-01 Giardinà, D; Marrazzo, A; Marucci, Gabriella; Piloni, M. G.; Quaglia, Wilma
“Structure-Activity Relationships Among Methoctramine Related Polymethylene Tetraamines. Effect of the Four Nitrogens on M2 Muscarinic Blocking Activity as Revealed by Symmetrical and Unsymmetrical Polyamines”.
1991-01-01 Quaglia, Wilma; Melchiorre, C; Giardinà, D; Marucci, Gabriella; Minarini, A; Tumiatti, V.
“Synthesis and Pharmacological Activity of Some New Pyridazinones”.
1992-01-01 Corsano, S; Strappaghetti, G; Codagnone, A; Scapicchi, R; Marucci, Gabriella
. “Synthesis, Pharmacological “Evaluation and Selectivity Profile of Isomeric 2-Phenyl-2-Cyclohexyl-4-[(Dimethylamino)Methyl]-1,3-Dithiolane Methiodides, as Potent Antimuscarinic Agents”.
1992-01-01 Angeli, Piero; Brasili, L; Gulini, U; Paparelli, F; Marucci, Gabriella
“Stereoselectivity at α-Adrenoreceptor Subtypes: Observations With the enantiomers of WB 4101 Separated Through Their Amides of N-Tosyl-(S)-Proline”.
1992-01-01 Andrisano, V; Marucci, Gabriella; Melchiorre, C; AND TUMIATTI, V.
“Synthesis and Pharmacological Evaluation of Enantiomerically Pure 4-Deoxy-4-Fluoro-Muscarines”.
1992-01-01 Bravo, P; Resnati, G; Angeli, Piero; Frigerio, M; Viani, F; Arnone, A; Marucci, Gabriella; Cantalamessa, Franco
“Pharmacological Characterization of Chiral Muscarinic Antagonists cis -2- phenyl-2- cyclohexyl-r-5-[(dimethylamino)-methyl]-1,3-oxathiolane-3-Oxide methiodides”.
1992-01-01 Angeli, Piero; Balduini, W; Brasili, L; Cantalamessa, Franco; Cattabeni, F; Marucci, Gabriella
“New Pyridazinones: Synthesis and Correlation Between Structure and α-Blocking Activity”.
1993-01-01 Corsano, S; Scapicchi, R; Strappaghetti, G; Marucci, Gabriella; Paparelli, F.
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 4. Effect of aryl and alkyl Substituents at Position 3 on α-adrenoreceptor blocking activity
1993-01-01 Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Melchiorre, C.
“N,N-diethylaminoethanol and N-methyl-4-piperidinol Esters of 2,2-diphenyl-2-Ethylthioacetic Acid as Potent and Selective Muscarinic Antagonist”.
1993-01-01 Scapecchi, S; Angeli, Piero; Dei, S; Gualtieri, F; Marucci, Gabriella; Romanelli, M. N.; Teodori, E.
“1,3 Oxathiolane Muscarinic Ligands Modified at the Cationic Head”.
1994-01-01 Teodori, E; Dei, S; Romanelli, M. N.; Scapecchi, S; Gualtieri, F; Angeli, Piero; Marucci, Gabriella; Matucci, R.
“Dialkylaminoalkyl Esters of 2,2 Diphenyl-2-Alkylthioacetic Acids: A New Class of Potent and Functionally Selective Muscarinic Antagonists”.
1994-01-01 Scapecchi, S; Angeli, Piero; Dei, S; Gualtieri, F; Marucci, Gabriella; Moriconi, R; Paparelli, F; Romanelli, M. N.; Teodori, E.
“Novel and Highly Selective Postsynaptic α-Adrenoreceptor Antagonists: Synthesis and Structure-Activity Relationships of Alkane-Bridged [4-(phenoxyethyl)-1-piperazinyl]-3 (2H)-pyridazinones”.
1995-01-01 Corsano, S; Scapicchi, R; Strappaghetti, G; Paparelli, F; Marucci, Gabriella
Separation of alpha-adrenergic and imidazoline/guanidinium receptive sites (IGRS) activity in a series of imidazoline analogues of cirazoline
1995-01-01 Brasili, L.; Pigini, Maria; Marucci, Gabriella; Quaglia, Wilma; Malmusi, L.; Lanier, S. M.; Lanier, B.
“Synthesis and α-Adrenoreceptor Blocking Properties of Phenoxybenzamine-Related (2-Chloroethyl)-(2,3-dihydrobenzo-[1,4] dioxin-2-ylmethyl)-(2-phenoxyethyl) Amines”.
1995-01-01 Giardinà, D; Crucianelli, M; Marucci, Gabriella; Paparelli, F; Melchiorre, C.
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 5. Effects of Modification of the side chain on alpha-adrenoreceptor blocking Activity
1996-01-01 Quaglia, Wilma; Giannella, Mario; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Tayebati, Seyed Khosrow; Melchiorre, C.
“Tetraamines as Lead Compounds for the “Pharmacological Evaluation of Prazosin and Doxazosin-related Compounds with Modified Piperazine Ring”.
1996-01-01 Giardinà, D; Crucianelli, M; Marucci, Gabriella; Melchiorre, C; Polidori, Carlo; Pompei, Pierluigi; Massi, Maurizio
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