Sfoglia per Autore
First TiCl4-Mediated Diastereoslective Reduction of alpha-Nitro Ketones to beta-Nitro Alcohols by BH3.SMe2
2000-01-01 Ballini, Roberto; Bosica, Giovanna; Marcantoni, Enrico; Vita, Patrizia; Bartoli, G.
Stereoselective synthesis of nicotinamide β-riboside and nucleoside analogs
2004-01-01 Franchetti, Palmarisa; Pasqualini, M.; Petrelli, Riccardo; Ricciutelli, Massimo; Vita, Patrizia; Cappellacci, Loredana
3’-C-Methyl-ribosyl nucleosides as cytotoxic compounds
2005-01-01 Cappellacci, L.; Franchetti, P.; Grifantini, M.; Pasqualini, M.; Petrelli, R.; Vita, P.; Jayaram, H.; Horvath, Z.; Szekeres, T.
Affinity and selectivity of tecadenoson, 2-chloro-tecadenoson and 2’-C-methyl analogues at bovine and pig A1 adenosine receptor
2005-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M.; Costa, B.; Spinetti, F.; Martini, C.; Klotz, K.; Lavecchia, A.
Synthesis and Biological Evaluation of NAD Analogs as Human Pyridine Nucleotide Adenylyltransferase Inhibitors
2005-01-01 Franchetti, Palmarisa; Petrelli, Riccardo; Cappellacci, Loredana; Pasqualini, M.; Vita, Patrizia; Sorci, L.; Mazzola, F.; Raffaelli, N.; Magni, G.
Ribose-modified mizoribine analogues: synthesis and biological evaluation
2005-01-01 Franchetti, Palmarisa; Pasqualini, M.; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Jayaram, H. N.
Structure-affinity relathionships of 5'-carbamoyl- and 5'-thionocarbamoyl derivatives of the A1 selective adenosine receptor agonist 2'-MeCCPA as partial A1 agonists
2005-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; B., Costa; C., Martini; A., Lavecchia; Kn, Klotz; Grifantini, Mario
2’-C-Methyl derivatives of tecadenoson and 2-chloro-tecadenoson with increased selectivity for human A1 adenosine receptor
2006-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M; Costa, B; Spinetti, F; Martini, C; Klotz, K. N.; Lavecchia, A; Grifantini, Mario
Purine and pyrimidine nucleoside analogs of 3'-C-methyladenosine as antitumor agents
2006-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Riccioni, S.; Vita, Patrizia; Jayaram, H. N.; Grifantini, Mario
Inhibition of HIV-1 replication in macrophages by red blood cell-mediated delivery of a heterodinucleotide of lamivudine and tenofovir
2007-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Rossi, L.; Pierige', F.; Serafini, S.; Magnani, M.; Balestra, E.; Perno, C. F.
ATP-mimetics derived from 2 '(3 ')-C-methyladenosine as human P2Y2 agonists
2008-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Vita, Patrizia; Jacobson, K. A.; Maddileti, S.; Harden, T. K.; Grifantini, Mario
Synthesis and antitumor activity of a heterodinucleotide of BVDU and Gemcitabine
2008-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario
5'-Chloro-5'-deoxy-N6-(±)-endo-norbornyladenosine, a potent and highly selective human A1 adenosine receptor agonist modulates neuropathic pain in mice.
2009-01-01 Livio, Luongo; Cappellacci, Loredana; Enza, Palazzo; Claudia, Rossi; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario; Sabatino, Maione
Sugar-modified nucleosides: synthesis, conformational analysis and biological evaluation
2009-01-01 Vita, Patrizia
New N6-substituted adenosine and 3’-C-methyl-adenosine derivatives as antitumor agents
2009-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Kusumanchi, P; Kumar, M; Jayaram, Hn; Grifantini, Mario
Selective inhibition of nicotinamide adenine kinases (NADKs) by compact NAD mimics
2009-01-01 Petrelli, Riccardo; Felczak, K; Chen, L; Vita, Patrizia; Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Di Stefano, M; Magni, G; Pankiewicz, K.
EFFECTS OF METAL(III) COORDINATION ON BIOLOGICAL ACTIVITY OF 2,2'-BIPYRIDYL-6-CARBOTHIOAMIDE (BPYTA), A POTENT R2 RIBONUCLEOTIDE REDUCTASE INHIBITOR
2010-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Heffeter P., Kowol CR; Franchetti, Palmarisa
Dual-target dimeric molecules with antitumor properties. Synthesis and biological activity of 3’-C-methyladenosine-valproates
2010-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Jayaram, Hn; Grifantini, Mario
5'-CHLORO-5'-DEOXY-N6-(±)-endo-NORBORNYLADENOSINE, A POTENT AND HIGHLY SELECTIVE HUMAN A1 ADENOSINE RECEPTOR AGONIST, PREVENTS HYPERALGESIA/ALLODYNIA AND EARLY OVER-EXPRESSION OF PRO-APOPTOTIC AND PRO-INFLAMMATORY GENES IN A MICE MODEL OF NEUROPATHIC PAIN
2010-01-01 V., De Novellis; Cappellacci, Loredana; L., Luongo; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario; S., Maione
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
First TiCl4-Mediated Diastereoslective Reduction of alpha-Nitro Ketones to beta-Nitro Alcohols by BH3.SMe2 | 1-gen-2000 | Ballini, Roberto; Bosica, Giovanna; Marcantoni, Enrico; Vita, Patrizia; Bartoli, G. | Articolo | |
Stereoselective synthesis of nicotinamide β-riboside and nucleoside analogs | 1-gen-2004 | Franchetti, Palmarisa; Pasqualini, M.; Petrelli, Riccardo; Ricciutelli, Massimo; Vita, Patrizia; Cappellacci, Loredana | Articolo | |
3’-C-Methyl-ribosyl nucleosides as cytotoxic compounds | 1-gen-2005 | Cappellacci, L.; Franchetti, P.; Grifantini, M.; Pasqualini, M.; Petrelli, R.; Vita, P.; Jayaram, H.; Horvath, Z.; Szekeres, T. | Contributo in atto di convegno su volume | |
Affinity and selectivity of tecadenoson, 2-chloro-tecadenoson and 2’-C-methyl analogues at bovine and pig A1 adenosine receptor | 1-gen-2005 | Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M.; Costa, B.; Spinetti, F.; Martini, C.; Klotz, K.; Lavecchia, A. | Poster atto convegno su volume | |
Synthesis and Biological Evaluation of NAD Analogs as Human Pyridine Nucleotide Adenylyltransferase Inhibitors | 1-gen-2005 | Franchetti, Palmarisa; Petrelli, Riccardo; Cappellacci, Loredana; Pasqualini, M.; Vita, Patrizia; Sorci, L.; Mazzola, F.; Raffaelli, N.; Magni, G. | Articolo | |
Ribose-modified mizoribine analogues: synthesis and biological evaluation | 1-gen-2005 | Franchetti, Palmarisa; Pasqualini, M.; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Jayaram, H. N. | Articolo | |
Structure-affinity relathionships of 5'-carbamoyl- and 5'-thionocarbamoyl derivatives of the A1 selective adenosine receptor agonist 2'-MeCCPA as partial A1 agonists | 1-gen-2005 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; B., Costa; C., Martini; A., Lavecchia; Kn, Klotz; Grifantini, Mario | Poster atto convegno su rivista | |
2’-C-Methyl derivatives of tecadenoson and 2-chloro-tecadenoson with increased selectivity for human A1 adenosine receptor | 1-gen-2006 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M; Costa, B; Spinetti, F; Martini, C; Klotz, K. N.; Lavecchia, A; Grifantini, Mario | Poster atto convegno su rivista | |
Purine and pyrimidine nucleoside analogs of 3'-C-methyladenosine as antitumor agents | 1-gen-2006 | Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Riccioni, S.; Vita, Patrizia; Jayaram, H. N.; Grifantini, Mario | Articolo | |
Inhibition of HIV-1 replication in macrophages by red blood cell-mediated delivery of a heterodinucleotide of lamivudine and tenofovir | 1-gen-2007 | Franchetti, Palmarisa; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Rossi, L.; Pierige', F.; Serafini, S.; Magnani, M.; Balestra, E.; Perno, C. F. | Articolo | |
ATP-mimetics derived from 2 '(3 ')-C-methyladenosine as human P2Y2 agonists | 1-gen-2008 | Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Vita, Patrizia; Jacobson, K. A.; Maddileti, S.; Harden, T. K.; Grifantini, Mario | Poster atto convegno su rivista | |
Synthesis and antitumor activity of a heterodinucleotide of BVDU and Gemcitabine | 1-gen-2008 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario | Articolo | |
5'-Chloro-5'-deoxy-N6-(±)-endo-norbornyladenosine, a potent and highly selective human A1 adenosine receptor agonist modulates neuropathic pain in mice. | 1-gen-2009 | Livio, Luongo; Cappellacci, Loredana; Enza, Palazzo; Claudia, Rossi; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario; Sabatino, Maione | Poster atto convegno su volume | |
Sugar-modified nucleosides: synthesis, conformational analysis and biological evaluation | 1-gen-2009 | Vita, Patrizia | Doctoral Thesis | |
New N6-substituted adenosine and 3’-C-methyl-adenosine derivatives as antitumor agents | 1-gen-2009 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Kusumanchi, P; Kumar, M; Jayaram, Hn; Grifantini, Mario | Contributo in atto di convegno su volume | |
Selective inhibition of nicotinamide adenine kinases (NADKs) by compact NAD mimics | 1-gen-2009 | Petrelli, Riccardo; Felczak, K; Chen, L; Vita, Patrizia; Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Di Stefano, M; Magni, G; Pankiewicz, K. | Contributo in atto di convegno su volume | |
EFFECTS OF METAL(III) COORDINATION ON BIOLOGICAL ACTIVITY OF 2,2'-BIPYRIDYL-6-CARBOTHIOAMIDE (BPYTA), A POTENT R2 RIBONUCLEOTIDE REDUCTASE INHIBITOR | 1-gen-2010 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Heffeter P., Kowol CR; Franchetti, Palmarisa | Poster atto convegno su volume | |
Dual-target dimeric molecules with antitumor properties. Synthesis and biological activity of 3’-C-methyladenosine-valproates | 1-gen-2010 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Jayaram, Hn; Grifantini, Mario | Poster atto convegno su volume | |
5'-CHLORO-5'-DEOXY-N6-(±)-endo-NORBORNYLADENOSINE, A POTENT AND HIGHLY SELECTIVE HUMAN A1 ADENOSINE RECEPTOR AGONIST, PREVENTS HYPERALGESIA/ALLODYNIA AND EARLY OVER-EXPRESSION OF PRO-APOPTOTIC AND PRO-INFLAMMATORY GENES IN A MICE MODEL OF NEUROPATHIC PAIN | 1-gen-2010 | V., De Novellis; Cappellacci, Loredana; L., Luongo; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario; S., Maione | Contributo in atto di convegno su rivista | |
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario | Poster atto convegno su volume |
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