Sfoglia per Autore
Stereoselective synthesis of nicotinamide β-riboside and nucleoside analogs
2004-01-01 Franchetti, Palmarisa; Pasqualini, M.; Petrelli, Riccardo; Ricciutelli, Massimo; Vita, Patrizia; Cappellacci, Loredana
3’-C-Methyl-ribosyl nucleosides as cytotoxic compounds
2005-01-01 Cappellacci, L.; Franchetti, P.; Grifantini, M.; Pasqualini, M.; Petrelli, R.; Vita, P.; Jayaram, H.; Horvath, Z.; Szekeres, T.
Affinity and selectivity of tecadenoson, 2-chloro-tecadenoson and 2’-C-methyl analogues at bovine and pig A1 adenosine receptor
2005-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M.; Costa, B.; Spinetti, F.; Martini, C.; Klotz, K.; Lavecchia, A.
Antitumor Activity of C-Methyl-beta-D-ribofuranosyladenine Nucleosides Ribonucleotide Reductase Inhibitors
2005-01-01 Franchetti, P.; Cappellacci, Loredana; Pasqualini, M.; Petrelli, Riccardo; Vita, P.; Jayaram, H. N.; Horvath, Z.; Szekeres, T.; Grifantini, M.
The antitumor effects of 3’-methyl-adenosine mediated by inhibition of ribonucleotide reductase.
2005-01-01 Franchetti, P; Cappellacci, Loredana; Pasqualini, M; Petrelli, Riccardo; Vita, P; Jayaram, H. N.; Horvath, Z; Szekeres, T; Grifantini, M.
Synthesis, conformational analysis, and biological activity of new analogues of thiazole-4-carboxamide adenine dinucleotide (TAD) as IMP dehydrogenase inhibitors
2005-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Pasqualini, M.; Petrelli, Riccardo; Jayaprakasan, V.; Jayaram, H. N.; Boyd, D. B.; Jain, M. D.; Grifantini, Mario
Synthesis, Biological Evaluation and Molecular Modeling of Ribose-modified Adenosine Analogues as Adenosine Receptor Agonists
2005-01-01 Cappellacci, Loredana; Franchetti, P.; Pasqualini, M.; Petrelli, Riccardo; Vita, P.; Lavecchia, A.; Novellino, E.; Costa, B.; Martini, C.; Klotz, K. N.; Grifantini, M.
Structure-affinity relathionships of 5'-carbamoyl- and 5'-thionocarbamoyl derivatives of the A1 selective adenosine receptor agonist 2'-MeCCPA as partial A1 agonists
2005-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; B., Costa; C., Martini; A., Lavecchia; Kn, Klotz; Grifantini, Mario
Synthesis and Biological Evaluation of NAD Analogs as Human Pyridine Nucleotide Adenylyltransferase Inhibitors
2005-01-01 Franchetti, Palmarisa; Petrelli, Riccardo; Cappellacci, Loredana; Pasqualini, M.; Vita, Patrizia; Sorci, L.; Mazzola, F.; Raffaelli, N.; Magni, G.
Ribose-modified mizoribine analogues: synthesis and biological evaluation
2005-01-01 Franchetti, Palmarisa; Pasqualini, M.; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Jayaram, H. N.
2’-C-Methyl derivatives of tecadenoson and 2-chloro-tecadenoson with increased selectivity for human A1 adenosine receptor
2006-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M; Costa, B; Spinetti, F; Martini, C; Klotz, K. N.; Lavecchia, A; Grifantini, Mario
Purine and pyrimidine nucleoside analogs of 3'-C-methyladenosine as antitumor agents
2006-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Riccioni, S.; Vita, Patrizia; Jayaram, H. N.; Grifantini, Mario
Inhibition of HIV-1 replication in macrophages by red blood cell-mediated delivery of a heterodinucleotide of lamivudine and tenofovir
2007-01-01 Franchetti, Palmarisa; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Rossi, L.; Pierige', F.; Serafini, S.; Magnani, M.; Balestra, E.; Perno, C. F.
Initial-rate kinetics of human NMN-adenylyltransferases: substrate and metal ion specificity, inhibition by products and multisubstrate analogues, and isozyme contributions to NAD+ biosynthesis
2007-01-01 Sorci, L.; Cimadamore, F.; Scotti, S.; Petrelli, Riccardo; Cappellacci, Loredana; Franchetti, P.; Orsomando, G.; Magni, G.
SYNTHESIS OF NAD ANALOGS AS SELECTIVE INHIBITORS OF INOSINE MONOPHOSPHATE DEHYDROGENASE
2007-01-01 Bonnac, L; Chen, L; Gao, G. Y.; Petrelli, Riccardo; Bennett, E. M.; Pankiewicz, K. W.
DESIGN AND SYNTHESIS OF NOVEL INHIBITORS OF INOSINE MONOPHOSPHATE DEHYDROGENASE
2007-01-01 Gao, G. Y.; Bonnac, L.; Chen, L; Felczak, K.; Kullberg, M.; Petrelli, Riccardo; Bennett, E. M.; Pankiewicz, K. W.
ATP-mimetics derived from 2 '(3 ')-C-methyladenosine as human P2Y2 agonists
2008-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Vita, Patrizia; Jacobson, K. A.; Maddileti, S.; Harden, T. K.; Grifantini, Mario
Synthesis and antitumor activity of a heterodinucleotide of BVDU and Gemcitabine
2008-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario
Synthesis and potency of novel uracil nucleotides and derivatives as P2Y(2) and P2Y(6) receptor agonists
2008-01-01 Ko, H.; Carter, R. L.; Cosyn, L.; Petrelli, Riccardo; DE CASTRO, S.; Besada, P.; Zhou, Y.; Cappellacci, Loredana; Franchetti, P.; Grifantini, M.; VAN CALENBERGH, S.; Harden, T. K.; Jacobson, K. A.
Bis(sulfonamide) isosters of mycophenolic adenine dinucleotide analogues. inhibition of inosine monophosphate dehydrogenase.
2008-01-01 Chen, L; Petrelli, Riccardo; Olesiak, M; Wilson, Dj; Labello, Np; Pankiewicz, Kw
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Stereoselective synthesis of nicotinamide β-riboside and nucleoside analogs | 1-gen-2004 | Franchetti, Palmarisa; Pasqualini, M.; Petrelli, Riccardo; Ricciutelli, Massimo; Vita, Patrizia; Cappellacci, Loredana | Articolo | |
3’-C-Methyl-ribosyl nucleosides as cytotoxic compounds | 1-gen-2005 | Cappellacci, L.; Franchetti, P.; Grifantini, M.; Pasqualini, M.; Petrelli, R.; Vita, P.; Jayaram, H.; Horvath, Z.; Szekeres, T. | Contributo in atto di convegno su volume | |
Affinity and selectivity of tecadenoson, 2-chloro-tecadenoson and 2’-C-methyl analogues at bovine and pig A1 adenosine receptor | 1-gen-2005 | Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M.; Costa, B.; Spinetti, F.; Martini, C.; Klotz, K.; Lavecchia, A. | Poster atto convegno su volume | |
Antitumor Activity of C-Methyl-beta-D-ribofuranosyladenine Nucleosides Ribonucleotide Reductase Inhibitors | 1-gen-2005 | Franchetti, P.; Cappellacci, Loredana; Pasqualini, M.; Petrelli, Riccardo; Vita, P.; Jayaram, H. N.; Horvath, Z.; Szekeres, T.; Grifantini, M. | Articolo | |
The antitumor effects of 3’-methyl-adenosine mediated by inhibition of ribonucleotide reductase. | 1-gen-2005 | Franchetti, P; Cappellacci, Loredana; Pasqualini, M; Petrelli, Riccardo; Vita, P; Jayaram, H. N.; Horvath, Z; Szekeres, T; Grifantini, M. | Contributo in atto di convegno su volume | |
Synthesis, conformational analysis, and biological activity of new analogues of thiazole-4-carboxamide adenine dinucleotide (TAD) as IMP dehydrogenase inhibitors | 1-gen-2005 | Franchetti, Palmarisa; Cappellacci, Loredana; Pasqualini, M.; Petrelli, Riccardo; Jayaprakasan, V.; Jayaram, H. N.; Boyd, D. B.; Jain, M. D.; Grifantini, Mario | Articolo | |
Synthesis, Biological Evaluation and Molecular Modeling of Ribose-modified Adenosine Analogues as Adenosine Receptor Agonists | 1-gen-2005 | Cappellacci, Loredana; Franchetti, P.; Pasqualini, M.; Petrelli, Riccardo; Vita, P.; Lavecchia, A.; Novellino, E.; Costa, B.; Martini, C.; Klotz, K. N.; Grifantini, M. | Articolo | |
Structure-affinity relathionships of 5'-carbamoyl- and 5'-thionocarbamoyl derivatives of the A1 selective adenosine receptor agonist 2'-MeCCPA as partial A1 agonists | 1-gen-2005 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; B., Costa; C., Martini; A., Lavecchia; Kn, Klotz; Grifantini, Mario | Poster atto convegno su rivista | |
Synthesis and Biological Evaluation of NAD Analogs as Human Pyridine Nucleotide Adenylyltransferase Inhibitors | 1-gen-2005 | Franchetti, Palmarisa; Petrelli, Riccardo; Cappellacci, Loredana; Pasqualini, M.; Vita, Patrizia; Sorci, L.; Mazzola, F.; Raffaelli, N.; Magni, G. | Articolo | |
Ribose-modified mizoribine analogues: synthesis and biological evaluation | 1-gen-2005 | Franchetti, Palmarisa; Pasqualini, M.; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Jayaram, H. N. | Articolo | |
2’-C-Methyl derivatives of tecadenoson and 2-chloro-tecadenoson with increased selectivity for human A1 adenosine receptor | 1-gen-2006 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Pasqualini, M; Costa, B; Spinetti, F; Martini, C; Klotz, K. N.; Lavecchia, A; Grifantini, Mario | Poster atto convegno su rivista | |
Purine and pyrimidine nucleoside analogs of 3'-C-methyladenosine as antitumor agents | 1-gen-2006 | Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Riccioni, S.; Vita, Patrizia; Jayaram, H. N.; Grifantini, Mario | Articolo | |
Inhibition of HIV-1 replication in macrophages by red blood cell-mediated delivery of a heterodinucleotide of lamivudine and tenofovir | 1-gen-2007 | Franchetti, Palmarisa; Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Rossi, L.; Pierige', F.; Serafini, S.; Magnani, M.; Balestra, E.; Perno, C. F. | Articolo | |
Initial-rate kinetics of human NMN-adenylyltransferases: substrate and metal ion specificity, inhibition by products and multisubstrate analogues, and isozyme contributions to NAD+ biosynthesis | 1-gen-2007 | Sorci, L.; Cimadamore, F.; Scotti, S.; Petrelli, Riccardo; Cappellacci, Loredana; Franchetti, P.; Orsomando, G.; Magni, G. | Articolo | |
SYNTHESIS OF NAD ANALOGS AS SELECTIVE INHIBITORS OF INOSINE MONOPHOSPHATE DEHYDROGENASE | 1-gen-2007 | Bonnac, L; Chen, L; Gao, G. Y.; Petrelli, Riccardo; Bennett, E. M.; Pankiewicz, K. W. | Contributo in atto di convegno su volume | |
DESIGN AND SYNTHESIS OF NOVEL INHIBITORS OF INOSINE MONOPHOSPHATE DEHYDROGENASE | 1-gen-2007 | Gao, G. Y.; Bonnac, L.; Chen, L; Felczak, K.; Kullberg, M.; Petrelli, Riccardo; Bennett, E. M.; Pankiewicz, K. W. | Contributo in atto di convegno su volume | |
ATP-mimetics derived from 2 '(3 ')-C-methyladenosine as human P2Y2 agonists | 1-gen-2008 | Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Vita, Patrizia; Jacobson, K. A.; Maddileti, S.; Harden, T. K.; Grifantini, Mario | Poster atto convegno su rivista | |
Synthesis and antitumor activity of a heterodinucleotide of BVDU and Gemcitabine | 1-gen-2008 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, Patrizia; Petrelli, Riccardo; Grifantini, Mario | Articolo | |
Synthesis and potency of novel uracil nucleotides and derivatives as P2Y(2) and P2Y(6) receptor agonists | 1-gen-2008 | Ko, H.; Carter, R. L.; Cosyn, L.; Petrelli, Riccardo; DE CASTRO, S.; Besada, P.; Zhou, Y.; Cappellacci, Loredana; Franchetti, P.; Grifantini, M.; VAN CALENBERGH, S.; Harden, T. K.; Jacobson, K. A. | Articolo | |
Bis(sulfonamide) isosters of mycophenolic adenine dinucleotide analogues. inhibition of inosine monophosphate dehydrogenase. | 1-gen-2008 | Chen, L; Petrelli, Riccardo; Olesiak, M; Wilson, Dj; Labello, Np; Pankiewicz, Kw | Articolo |
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