Sfoglia per Autore
Molecular modeling study on potent and selective adenosine A3 receptor agonists.
2010-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria
Neuropeptide S Receptor: recent updates on non-peptide antagonist discovery
2011-01-01 DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria
Evidence for the existence of a specific G protein-coupled receptor activated by guanosine
2011-01-01 Volpini, Rosaria; Marucci, Gabriella; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Mishra, Cr; Thomas, Ajiroghene; Cristalli, Gloria
Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17
2011-01-01 Buccioni, Michela; Marucci, Gabriella; DAL BEN, Diego; Giacobbe, Dania; Lambertucci, Catia; Soverchia, Laura; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria
Innovative functional cAMP assay: application to the pharmacological characterization of GPR17
2012-01-01 Marucci, Gabriella; Buccioni, Michela; Ceruti, S; DAL BEN, Diego; Giacobbe, D; Lambertucci, Catia; Lecca, D; Thomas, Ajiroghene; Volpini, Rosaria; Abbracchio, Mp; Cristalli, Gloria
Functional cAMP assay optimization at CHO cells expressing A2A adenosine receptors and stably transfected with firefly luciferase biosensor
2012-01-01 Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Giacobbe, D; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Simulation and comparative analysis of binding modes of nucleoside and non-nucleoside agonists at the A2B adenosine receptor
2013-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Thomas, Ajiroghene; Volpini, Rosaria
Evaluation of adenine as scaffold for the development of novel P2X3 receptor antagonists
2013-01-01 Lambertucci, Catia; Sundukova, M; Kachare, Dd; Panmand, Ds; DAL BEN, Diego; Buccioni, Michela; Marucci, Gabriella; Marchenkova, A; Thomas, Ajiroghene; Nistri, A; Cristalli, Gloria; Volpini, Rosaria
8-(2-Furyl)adenine derivatives as A2A adenosine receptor ligands
2013-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Thomas, Ajiroghene; K. N., Klotz; S., Federico; B., Cacciari; G., Spalluto; Volpini, Rosaria
Synthesis of ligands for receptors involved in neurodegeneration
2013-03-25 Thomas, Ajiroghene
Purinergic P2X receptors: Structural models and analysis of receptor-ligand interaction
2014-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Thomas, Ajiroghene; Marucci, Gabriella; Volpini, Rosaria
Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: Insight into the receptor activation switch
2014-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Kachler, S; Falgner, N; Marucci, Gabriella; Thomas, Ajiroghene; Cristalli, Gloria; Volpini, Rosaria; Klotz, K. N.
Antiproliferative Evaluation of Isofuranodiene on Breast and Prostate Cancer Cell Lines
2014-01-01 Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Maggi, Filippo; Papa, Fabrizio; Thomas, Ajiroghene; Santinelli, Claudia; Marucci, Gabriella
Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation
2015-01-01 Flavia, Varano; Daniela, Catarzi; Lucia, Squarcialupi; Marco, Betti; Fabrizio, Vincenzi; Annalisa, Ravani; Katia, Varani; DAL BEN, Diego; Thomas, Ajiroghene; Volpini, Rosaria; Vittoria, Colotta
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies
2015-01-01 Daniela, Catarzi; Flavia, Varano; Daniela, Poli; Lucia, Squarcialupi; Marco, Betti; Letizia, Trincavelli; Claudia, Martini; DAL BEN, Diego; Thomas, Ajiroghene; Volpini, Rosaria; Vittoria, Colotta
Medicinal Chemistry of P2X Receptors: Agonists and Orthosteric Antagonists
2015-01-01 Lambertucci, Catia; DAL BEN, Diego; Buccioni, Michela; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria
New substituted 9-propyladenine derivatives as A2Aadenosine receptor antagonists
2015-01-01 Lambertucci, Catia; Buccioni, Michela; DAL BEN, Diego; Sonia, Kachler; Marucci, Gabriella; Spinaci, Andrea; Thomas, Ajiroghene; Karl Norbert, Klotz; Volpini, Rosaria
Purinergic P2X receptors: Structural models and analysis of ligand-target interaction
2015-01-01 DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria
33rd camerino-Cyprus Symposium - Receptor Chemistry: Reality and Vision
2016-01-01 Angeli, Piero; DEL BELLO, Fabio; Giannella, Mario; Caprioli, Giovanni; Giorgioni, Gianfabio; Piergentili, Alessandro; Petrelli, Riccardo; Quaglia, Wilma; Thomas, Ajiroghene; Mavromoustakos, Thomas; Tsotinis, Andreas
The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor
2016-01-01 Thomas, Ajiroghene; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Santinelli, Claudia; Spinaci, Andrea; Kachler, S.; Klotz, K. N.; Volpini, Rosaria
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Molecular modeling study on potent and selective adenosine A3 receptor agonists. | 1-gen-2010 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Neuropeptide S Receptor: recent updates on non-peptide antagonist discovery | 1-gen-2011 | DAL BEN, Diego; Antonini, Ippolito; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Evidence for the existence of a specific G protein-coupled receptor activated by guanosine | 1-gen-2011 | Volpini, Rosaria; Marucci, Gabriella; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Lammi, C; Mishra, Cr; Thomas, Ajiroghene; Cristalli, Gloria | Articolo | |
Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17 | 1-gen-2011 | Buccioni, Michela; Marucci, Gabriella; DAL BEN, Diego; Giacobbe, Dania; Lambertucci, Catia; Soverchia, Laura; Thomas, Ajiroghene; Volpini, Rosaria; Cristalli, Gloria | Articolo | |
Innovative functional cAMP assay: application to the pharmacological characterization of GPR17 | 1-gen-2012 | Marucci, Gabriella; Buccioni, Michela; Ceruti, S; DAL BEN, Diego; Giacobbe, D; Lambertucci, Catia; Lecca, D; Thomas, Ajiroghene; Volpini, Rosaria; Abbracchio, Mp; Cristalli, Gloria | Abstract atto convegno su rivista | |
Functional cAMP assay optimization at CHO cells expressing A2A adenosine receptors and stably transfected with firefly luciferase biosensor | 1-gen-2012 | Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Giacobbe, D; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Abstract atto convegno su rivista | |
Simulation and comparative analysis of binding modes of nucleoside and non-nucleoside agonists at the A2B adenosine receptor | 1-gen-2013 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Thomas, Ajiroghene; Volpini, Rosaria | Articolo | |
Evaluation of adenine as scaffold for the development of novel P2X3 receptor antagonists | 1-gen-2013 | Lambertucci, Catia; Sundukova, M; Kachare, Dd; Panmand, Ds; DAL BEN, Diego; Buccioni, Michela; Marucci, Gabriella; Marchenkova, A; Thomas, Ajiroghene; Nistri, A; Cristalli, Gloria; Volpini, Rosaria | Articolo | |
8-(2-Furyl)adenine derivatives as A2A adenosine receptor ligands | 1-gen-2013 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Thomas, Ajiroghene; K. N., Klotz; S., Federico; B., Cacciari; G., Spalluto; Volpini, Rosaria | Articolo | |
Synthesis of ligands for receptors involved in neurodegeneration | 25-mar-2013 | Thomas, Ajiroghene | Doctoral Thesis | |
Purinergic P2X receptors: Structural models and analysis of receptor-ligand interaction | 1-gen-2014 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Thomas, Ajiroghene; Marucci, Gabriella; Volpini, Rosaria | Abstract atto convegno su rivista | |
Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: Insight into the receptor activation switch | 1-gen-2014 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Kachler, S; Falgner, N; Marucci, Gabriella; Thomas, Ajiroghene; Cristalli, Gloria; Volpini, Rosaria; Klotz, K. N. | Articolo | |
Antiproliferative Evaluation of Isofuranodiene on Breast and Prostate Cancer Cell Lines | 1-gen-2014 | Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Maggi, Filippo; Papa, Fabrizio; Thomas, Ajiroghene; Santinelli, Claudia; Marucci, Gabriella | Articolo | |
Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation | 1-gen-2015 | Flavia, Varano; Daniela, Catarzi; Lucia, Squarcialupi; Marco, Betti; Fabrizio, Vincenzi; Annalisa, Ravani; Katia, Varani; DAL BEN, Diego; Thomas, Ajiroghene; Volpini, Rosaria; Vittoria, Colotta | Articolo | |
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies | 1-gen-2015 | Daniela, Catarzi; Flavia, Varano; Daniela, Poli; Lucia, Squarcialupi; Marco, Betti; Letizia, Trincavelli; Claudia, Martini; DAL BEN, Diego; Thomas, Ajiroghene; Volpini, Rosaria; Vittoria, Colotta | Articolo | |
Medicinal Chemistry of P2X Receptors: Agonists and Orthosteric Antagonists | 1-gen-2015 | Lambertucci, Catia; DAL BEN, Diego; Buccioni, Michela; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria | Articolo | |
New substituted 9-propyladenine derivatives as A2Aadenosine receptor antagonists | 1-gen-2015 | Lambertucci, Catia; Buccioni, Michela; DAL BEN, Diego; Sonia, Kachler; Marucci, Gabriella; Spinaci, Andrea; Thomas, Ajiroghene; Karl Norbert, Klotz; Volpini, Rosaria | Articolo | |
Purinergic P2X receptors: Structural models and analysis of ligand-target interaction | 1-gen-2015 | DAL BEN, Diego; Buccioni, Michela; Lambertucci, Catia; Marucci, Gabriella; Thomas, Ajiroghene; Volpini, Rosaria | Articolo | |
33rd camerino-Cyprus Symposium - Receptor Chemistry: Reality and Vision | 1-gen-2016 | Angeli, Piero; DEL BELLO, Fabio; Giannella, Mario; Caprioli, Giovanni; Giorgioni, Gianfabio; Piergentili, Alessandro; Petrelli, Riccardo; Quaglia, Wilma; Thomas, Ajiroghene; Mavromoustakos, Thomas; Tsotinis, Andreas | Cura di atti, volumi e cataloghi | |
The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor | 1-gen-2016 | Thomas, Ajiroghene; Buccioni, Michela; DAL BEN, Diego; Lambertucci, Catia; Marucci, Gabriella; Santinelli, Claudia; Spinaci, Andrea; Kachler, S.; Klotz, K. N.; Volpini, Rosaria | Articolo |
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