Sfoglia per Titolo
Synthesis and pharmacological characterization of chiral pyrrolidinylfuran derivatives: The discovery of new functionally selective muscarinic agonists
2008-01-01 Scapecchi, S.; Nesi, M.; Matucci, R.; Bellucci, C.; Buccioni, Michela; Dei, S.; Guandalini, L.; Manetti, D.; Martini, E.; Marucci, Gabriella; Romanelli, M. N.; Teodori, E.; Cirilli, R.
Synthesis and pharmacological characterization of enantiomerically pure muscarinic agonists: difluoromuscarines
1997-01-01 Angeli, Piero; Cantalamessa, Franco; Cavagna, Roberto; Conti, Paola; De Amici, Marco; De Micheli, Marco; Gamba, Anna; Marucci, Gabriella
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine
2000-01-01 DE AMICI, M.; Dallanoce, C.; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; DE MICHELIS, C.
SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF RIBOSE-MODIFIED ADENOSINE DERIVATIVES AS P1 RECEPTOR LIGANDS
2016-01-01 Scortichini, Mirko; Petrelli, Riccardo; Kachler, S.; Luongo, L.; Maione, S.; NGAHANG KAMTE, LANDRY STEPHANE; Lavecchia, A.; Klotz, K. N; Cappellacci, Loredana
Synthesis and pharmacological evaluation of 4-phenoxy-1,2,3,4-tetrahydroisoquinolines and 4,5,6,6a-tetrahydrochromeno [2,3,4-de]isoquinolines
2008-01-01 Giorgioni, Gianfabio; Ruggieri, Sabrina; Claudi, Francesco; DI STEFANO, A.; Ljung, E.; Carlsson, T.
“Synthesis and Pharmacological Evaluation of Enantiomerically Pure 4-Deoxy-4-Fluoro-Muscarines”.
1992-01-01 Bravo, P; Resnati, G; Angeli, Piero; Frigerio, M; Viani, F; Arnone, A; Marucci, Gabriella; Cantalamessa, Franco
Synthesis and pharmacological profile of a series of 1-substituted-2-carbonyl derivatives of diphenidol: novel M4 muscarinic receptor antagonists
2008-01-01 Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Fazio, N; Marucci, Gabriella; Recanatini, M; Spampanato, S.
Synthesis and pharmacological testing of polyaminoquinolines as blockers of the apamin-sensitive Ca2+-activated K+ channel (SKCa)
2007-01-01 Fletcher, D. I.; Ganellin, C. R.; Piergentili, Alessandro; Dunn, P. M.; Jenkinson, D. H.
Synthesis and physico-chemical properties of a novel series of aromatic electron acceptors based on N-heterocycles
2012-01-01 Bianca, Furdui; Rodica M., Dinica; Tabacaru, Aurel; Pettinari, Claudio
Synthesis and potency of novel uracil nucleotides and derivatives as P2Y(2) and P2Y(6) receptor agonists
2008-01-01 Ko, H.; Carter, R. L.; Cosyn, L.; Petrelli, Riccardo; DE CASTRO, S.; Besada, P.; Zhou, Y.; Cappellacci, Loredana; Franchetti, P.; Grifantini, M.; VAN CALENBERGH, S.; Harden, T. K.; Jacobson, K. A.
Synthesis and practical applications of 2-(2-nitroalkyl) pyrroles
2020-01-01 Palmieri, Alessandro; Petrini, Marino
Synthesis and Preliminary Evaluation of L-Dopa/Benserazide Conjugates as dual Acting Codrugs
2006-01-01 A., Di Stefano; P., Sozio; A., Iannitelli; A., Cocco; G., Orlando; Ricciutelli, Massimo
Synthesis and Preliminary Pharmacological Evaluation of 5-Hydroxy- and 5,6-Dihydroxy-1,2,3,7,12,12a-hexahydrobenzo [5,6]cyclohepta[1,2,3-ij]isoquinoline Derivatives as Dopamine Receptor Ligands
2001-01-01 Cingolani, Gian Mario; DI STEFANO, A.; Napolitani, F.; Mosciatti, B.; Giorgioni, Gianfabio; Cinone, N.; Brunetti, L.; Luisi, G.; Michelotto, B.; Orlando, G.; Costa, B.; Lucacchini, A.; Martini, C.; Claudi, Francesco
Synthesis and properties of poly(pyrazolyl)borate and related boron-centered scorpionate ligands. Part A: pyrazole-based systems
2010-01-01 Santini, Carlo; Pellei, Maura; GIOIA LOBBIA, Giancarlo; Papini, Grazia
Synthesis and properties of poly(pyrazolyl)borate and related boron-centered scorpionate ligands. Part B: imidazole-, triazole- and other heterocycle-based systems
2010-01-01 Pellei, Maura; GIOIA LOBBIA, Giancarlo; Papini, Grazia; Santini, Carlo
Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers
2023-01-01 Verboni, M.; Perinelli, D. R.; Qiu, C. Y.; Tiboni, M.; Aluigi, A.; Lucarini, S.; Lam, J. K. W.; Duranti, A.
Synthesis and radical cyclization of 2-allylamino-3-chloropropylphenyl sulfones to 2,4-disubstituted pyrrolidines
1998-01-01 Giovannini, R.; Petrini, Marino
Synthesis and receptor affinity of polysubstituted adenosines
1999-01-01 Vittori, Sauro; Camaioni, E; Costanzi, S; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria
Synthesis and SAR of group 11 N-heterocyclic carbene complexes
2013-01-01 Pellei, Maura; Marinelli, Marika; GIOIA LOBBIA, Giancarlo; Cimarelli, Cristina; Giorgioni, Gianfabio; C., Marzano; V., Gandin; A., Dolmella; Santini, Carlo
Synthesis and SAR of symmetrical and non-symmetrical 11th group-NHC complexes
2013-01-01 Marinelli, Marika; Pellei, Maura; GIOIA LOBBIA, Giancarlo; Trasatti, Andrea; Santini, Carlo
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Synthesis and pharmacological characterization of chiral pyrrolidinylfuran derivatives: The discovery of new functionally selective muscarinic agonists | 1-gen-2008 | Scapecchi, S.; Nesi, M.; Matucci, R.; Bellucci, C.; Buccioni, Michela; Dei, S.; Guandalini, L.; Manetti, D.; Martini, E.; Marucci, Gabriella; Romanelli, M. N.; Teodori, E.; Cirilli, R. | Articolo | |
Synthesis and pharmacological characterization of enantiomerically pure muscarinic agonists: difluoromuscarines | 1-gen-1997 | Angeli, Piero; Cantalamessa, Franco; Cavagna, Roberto; Conti, Paola; De Amici, Marco; De Micheli, Marco; Gamba, Anna; Marucci, Gabriella | Articolo | |
Synthesis and pharmacological characterization of new chiral derivatives of muscarine and allo-muscarine | 1-gen-2000 | DE AMICI, M.; Dallanoce, C.; Angeli, Piero; Marucci, Gabriella; Cantalamessa, Franco; DE MICHELIS, C. | Articolo | |
SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF RIBOSE-MODIFIED ADENOSINE DERIVATIVES AS P1 RECEPTOR LIGANDS | 1-gen-2016 | Scortichini, Mirko; Petrelli, Riccardo; Kachler, S.; Luongo, L.; Maione, S.; NGAHANG KAMTE, LANDRY STEPHANE; Lavecchia, A.; Klotz, K. N; Cappellacci, Loredana | Contributo in atto di convegno su volume | |
Synthesis and pharmacological evaluation of 4-phenoxy-1,2,3,4-tetrahydroisoquinolines and 4,5,6,6a-tetrahydrochromeno [2,3,4-de]isoquinolines | 1-gen-2008 | Giorgioni, Gianfabio; Ruggieri, Sabrina; Claudi, Francesco; DI STEFANO, A.; Ljung, E.; Carlsson, T. | Articolo | |
“Synthesis and Pharmacological Evaluation of Enantiomerically Pure 4-Deoxy-4-Fluoro-Muscarines”. | 1-gen-1992 | Bravo, P; Resnati, G; Angeli, Piero; Frigerio, M; Viani, F; Arnone, A; Marucci, Gabriella; Cantalamessa, Franco | Articolo | |
Synthesis and pharmacological profile of a series of 1-substituted-2-carbonyl derivatives of diphenidol: novel M4 muscarinic receptor antagonists | 1-gen-2008 | Varoli, L; Angeli, Piero; Buccioni, Michela; Burnelli, S; Fazio, N; Marucci, Gabriella; Recanatini, M; Spampanato, S. | Articolo | |
Synthesis and pharmacological testing of polyaminoquinolines as blockers of the apamin-sensitive Ca2+-activated K+ channel (SKCa) | 1-gen-2007 | Fletcher, D. I.; Ganellin, C. R.; Piergentili, Alessandro; Dunn, P. M.; Jenkinson, D. H. | Articolo | |
Synthesis and physico-chemical properties of a novel series of aromatic electron acceptors based on N-heterocycles | 1-gen-2012 | Bianca, Furdui; Rodica M., Dinica; Tabacaru, Aurel; Pettinari, Claudio | Articolo | |
Synthesis and potency of novel uracil nucleotides and derivatives as P2Y(2) and P2Y(6) receptor agonists | 1-gen-2008 | Ko, H.; Carter, R. L.; Cosyn, L.; Petrelli, Riccardo; DE CASTRO, S.; Besada, P.; Zhou, Y.; Cappellacci, Loredana; Franchetti, P.; Grifantini, M.; VAN CALENBERGH, S.; Harden, T. K.; Jacobson, K. A. | Articolo | |
Synthesis and practical applications of 2-(2-nitroalkyl) pyrroles | 1-gen-2020 | Palmieri, Alessandro; Petrini, Marino | Articolo | |
Synthesis and Preliminary Evaluation of L-Dopa/Benserazide Conjugates as dual Acting Codrugs | 1-gen-2006 | A., Di Stefano; P., Sozio; A., Iannitelli; A., Cocco; G., Orlando; Ricciutelli, Massimo | Articolo | |
Synthesis and Preliminary Pharmacological Evaluation of 5-Hydroxy- and 5,6-Dihydroxy-1,2,3,7,12,12a-hexahydrobenzo [5,6]cyclohepta[1,2,3-ij]isoquinoline Derivatives as Dopamine Receptor Ligands | 1-gen-2001 | Cingolani, Gian Mario; DI STEFANO, A.; Napolitani, F.; Mosciatti, B.; Giorgioni, Gianfabio; Cinone, N.; Brunetti, L.; Luisi, G.; Michelotto, B.; Orlando, G.; Costa, B.; Lucacchini, A.; Martini, C.; Claudi, Francesco | Articolo | |
Synthesis and properties of poly(pyrazolyl)borate and related boron-centered scorpionate ligands. Part A: pyrazole-based systems | 1-gen-2010 | Santini, Carlo; Pellei, Maura; GIOIA LOBBIA, Giancarlo; Papini, Grazia | Articolo | |
Synthesis and properties of poly(pyrazolyl)borate and related boron-centered scorpionate ligands. Part B: imidazole-, triazole- and other heterocycle-based systems | 1-gen-2010 | Pellei, Maura; GIOIA LOBBIA, Giancarlo; Papini, Grazia; Santini, Carlo | Articolo | |
Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers | 1-gen-2023 | Verboni, M.; Perinelli, D. R.; Qiu, C. Y.; Tiboni, M.; Aluigi, A.; Lucarini, S.; Lam, J. K. W.; Duranti, A. | Articolo | |
Synthesis and radical cyclization of 2-allylamino-3-chloropropylphenyl sulfones to 2,4-disubstituted pyrrolidines | 1-gen-1998 | Giovannini, R.; Petrini, Marino | Articolo | |
Synthesis and receptor affinity of polysubstituted adenosines | 1-gen-1999 | Vittori, Sauro; Camaioni, E; Costanzi, S; Volpini, Rosaria; Klotz, K. N.; Cristalli, Gloria | Articolo | |
Synthesis and SAR of group 11 N-heterocyclic carbene complexes | 1-gen-2013 | Pellei, Maura; Marinelli, Marika; GIOIA LOBBIA, Giancarlo; Cimarelli, Cristina; Giorgioni, Gianfabio; C., Marzano; V., Gandin; A., Dolmella; Santini, Carlo | Contributo in atto di convegno su volume | |
Synthesis and SAR of symmetrical and non-symmetrical 11th group-NHC complexes | 1-gen-2013 | Marinelli, Marika; Pellei, Maura; GIOIA LOBBIA, Giancarlo; Trasatti, Andrea; Santini, Carlo | Poster atto convegno su volume |
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