Sfoglia per Autore
A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus
2016-01-01 Mammoli, Valerio; Bonifazi, Alessandro; DAL BEN, Diego; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Thomas, Ajiroghene; Newman, Amy H; Ferré, Sergi; Sanchez Soto, Marta; Keck, Thomas M; DEL BELLO, Fabio
Synergic stimulation of serotonin 5-HT1A receptor and α2-adrenoceptors for neuropathic pain relief: Preclinical effects of 2-substituted imidazoline derivatives
2017-01-01 Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Micheli, Laura; DEL BELLO, Fabio; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Novel muscarinic acetylcholine receptor hybrid ligands embedding quinuclidine and 1,4-dioxane fragments
2017-01-01 DEL BELLO, Fabio; Bonifazi, Alessandro; Giorgioni, Gianfabio; Petrelli, Riccardo; Quaglia, Wilma; Altomare, Angela; Falcicchio, Aurelia; Matucci, Rosanna; Vistoli, Giulio; Piergentili, Alessandro
77-LH-28-1 as a model for the rational design of selective dopamine D4 receptor ligands
2017-01-01 DEL BELLO, Fabio; Bonifazi, Alessandro; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Quaglia, Wilma; Matucci, Rosanna
Exploring the Role of N6‐Substituents in Potent Dual Acting 5'‐C‐Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice
2017-01-01 Petrelli, Riccardo; Scortichini, Mirko; Kachler, Sonja; Boccella, Serena; Cerchia, Carmen; Torquati, Ilaria; DEL BELLO, Fabio; Salvemini, Daniela; Novellino, Ettore; Luongo, Livio; Maione, Sabatino; A Jacobson, Kenneth; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
The replacement of the 2-methoxy substituent of N-((6,6-diphenyl-1,4-dioxan-2-yl)methyl)-2-(2-methoxyphenoxy)ethan-1-amine improves the selectivity for 5-HT1A receptor over α1-adrenoceptor and D2-like receptor subtypes
2017-01-01 DEL BELLO, Fabio; Bonifazi, Alessandro; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Petrelli, Riccardo; Cifani, Carlo; MICIONI DI BONAVENTURA, Maria Vittoria; Keck, Thomas M; Mazzolari, Angelica; Vistoli, Giulio; Cilia, Antonio; Poggesi, Elena; Matucci, Rosanna; Quaglia, Wilma
4WD to Travel Inside the 5-HT1A Receptor World
2017-01-01 Quaglia, Wilma; Cifani, Carlo; Del Bello, Fabio; Giannella, Mario; Giorgioni, Gianfabio; Bonaventura, Maria Vittoria Micioni Di; Piergentili, Alessandro
An Efficient Lewis Acid Catalyzed Povarov Reaction for the One-Pot Stereocontrolled Synthesis of Polyfunctionalized Tetrahydroquinolines
2017-01-01 Cimarelli, Cristina; Bordi, Samuele; Piermattei, Pamela; Pellei, Maura; DEL BELLO, Fabio; Marcantoni, Enrico
Design, synthesis, reactivity, biological and catalytic applications of functionalized bis(pyrazolyl)acetate copper complexes
2018-01-01 Bagnarelli, L.; Luciani, Lorenzo; Romagnoli, M.; Del Bello, F.; Quaglia, W.; Cimarelli, C.; Gabrielli, S.; Santini, C.; Pellei, M.
Rational design and biological evaluation of novel conjugated heteroscorpionate ligands and related Copper(I/II) complexes
2018-01-01 Santini, Carlo; Pellei, Maura; Bagnarelli, Luca; Cimarelli, Cristina; DEL BELLO, Fabio; Quaglia, Wilma; Morelli, Maria Beatrice; Amantini, Consuelo; Valentina, Gandin; Cristina, Marzano
Efficient Lewis Acid Systems for the A3 Coupling reaction
2018-01-01 Cimarelli, C.; Navazio, F.; Rossi, F. V.; Del Bello, F.; Marcantoni, E.
New insights in Au-NHCs complexes as anticancer agents
2018-01-01 Porchia, Marina; Pellei, Maura; Marinelli, Marika; Tisato, Francesco; Del Bello, Fabio; Santini, Carlo
The first water-soluble copper(I) complexes bearing sulfonated imidazole- and benzimidazole-derived N-heterocyclic carbenes: Synthesis and anticancer studies
2018-01-01 Pellei, Maura; Gandin, Valentina; Marzano, Cristina; Marinelli, Marika; Del Bello, Fabio; Santini, Carlo
Structure-Based Design, Synthesis and in vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists
2018-01-01 Petrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; DEL BELLO, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana
Front Cover, European Journal of Medicinal, Issue 146, 25 February 2018.
2018-01-01 Porchia, Marina; Pellei, Maura; Marinelli, Marika; Tisato, Francesco; DEL BELLO, Fabio; Santini, Carlo
Novel antitumor copper(ii) complexes designed to act through synergistic mechanisms of action, due to the presence of an NMDA receptor ligand and copper in the same chemical entity
2018-01-01 Morelli, Maria Beatrice; Amantini, Consuelo; Santoni, Giorgio; Pellei, Maura; Santini, Carlo; Cimarelli, Cristina; Marcantoni, Enrico; Petrini, Marino; Del Bello, Fabio; Giorgioni, Gianfabio; Piergentili, Alessandro; Quaglia, Wilma
1-[3-(4-Butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1) as a Model for the Rational Design of a Novel Class of Brain Penetrant Ligands with High Affinity and Selectivity for Dopamine D4 Receptor
2018-01-01 Del Bello, Fabio; Bonifazi, Alessandro; Giorgioni, Gianfabio; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Petrelli, Riccardo; Piergentili, Alessandro; Fontana, Stefano; Mammoli, Valerio; Yano, Hideaki; Matucci, Rosanna; Vistoli, Giulio; Quaglia, Wilma
Syntheses, biological and catalytic studies of copper complexes bearing bis(azol-1-yl)-acetato heteroscorpionate ligands
2019-01-01 Bagnarelli, Luca; Santini, Carlo; Gabrielli, Serena; Gandin, Valentina; Marzano, Cristina; DEL BELLO, Fabio; Pellei, Maura
Synthesis, reactivity and biological studies of bioconjugated bis(pyrazolyl)acetate copper complexes
2019-01-01 Santini, C.; Bagnarelli, L.; Luciani, L.; Scorcelletti, F.; Del Bello, F.; Quaglia, W.; Marzano, C.; Gandin, V.; Pellei, M.
Role of the NMDA Receptor in the Antitumor Activity of Chiral 1,4-Dioxane Ligands in MCF-7 and SKBR3 Breast Cancer Cells
2019-01-01 Morelli, Maria Beatrice; Amantini, Consuelo; Nabissi, Massimo; Santoni, Giorgio; Wünsch, Bernhard; Schepmann, Dirk; Cimarelli, Cristina; Pellei, Maura; Santini, Carlo; Fontana, Stefano; Mammoli, Valerio; Quaglia, Wilma; Bonifazi, Alessandro; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Del Bello, Fabio
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus | 1-gen-2016 | Mammoli, Valerio; Bonifazi, Alessandro; DAL BEN, Diego; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma; Thomas, Ajiroghene; Newman, Amy H; Ferré, Sergi; Sanchez Soto, Marta; Keck, Thomas M; DEL BELLO, Fabio | Articolo | |
Synergic stimulation of serotonin 5-HT1A receptor and α2-adrenoceptors for neuropathic pain relief: Preclinical effects of 2-substituted imidazoline derivatives | 1-gen-2017 | Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Micheli, Laura; DEL BELLO, Fabio; Giannella, Mario; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | Articolo | |
Novel muscarinic acetylcholine receptor hybrid ligands embedding quinuclidine and 1,4-dioxane fragments | 1-gen-2017 | DEL BELLO, Fabio; Bonifazi, Alessandro; Giorgioni, Gianfabio; Petrelli, Riccardo; Quaglia, Wilma; Altomare, Angela; Falcicchio, Aurelia; Matucci, Rosanna; Vistoli, Giulio; Piergentili, Alessandro | Articolo | |
77-LH-28-1 as a model for the rational design of selective dopamine D4 receptor ligands | 1-gen-2017 | DEL BELLO, Fabio; Bonifazi, Alessandro; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Quaglia, Wilma; Matucci, Rosanna | Poster atto convegno su volume | |
Exploring the Role of N6‐Substituents in Potent Dual Acting 5'‐C‐Ethyltetrazolyladenosine Derivatives: Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice | 1-gen-2017 | Petrelli, Riccardo; Scortichini, Mirko; Kachler, Sonja; Boccella, Serena; Cerchia, Carmen; Torquati, Ilaria; DEL BELLO, Fabio; Salvemini, Daniela; Novellino, Ettore; Luongo, Livio; Maione, Sabatino; A Jacobson, Kenneth; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana | Articolo | |
The replacement of the 2-methoxy substituent of N-((6,6-diphenyl-1,4-dioxan-2-yl)methyl)-2-(2-methoxyphenoxy)ethan-1-amine improves the selectivity for 5-HT1A receptor over α1-adrenoceptor and D2-like receptor subtypes | 1-gen-2017 | DEL BELLO, Fabio; Bonifazi, Alessandro; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Petrelli, Riccardo; Cifani, Carlo; MICIONI DI BONAVENTURA, Maria Vittoria; Keck, Thomas M; Mazzolari, Angelica; Vistoli, Giulio; Cilia, Antonio; Poggesi, Elena; Matucci, Rosanna; Quaglia, Wilma | Articolo | |
4WD to Travel Inside the 5-HT1A Receptor World | 1-gen-2017 | Quaglia, Wilma; Cifani, Carlo; Del Bello, Fabio; Giannella, Mario; Giorgioni, Gianfabio; Bonaventura, Maria Vittoria Micioni Di; Piergentili, Alessandro | Capitolo di libro o voce di enciclopedia | |
An Efficient Lewis Acid Catalyzed Povarov Reaction for the One-Pot Stereocontrolled Synthesis of Polyfunctionalized Tetrahydroquinolines | 1-gen-2017 | Cimarelli, Cristina; Bordi, Samuele; Piermattei, Pamela; Pellei, Maura; DEL BELLO, Fabio; Marcantoni, Enrico | Articolo | |
Design, synthesis, reactivity, biological and catalytic applications of functionalized bis(pyrazolyl)acetate copper complexes | 1-gen-2018 | Bagnarelli, L.; Luciani, Lorenzo; Romagnoli, M.; Del Bello, F.; Quaglia, W.; Cimarelli, C.; Gabrielli, S.; Santini, C.; Pellei, M. | Contributo in atto di convegno su volume | |
Rational design and biological evaluation of novel conjugated heteroscorpionate ligands and related Copper(I/II) complexes | 1-gen-2018 | Santini, Carlo; Pellei, Maura; Bagnarelli, Luca; Cimarelli, Cristina; DEL BELLO, Fabio; Quaglia, Wilma; Morelli, Maria Beatrice; Amantini, Consuelo; Valentina, Gandin; Cristina, Marzano | Contributo in atto di convegno su volume | |
Efficient Lewis Acid Systems for the A3 Coupling reaction | 1-gen-2018 | Cimarelli, C.; Navazio, F.; Rossi, F. V.; Del Bello, F.; Marcantoni, E. | Poster atto convegno su volume | |
New insights in Au-NHCs complexes as anticancer agents | 1-gen-2018 | Porchia, Marina; Pellei, Maura; Marinelli, Marika; Tisato, Francesco; Del Bello, Fabio; Santini, Carlo | Articolo | |
The first water-soluble copper(I) complexes bearing sulfonated imidazole- and benzimidazole-derived N-heterocyclic carbenes: Synthesis and anticancer studies | 1-gen-2018 | Pellei, Maura; Gandin, Valentina; Marzano, Cristina; Marinelli, Marika; Del Bello, Fabio; Santini, Carlo | Articolo | |
Structure-Based Design, Synthesis and in vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists | 1-gen-2018 | Petrelli, Riccardo; Scortichini, Mirko; Belardo, Carmela; Boccella, Serena; Luongo, Livio; Capone, Fabio; Kachler, Sonja; Vita, Patrizia; DEL BELLO, Fabio; Maione, Sabatino; Lavecchia, Antonio; Klotz, Karl-Norbert; Cappellacci, Loredana | Articolo | |
Front Cover, European Journal of Medicinal, Issue 146, 25 February 2018. | 1-gen-2018 | Porchia, Marina; Pellei, Maura; Marinelli, Marika; Tisato, Francesco; DEL BELLO, Fabio; Santini, Carlo | Altre tipologie di pubblicazione (Recensione) | |
Novel antitumor copper(ii) complexes designed to act through synergistic mechanisms of action, due to the presence of an NMDA receptor ligand and copper in the same chemical entity | 1-gen-2018 | Morelli, Maria Beatrice; Amantini, Consuelo; Santoni, Giorgio; Pellei, Maura; Santini, Carlo; Cimarelli, Cristina; Marcantoni, Enrico; Petrini, Marino; Del Bello, Fabio; Giorgioni, Gianfabio; Piergentili, Alessandro; Quaglia, Wilma | Articolo | |
1-[3-(4-Butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1) as a Model for the Rational Design of a Novel Class of Brain Penetrant Ligands with High Affinity and Selectivity for Dopamine D4 Receptor | 1-gen-2018 | Del Bello, Fabio; Bonifazi, Alessandro; Giorgioni, Gianfabio; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Petrelli, Riccardo; Piergentili, Alessandro; Fontana, Stefano; Mammoli, Valerio; Yano, Hideaki; Matucci, Rosanna; Vistoli, Giulio; Quaglia, Wilma | Articolo | |
Syntheses, biological and catalytic studies of copper complexes bearing bis(azol-1-yl)-acetato heteroscorpionate ligands | 1-gen-2019 | Bagnarelli, Luca; Santini, Carlo; Gabrielli, Serena; Gandin, Valentina; Marzano, Cristina; DEL BELLO, Fabio; Pellei, Maura | Contributo in atto di convegno su volume | |
Synthesis, reactivity and biological studies of bioconjugated bis(pyrazolyl)acetate copper complexes | 1-gen-2019 | Santini, C.; Bagnarelli, L.; Luciani, L.; Scorcelletti, F.; Del Bello, F.; Quaglia, W.; Marzano, C.; Gandin, V.; Pellei, M. | Contributo in atto di convegno su volume | |
Role of the NMDA Receptor in the Antitumor Activity of Chiral 1,4-Dioxane Ligands in MCF-7 and SKBR3 Breast Cancer Cells | 1-gen-2019 | Morelli, Maria Beatrice; Amantini, Consuelo; Nabissi, Massimo; Santoni, Giorgio; Wünsch, Bernhard; Schepmann, Dirk; Cimarelli, Cristina; Pellei, Maura; Santini, Carlo; Fontana, Stefano; Mammoli, Valerio; Quaglia, Wilma; Bonifazi, Alessandro; Giannella, Mario; Giorgioni, Gianfabio; Piergentili, Alessandro; Del Bello, Fabio | Articolo |
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