Sfoglia per Autore
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario
Synthesis and Enzymatic Evaluation of NAD Mimics as Nicotinamide Adenine Dinucleotide Kinase (NADK) Inhibitors
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Krzysztof, Felczak; Vita, Patrizia; Torquati, Ilaria; Palmarisa, Franchetti; Michele Di, Stefano; Giulio, Magni; Mario, Grifantini; Krzysztof W., Pankiewicz
Bisphosphonate Derivatives of 2’-C-Methyl-, and 3’-C-Methyl-Adenosine as Ligands at P2Y1 and P2Y2 Receptors
2012-01-01 Petrelli, Riccardo; Vita, Patrizia; Franchetti, P; Torquati, Ilaria; Barrett, O. M.; Harden, Kt; Grifantini, M; Cappellacci, Loredana
Design, synthesis and biological evaluation of novel inhibitors of NAD kinase
2012-01-01 Torquati, Ilaria; Vita, Patrizia; Petrelli, Riccardo; Di Stefano, M; Cappellacci, Loredana
PROBING BINDING REQUIREMENTS OF NAD KINASE WITH MODIFIED NAD ANALOGUES
2012-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krzysztof, Felczak; Palmarisa, Franchetti; Mario, Grifantini; Michele Di, Stefano; Giulio, Magni; Krzysztof W., Pankiewicz; Cappellacci, Loredana
Synthesis and biological evaluation of (methylene)bisphosphonate derivatives of 2’-C-methyl-, and 3’-C-methyl-adenosine
2012-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Palmarisa, Franchetti; Torquati, Ilaria; Matthew O., Barrett; Kendal T., Harden; Mario, Grifantini
ADP- and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 receptor ligands
2012-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Jacobson, Ka; Barrett, Mo; Franklin, D; Harden, Kt; Franchetti, Palmarisa; Grifantini, Mario
NOVEL 2-SUBSTITUTED 2’/3’-C-METHYL-ADENOSINE DERIVATIVES: SYNTHESIS AND BIOLOGICAL EVALUATION AGAINST TRYPANOSOMA BRUCEI
2013-01-01 Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Boccoli; A., Hofer; M., Vodnala; P., Franchetti; M., Grifantini; Cappellacci, Loredana
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE
2013-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; L., Luongo; F., Guida; M., De Chiaro; K. N., Klotz; S., Kachler; P., Franchetti; S., Maione; M., Grifantini; Cappellacci, Loredana
SINTESI E VALUTAZIONE BIOLOGICA DI INIBITORI DI ENZIMI CHIAVE NEL METABOLISMO DI BIOFILM BATTERICI
2013-01-01 Torquati, Ilaria; Petrelli, Riccardo; Moretti, M; Pierella, S; Fernicola, S; Stelitano, V; Rinaldo, S; Cutruzzolà, F; Cappellacci, Loredana
SYNTHESIS AND BIOLOGICAL EVALUATION OF NEW INHIBITORS OF ENZYMES INVOLVED IN c-di-GMP METABOLISM
2013-01-01 Petrelli, Riccardo; Torquati, Ilaria; S., Fernicola; V. Stelitano S., Rinaldo; G., Rampioni; M., Messina; L., Leoni; F., Cutruzzolà; Cappellacci, Loredana
5’-CHLORO-5’-DEOXY-N6-SUBSTITUTED ADENOSINE DERIVATIVES: SYNTHESIS, ADENOSINE RECEPTOR AFFINITY AND ANTINOCICEPTIVE ACTIVITY
2013-01-01 Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Luongo; K. N., Klotz; S., Kachler; F., Guida; M., De Chiaro; S., Maione; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana
Targeting biofilm formation by human pathogenic bacteria: functional and inhibition studies of diguanylate cyclases
2013-01-01 Fernicola, S; Rinaldo, S; Giardina, G; Torquati, Ilaria; Petrelli, Riccardo; Cappellacci, Loredana; Cutruzzolà, Francesca
Novel Inhibitors of Inosine Monophosphate Dehydrogenase in Patent Literature of the Last Decade
2013-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krysztof, Felczak; Daniel J., Wilson; Franchetti, Palmarisa; Cappellacci, Loredana
SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF NOVEL HYDRAZONE DERIVATIVES
2014-01-01 Petrelli, Riccardo; Torquati, Ilaria; Anders, Hofer; Olivia, Grubbström; Venkateswara Rao, Jonn; Praveen, Kusumanchi; Hiremagalur N., Jayaram; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana
IDENTIFICATION OF MOLECULES THAT INHIBITS c-di-GMP SYNTHESIS TO TARGET BIOFILM FORMATION
2014-01-01 Fernicola, S; Paiardini, A; Rinaldo, S; Torquati, Ilaria; Petrelli, Riccardo; Cappellacci, Loredana; Cutruzzolà, F.
STEREOSELECTIVE SYNTHESIS OF ISO-CARBOCYCLIC NUCLEOSIDE ANALOGUES AS POTENTIAL ANTIVIRAL DRUGS
2014-01-01 Torquati, Ilaria; Simon, Weising; Chris, Meier
4’-TETRAZOLYL-ALKYL-N6-SUBSTITUTED ADENOSINE DERIVATIVES AS HIGHLY POTENT DUAL ACTING A1 ADENOSINE RECEPTOR AGONISTS AND A3 ADENOSINE RECEPTOR ANTAGONISTS
2014-01-01 Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Francesca, Guida; Serena, Boccella; Antonio, Lavecchia; Karl Norbert, Klotz; Sonja, Kachler; Palmarisa, Franchetti; Mario, Grifantini; Sabatino, Maione; Cappellacci, Loredana
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE
2014-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Livio, Luongo; Francesca, Guida; Maria De, Chiaro; Karl Norbert, Klotz; Sonja, Kachler; Palmarisa, Franchetti; Sabatino, Maione; Mario, Grifantini; Cappellacci, Loredana
Novel Inhibitors of Inosine Monophosphate Dehydrogenase as Potential Anti-Cancer Drugs: A Patent Review (2002-2014)
2014-01-01 Petrelli, Riccardo; Torquati, Ilaria; Krzysztof, Felczak; Daniel J., Wilson; Cappellacci, Loredana
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario | Poster atto convegno su volume | |
Synthesis and Enzymatic Evaluation of NAD Mimics as Nicotinamide Adenine Dinucleotide Kinase (NADK) Inhibitors | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Krzysztof, Felczak; Vita, Patrizia; Torquati, Ilaria; Palmarisa, Franchetti; Michele Di, Stefano; Giulio, Magni; Mario, Grifantini; Krzysztof W., Pankiewicz | Poster atto convegno su volume | |
Bisphosphonate Derivatives of 2’-C-Methyl-, and 3’-C-Methyl-Adenosine as Ligands at P2Y1 and P2Y2 Receptors | 1-gen-2012 | Petrelli, Riccardo; Vita, Patrizia; Franchetti, P; Torquati, Ilaria; Barrett, O. M.; Harden, Kt; Grifantini, M; Cappellacci, Loredana | Poster atto convegno su volume | |
Design, synthesis and biological evaluation of novel inhibitors of NAD kinase | 1-gen-2012 | Torquati, Ilaria; Vita, Patrizia; Petrelli, Riccardo; Di Stefano, M; Cappellacci, Loredana | Contributo in atto di convegno su volume | |
PROBING BINDING REQUIREMENTS OF NAD KINASE WITH MODIFIED NAD ANALOGUES | 1-gen-2012 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krzysztof, Felczak; Palmarisa, Franchetti; Mario, Grifantini; Michele Di, Stefano; Giulio, Magni; Krzysztof W., Pankiewicz; Cappellacci, Loredana | Poster atto convegno su volume | |
Synthesis and biological evaluation of (methylene)bisphosphonate derivatives of 2’-C-methyl-, and 3’-C-methyl-adenosine | 1-gen-2012 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Palmarisa, Franchetti; Torquati, Ilaria; Matthew O., Barrett; Kendal T., Harden; Mario, Grifantini | Poster atto convegno su volume | |
ADP- and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 receptor ligands | 1-gen-2012 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Jacobson, Ka; Barrett, Mo; Franklin, D; Harden, Kt; Franchetti, Palmarisa; Grifantini, Mario | Contributo in atto di convegno su rivista | |
NOVEL 2-SUBSTITUTED 2’/3’-C-METHYL-ADENOSINE DERIVATIVES: SYNTHESIS AND BIOLOGICAL EVALUATION AGAINST TRYPANOSOMA BRUCEI | 1-gen-2013 | Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Boccoli; A., Hofer; M., Vodnala; P., Franchetti; M., Grifantini; Cappellacci, Loredana | Poster atto convegno su volume | |
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE | 1-gen-2013 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; L., Luongo; F., Guida; M., De Chiaro; K. N., Klotz; S., Kachler; P., Franchetti; S., Maione; M., Grifantini; Cappellacci, Loredana | Poster atto convegno su volume | |
SINTESI E VALUTAZIONE BIOLOGICA DI INIBITORI DI ENZIMI CHIAVE NEL METABOLISMO DI BIOFILM BATTERICI | 1-gen-2013 | Torquati, Ilaria; Petrelli, Riccardo; Moretti, M; Pierella, S; Fernicola, S; Stelitano, V; Rinaldo, S; Cutruzzolà, F; Cappellacci, Loredana | Contributo in atto di convegno su volume | |
SYNTHESIS AND BIOLOGICAL EVALUATION OF NEW INHIBITORS OF ENZYMES INVOLVED IN c-di-GMP METABOLISM | 1-gen-2013 | Petrelli, Riccardo; Torquati, Ilaria; S., Fernicola; V. Stelitano S., Rinaldo; G., Rampioni; M., Messina; L., Leoni; F., Cutruzzolà; Cappellacci, Loredana | Poster atto convegno su volume | |
5’-CHLORO-5’-DEOXY-N6-SUBSTITUTED ADENOSINE DERIVATIVES: SYNTHESIS, ADENOSINE RECEPTOR AFFINITY AND ANTINOCICEPTIVE ACTIVITY | 1-gen-2013 | Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Luongo; K. N., Klotz; S., Kachler; F., Guida; M., De Chiaro; S., Maione; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana | Poster atto convegno su volume | |
Targeting biofilm formation by human pathogenic bacteria: functional and inhibition studies of diguanylate cyclases | 1-gen-2013 | Fernicola, S; Rinaldo, S; Giardina, G; Torquati, Ilaria; Petrelli, Riccardo; Cappellacci, Loredana; Cutruzzolà, Francesca | Poster atto convegno su volume | |
Novel Inhibitors of Inosine Monophosphate Dehydrogenase in Patent Literature of the Last Decade | 1-gen-2013 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krysztof, Felczak; Daniel J., Wilson; Franchetti, Palmarisa; Cappellacci, Loredana | Articolo | |
SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF NOVEL HYDRAZONE DERIVATIVES | 1-gen-2014 | Petrelli, Riccardo; Torquati, Ilaria; Anders, Hofer; Olivia, Grubbström; Venkateswara Rao, Jonn; Praveen, Kusumanchi; Hiremagalur N., Jayaram; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana | Poster atto convegno su volume | |
IDENTIFICATION OF MOLECULES THAT INHIBITS c-di-GMP SYNTHESIS TO TARGET BIOFILM FORMATION | 1-gen-2014 | Fernicola, S; Paiardini, A; Rinaldo, S; Torquati, Ilaria; Petrelli, Riccardo; Cappellacci, Loredana; Cutruzzolà, F. | Poster atto convegno su volume | |
STEREOSELECTIVE SYNTHESIS OF ISO-CARBOCYCLIC NUCLEOSIDE ANALOGUES AS POTENTIAL ANTIVIRAL DRUGS | 1-gen-2014 | Torquati, Ilaria; Simon, Weising; Chris, Meier | Poster atto convegno su volume | |
4’-TETRAZOLYL-ALKYL-N6-SUBSTITUTED ADENOSINE DERIVATIVES AS HIGHLY POTENT DUAL ACTING A1 ADENOSINE RECEPTOR AGONISTS AND A3 ADENOSINE RECEPTOR ANTAGONISTS | 1-gen-2014 | Petrelli, Riccardo; Torquati, Ilaria; Livio, Luongo; Francesca, Guida; Serena, Boccella; Antonio, Lavecchia; Karl Norbert, Klotz; Sonja, Kachler; Palmarisa, Franchetti; Mario, Grifantini; Sabatino, Maione; Cappellacci, Loredana | Contributo in atto di convegno su rivista | |
N6/5’-DISUBSTITUTED ADENOSINE AND 2-CHLORO-ADENOSINE DERIVATIVES AS POTENT AND SELECTIVE A1 ADENOSINE RECEPTOR AGONISTS: SYNTHESIS, BINDING ASSAYS AND ANTINOCICEPTIVE ACTIVITY IN MICE | 1-gen-2014 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Livio, Luongo; Francesca, Guida; Maria De, Chiaro; Karl Norbert, Klotz; Sonja, Kachler; Palmarisa, Franchetti; Sabatino, Maione; Mario, Grifantini; Cappellacci, Loredana | Poster atto convegno su rivista | |
Novel Inhibitors of Inosine Monophosphate Dehydrogenase as Potential Anti-Cancer Drugs: A Patent Review (2002-2014) | 1-gen-2014 | Petrelli, Riccardo; Torquati, Ilaria; Krzysztof, Felczak; Daniel J., Wilson; Cappellacci, Loredana | Capitolo di libro o voce di enciclopedia |
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