Sfoglia per Autore
Effect of Deoxamuscarine Etherification on M2 and M3 Muscarinic Affinity and Efficacy
1992-01-01 Livio, Brasili; Mario, Giannella; Alessandro, Piergentili; Tayebati, Seyed Khosrow
Resolution and muscarinic activity of (+)- and ( – )-4a-methyl-3b- hydroxy-1a -(N,N-dimethylaminomethyl) cyclopentane methiodide [(+)-deoxamuscarine]
1992-01-01 Alessandro, Piergentili; Tayebati, Seyed Khosrow; Mario, Giannella
Hypotensive effect of intravenous injection of tachykinins in conscious, freely moving spontaneously hypertensive and Wistar Kyoto rats.
1993-01-01 Pompei, Pierluigi; Tayebati, Seyed Khosrow; Polidori, Carlo; Perfumi, Marina Cecilia; De Caro, G; Massi, Maurizio
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 4. Effect of aryl and alkyl Substituents at Position 3 on α-adrenoreceptor blocking activity
1993-01-01 Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Melchiorre, C.
Synthesis and Muscarinic Receptors Affinity of a series of Antagonist Bivalent Ligands
1994-01-01 Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow; F., Paparelli; L., Malmusi; L., Brasili
Synthesis and muscarinic properties of (1S*,3R*,5R*)-trimethyl(1-methyl-6-oxabicyclo[3.1.0]hex-3-yl)methyl ammonium iodide
1994-01-01 Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Rafaiani, Giovanni; Tayebati, Seyed Khosrow
Age-related Changes in the Density of Muscarinic Cholinergic M1 and M2 Receptor Subtypes in Pyramidal Neurons or the rat Hippocampus
1995-01-01 Amenta, Francesco; A., Liu; Giannella, Mario; Pigini, Maria; Tayebati, Seyed Khosrow; AND D., Zaccheo
Muscarinic Thioligands with Cyclopentane Nucleus
1996-01-01 Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow; Amenta, Francesco; Sabbatini, M.; Giannella, Mario
Discovery of Highly Selective Imidazoline Receptor Ligands
1996-01-01 L., Brasili; Pigini, Maria; R., Moriconi; A., Carotti; P., Bousquet; M., Dontenwill; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 5. Effects of Modification of the side chain on alpha-adrenoreceptor blocking Activity
1996-01-01 Quaglia, Wilma; Giannella, Mario; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Tayebati, Seyed Khosrow; Melchiorre, C.
Synthesis, Absolute Configuration, and Biological Profile of the Enantiomers of trans-[2-(2,6-Dimethoxypheoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (Mephendioxan), a Potent Competitive alpha 1A-Adrenoreceptor Antagonist
1996-01-01 Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; A., Leonardi; C., Taddei; C., Melchiorre
Byciclic dioxolanes as potential antimuscarinic agents
1996-01-01 Piergentili, Alessandro; Angeli, Piero; Giannella, Mario; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow
Postnatal development of dopamine D1-like and D2-like receptors in the rat kidney: a radioligand binding study
1997-01-01 G., Tenore; P., Barili; M., Sabbatini; Tayebati, Seyed Khosrow; Amenta, Francesco
Imidazoline receptors: Qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity
1997-01-01 Pigini, Maria; Bousquet, P; Carotti, A; Dontenwill, M; Giannella, Mario; Moriconi, R; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow; Brasili, L.
Use of frozen sections for the pharmacological characterization of compounds active on neurotransmitter receptors
1997-01-01 Tayebati, Seyed Khosrow; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Sabbatini, M.; Amenta, Francesco
Dopamine D4 receptor in human peripheral blood lymphocytes: a radioligand binding assay study
1997-01-01 A., Ricci; E., Bronzetti; L., Felici; Tayebati, Seyed Khosrow; Amenta, Francesco
MUSCARINIC CHOLINERGIC RECEPTORS SUBTYPES EXPRESSION BY HUMAN PLACENTA
1997-01-01 Tayebati, Seyed Khosrow; M., Sabbatini; D., Zaccheo; Amenta, Francesco
Autoradiographic localization of muscarinic cholinergic receptor subtypes in human placenta.
1998-01-01 Tayebati, Seyed Khosrow; Vitaioli, L; Zaccheo, D; Amenta, Francesco
Dopamine D2-like receptors on human peripheral blood lymphocytes: a radioligand binding assay and immunocytochemical study
1999-01-01 Amenta, Francesco; E., Bronzetti; L., Felici; A., Ricci; Tayebati, Seyed Khosrow
Evaluation of an Agonist Index: Affinity Ratio for Compounds Active on Muscarinic Cholinergic M2 Receptors
1999-01-01 Tayebati, Seyed Khosrow; Piergentili, Alessandro; Natale, D.; Amenta, Francesco
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Effect of Deoxamuscarine Etherification on M2 and M3 Muscarinic Affinity and Efficacy | 1-gen-1992 | Livio, Brasili; Mario, Giannella; Alessandro, Piergentili; Tayebati, Seyed Khosrow | Articolo | |
Resolution and muscarinic activity of (+)- and ( – )-4a-methyl-3b- hydroxy-1a -(N,N-dimethylaminomethyl) cyclopentane methiodide [(+)-deoxamuscarine] | 1-gen-1992 | Alessandro, Piergentili; Tayebati, Seyed Khosrow; Mario, Giannella | Articolo | |
Hypotensive effect of intravenous injection of tachykinins in conscious, freely moving spontaneously hypertensive and Wistar Kyoto rats. | 1-gen-1993 | Pompei, Pierluigi; Tayebati, Seyed Khosrow; Polidori, Carlo; Perfumi, Marina Cecilia; De Caro, G; Massi, Maurizio | Articolo | |
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 4. Effect of aryl and alkyl Substituents at Position 3 on α-adrenoreceptor blocking activity | 1-gen-1993 | Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; Marucci, Gabriella; Melchiorre, C. | Articolo | |
Synthesis and Muscarinic Receptors Affinity of a series of Antagonist Bivalent Ligands | 1-gen-1994 | Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow; F., Paparelli; L., Malmusi; L., Brasili | Articolo | |
Synthesis and muscarinic properties of (1S*,3R*,5R*)-trimethyl(1-methyl-6-oxabicyclo[3.1.0]hex-3-yl)methyl ammonium iodide | 1-gen-1994 | Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Rafaiani, Giovanni; Tayebati, Seyed Khosrow | Articolo | |
Age-related Changes in the Density of Muscarinic Cholinergic M1 and M2 Receptor Subtypes in Pyramidal Neurons or the rat Hippocampus | 1-gen-1995 | Amenta, Francesco; A., Liu; Giannella, Mario; Pigini, Maria; Tayebati, Seyed Khosrow; AND D., Zaccheo | Articolo | |
Muscarinic Thioligands with Cyclopentane Nucleus | 1-gen-1996 | Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow; Amenta, Francesco; Sabbatini, M.; Giannella, Mario | Articolo | |
Discovery of Highly Selective Imidazoline Receptor Ligands | 1-gen-1996 | L., Brasili; Pigini, Maria; R., Moriconi; A., Carotti; P., Bousquet; M., Dontenwill; Giannella, Mario; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow | Capitolo di libro o voce di enciclopedia | |
Structure- Activity Relationships in 1,4-Benzodioxan-related Compounds. 5. Effects of Modification of the side chain on alpha-adrenoreceptor blocking Activity | 1-gen-1996 | Quaglia, Wilma; Giannella, Mario; Marucci, Gabriella; Piergentili, Alessandro; Pigini, Maria; Tayebati, Seyed Khosrow; Melchiorre, C. | Articolo | |
Synthesis, Absolute Configuration, and Biological Profile of the Enantiomers of trans-[2-(2,6-Dimethoxypheoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (Mephendioxan), a Potent Competitive alpha 1A-Adrenoreceptor Antagonist | 1-gen-1996 | Quaglia, Wilma; Pigini, Maria; Tayebati, Seyed Khosrow; Piergentili, Alessandro; Giannella, Mario; A., Leonardi; C., Taddei; C., Melchiorre | Articolo | |
Byciclic dioxolanes as potential antimuscarinic agents | 1-gen-1996 | Piergentili, Alessandro; Angeli, Piero; Giannella, Mario; Pigini, Maria; Quaglia, Wilma; Tayebati, Seyed Khosrow | Articolo | |
Postnatal development of dopamine D1-like and D2-like receptors in the rat kidney: a radioligand binding study | 1-gen-1997 | G., Tenore; P., Barili; M., Sabbatini; Tayebati, Seyed Khosrow; Amenta, Francesco | Articolo | |
Imidazoline receptors: Qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity | 1-gen-1997 | Pigini, Maria; Bousquet, P; Carotti, A; Dontenwill, M; Giannella, Mario; Moriconi, R; Piergentili, Alessandro; Quaglia, Wilma; Tayebati, Seyed Khosrow; Brasili, L. | Articolo | |
Use of frozen sections for the pharmacological characterization of compounds active on neurotransmitter receptors | 1-gen-1997 | Tayebati, Seyed Khosrow; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Sabbatini, M.; Amenta, Francesco | Articolo | |
Dopamine D4 receptor in human peripheral blood lymphocytes: a radioligand binding assay study | 1-gen-1997 | A., Ricci; E., Bronzetti; L., Felici; Tayebati, Seyed Khosrow; Amenta, Francesco | Articolo | |
MUSCARINIC CHOLINERGIC RECEPTORS SUBTYPES EXPRESSION BY HUMAN PLACENTA | 1-gen-1997 | Tayebati, Seyed Khosrow; M., Sabbatini; D., Zaccheo; Amenta, Francesco | Articolo | |
Autoradiographic localization of muscarinic cholinergic receptor subtypes in human placenta. | 1-gen-1998 | Tayebati, Seyed Khosrow; Vitaioli, L; Zaccheo, D; Amenta, Francesco | Articolo | |
Dopamine D2-like receptors on human peripheral blood lymphocytes: a radioligand binding assay and immunocytochemical study | 1-gen-1999 | Amenta, Francesco; E., Bronzetti; L., Felici; A., Ricci; Tayebati, Seyed Khosrow | Articolo | |
Evaluation of an Agonist Index: Affinity Ratio for Compounds Active on Muscarinic Cholinergic M2 Receptors | 1-gen-1999 | Tayebati, Seyed Khosrow; Piergentili, Alessandro; Natale, D.; Amenta, Francesco | Articolo |
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