Sfoglia per Autore
Effects of the selective adenosine A1 receptor agonist 5 '-chloro-5 '-deoxy-N6-(2-endo-norbornyl) adenosine on nociception in mice
2008-01-01 Marabese, I.; Cappellacci, Loredana; Franchetti, Palmarisa; DE NOVELLIS, V.; Klotz, K. N.; Grifantini, Mario; Maione, S.
Ribose-modified purine nucleosides as ribonucleotide reductase inhibitors. Synthesis, antitumor activity, and molecular modeling of N-6-substituted 3'-C-methyladenosine derivatives
2008-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Vita, P.; Petrelli, Riccardo; Lavecchia, A.; Jayaram, H. N.; Saiko, P.; Graser, G.; Szekeres, T.; Grifantini, Mario
5’-Carbamoyl Derivatives of 2'-C-Methyl-purine Nucleosides as Selective A1 Adenosine Receptor Agonists: Affinity, Efficacy and Selectivity for A1 Receptor from Different Species.
2008-01-01 Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Vita, P; Lavecchia, A; Costa, B; Spinetti, F; Martini, C; Klotz, K. N.; Grifantini, Mario
New N6-substituted adenosine and 3’-C-methyl-adenosine derivatives as antitumor agents
2009-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Kusumanchi, P; Kumar, M; Jayaram, Hn; Grifantini, Mario
Selective inhibition of nicotinamide adenine kinases (NADKs) by compact NAD mimics
2009-01-01 Petrelli, Riccardo; Felczak, K; Chen, L; Vita, Patrizia; Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Di Stefano, M; Magni, G; Pankiewicz, K.
HISTONE DEACETYLASE (HDAC) INHIBITION MODULATES INTRACELLULAR DEOXYNUCLEOTIDES (DNTP) POOLS AND POTENTIATES THE ANTITUMOR EFFECTS OF THE RIBONUCLEOTIDE REDUCTASE (RR) INHIBITOR 3’- METHYL-ADENOSINE (3’-ME-ADO) IN PROMYELOCITIC LEUKAEMIA CELL LINES.
2009-01-01 Meli, M; Tolomeo, M; Grifantini, Mario; Mai, A; Cappellacci, Loredana; Franchetti, Palmarisa; Saiko, P; Dusonchet, L.
Effects of 5'-chloro-5'-deoxy-N6-(±)-endo-norbornyl-adenosine, a potent and highly selective A1 adenosine receptor agonist, on neuropathic pain-induced behavioural and morphological changes in spinal microglia
2010-01-01 Luongo, L; Cappellacci, Loredana; Giordano, C; Petrelli, Riccardo; Guida, F; Franchetti, Palmarisa; Grifantini, Mario; Maione, S.
Dual-target dimeric molecules with antitumor properties. Synthesis and biological activity of 3’-C-methyladenosine-valproates
2010-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Jayaram, Hn; Grifantini, Mario
EFFECTS OF METAL(III) COORDINATION ON BIOLOGICAL ACTIVITY OF 2,2'-BIPYRIDYL-6-CARBOTHIOAMIDE (BPYTA), A POTENT R2 RIBONUCLEOTIDE REDUCTASE INHIBITOR
2010-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Heffeter P., Kowol CR; Franchetti, Palmarisa
Synthesis and biological activity of novel N6-substituted and 2,N6-disubstituted adenine ribo- and 3'-C-methyl-ribonucleosides as antitumor agents
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Franchetti, Palmarisa; Vita, Patrizia; Kusumanchi, P; Kumar, M; Jayaram, H. N.; Zhou, B; Yen, Y; Grifantini, Mario
Antitumor effects of novel co-drugs linking histone deacetylase and ribonucleotide reductase inhibitors in hematological tumors
2011-01-01 A., Ferro; Cappellacci, Loredana; A., Mingrino; Petrelli, Riccardo; M., Tolomeo; Vita, Patrizia; N., D’Alessandro; L., Dusonchet; Franchetti, Palmarisa; Grifantini, Mario; M., Meli
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands
2011-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario
Novel hydrazone derivatives having potent antitumor activity toward multi-drug resistant tumor cells
2012-01-01 Jayaram, Hn; Kusumanchi, P; Grifantini, Mario; Franchetti, Palmarisa; Cappellacci, Loredana; Petrelli, Riccardo
ADP- and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 receptor ligands
2012-01-01 Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Jacobson, Ka; Barrett, Mo; Franklin, D; Harden, Kt; Franchetti, Palmarisa; Grifantini, Mario
Novel Inhibitors of Inosine Monophosphate Dehydrogenase in Patent Literature of the Last Decade
2013-01-01 Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krysztof, Felczak; Daniel J., Wilson; Franchetti, Palmarisa; Cappellacci, Loredana
5’-CHLORO-5’-DEOXY-N6-SUBSTITUTED ADENOSINE DERIVATIVES: SYNTHESIS, ADENOSINE RECEPTOR AFFINITY AND ANTINOCICEPTIVE ACTIVITY
2013-01-01 Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Luongo; K. N., Klotz; S., Kachler; F., Guida; M., De Chiaro; S., Maione; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana
SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF NOVEL HYDRAZONE DERIVATIVES
2014-01-01 Petrelli, Riccardo; Torquati, Ilaria; Anders, Hofer; Olivia, Grubbström; Venkateswara Rao, Jonn; Praveen, Kusumanchi; Hiremagalur N., Jayaram; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana
Titolo | Data di pubblicazione | Autore(i) | Tipo | File |
---|---|---|---|---|
Effects of the selective adenosine A1 receptor agonist 5 '-chloro-5 '-deoxy-N6-(2-endo-norbornyl) adenosine on nociception in mice | 1-gen-2008 | Marabese, I.; Cappellacci, Loredana; Franchetti, Palmarisa; DE NOVELLIS, V.; Klotz, K. N.; Grifantini, Mario; Maione, S. | Poster atto convegno su rivista | |
Ribose-modified purine nucleosides as ribonucleotide reductase inhibitors. Synthesis, antitumor activity, and molecular modeling of N-6-substituted 3'-C-methyladenosine derivatives | 1-gen-2008 | Cappellacci, Loredana; Franchetti, Palmarisa; Vita, P.; Petrelli, Riccardo; Lavecchia, A.; Jayaram, H. N.; Saiko, P.; Graser, G.; Szekeres, T.; Grifantini, Mario | Articolo | |
5’-Carbamoyl Derivatives of 2'-C-Methyl-purine Nucleosides as Selective A1 Adenosine Receptor Agonists: Affinity, Efficacy and Selectivity for A1 Receptor from Different Species. | 1-gen-2008 | Cappellacci, Loredana; Franchetti, Palmarisa; Petrelli, Riccardo; Vita, P; Lavecchia, A; Costa, B; Spinetti, F; Martini, C; Klotz, K. N.; Grifantini, Mario | Articolo | |
New N6-substituted adenosine and 3’-C-methyl-adenosine derivatives as antitumor agents | 1-gen-2009 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Kusumanchi, P; Kumar, M; Jayaram, Hn; Grifantini, Mario | Contributo in atto di convegno su volume | |
Selective inhibition of nicotinamide adenine kinases (NADKs) by compact NAD mimics | 1-gen-2009 | Petrelli, Riccardo; Felczak, K; Chen, L; Vita, Patrizia; Cappellacci, Loredana; Franchetti, Palmarisa; Grifantini, Mario; Di Stefano, M; Magni, G; Pankiewicz, K. | Contributo in atto di convegno su volume | |
HISTONE DEACETYLASE (HDAC) INHIBITION MODULATES INTRACELLULAR DEOXYNUCLEOTIDES (DNTP) POOLS AND POTENTIATES THE ANTITUMOR EFFECTS OF THE RIBONUCLEOTIDE REDUCTASE (RR) INHIBITOR 3’- METHYL-ADENOSINE (3’-ME-ADO) IN PROMYELOCITIC LEUKAEMIA CELL LINES. | 1-gen-2009 | Meli, M; Tolomeo, M; Grifantini, Mario; Mai, A; Cappellacci, Loredana; Franchetti, Palmarisa; Saiko, P; Dusonchet, L. | Poster atto convegno su volume | |
Effects of 5'-chloro-5'-deoxy-N6-(±)-endo-norbornyl-adenosine, a potent and highly selective A1 adenosine receptor agonist, on neuropathic pain-induced behavioural and morphological changes in spinal microglia | 1-gen-2010 | Luongo, L; Cappellacci, Loredana; Giordano, C; Petrelli, Riccardo; Guida, F; Franchetti, Palmarisa; Grifantini, Mario; Maione, S. | Poster atto convegno su volume | |
Dual-target dimeric molecules with antitumor properties. Synthesis and biological activity of 3’-C-methyladenosine-valproates | 1-gen-2010 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Franchetti, Palmarisa; Jayaram, Hn; Grifantini, Mario | Poster atto convegno su volume | |
EFFECTS OF METAL(III) COORDINATION ON BIOLOGICAL ACTIVITY OF 2,2'-BIPYRIDYL-6-CARBOTHIOAMIDE (BPYTA), A POTENT R2 RIBONUCLEOTIDE REDUCTASE INHIBITOR | 1-gen-2010 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Grifantini, Mario; Heffeter P., Kowol CR; Franchetti, Palmarisa | Poster atto convegno su volume | |
Synthesis and biological activity of novel N6-substituted and 2,N6-disubstituted adenine ribo- and 3'-C-methyl-ribonucleosides as antitumor agents | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Franchetti, Palmarisa; Vita, Patrizia; Kusumanchi, P; Kumar, M; Jayaram, H. N.; Zhou, B; Yen, Y; Grifantini, Mario | Articolo | |
Antitumor effects of novel co-drugs linking histone deacetylase and ribonucleotide reductase inhibitors in hematological tumors | 1-gen-2011 | A., Ferro; Cappellacci, Loredana; A., Mingrino; Petrelli, Riccardo; M., Tolomeo; Vita, Patrizia; N., D’Alessandro; L., Dusonchet; Franchetti, Palmarisa; Grifantini, Mario; M., Meli | Poster atto convegno su volume | |
ADP-, and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 ligands | 1-gen-2011 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Kenneth A., Jacobson; Matthew, Barrett; T., Kendall Harden; Franchetti, Palmarisa; Grifantini, Mario | Poster atto convegno su volume | |
Novel hydrazone derivatives having potent antitumor activity toward multi-drug resistant tumor cells | 1-gen-2012 | Jayaram, Hn; Kusumanchi, P; Grifantini, Mario; Franchetti, Palmarisa; Cappellacci, Loredana; Petrelli, Riccardo | 07 BREVETTO | |
ADP- and ATP-mimetics derived from 2'(3')-C-methyladenosine as human P2Y1 and P2Y2 receptor ligands | 1-gen-2012 | Cappellacci, Loredana; Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Jacobson, Ka; Barrett, Mo; Franklin, D; Harden, Kt; Franchetti, Palmarisa; Grifantini, Mario | Contributo in atto di convegno su rivista | |
Novel Inhibitors of Inosine Monophosphate Dehydrogenase in Patent Literature of the Last Decade | 1-gen-2013 | Petrelli, Riccardo; Vita, Patrizia; Torquati, Ilaria; Krysztof, Felczak; Daniel J., Wilson; Franchetti, Palmarisa; Cappellacci, Loredana | Articolo | |
5’-CHLORO-5’-DEOXY-N6-SUBSTITUTED ADENOSINE DERIVATIVES: SYNTHESIS, ADENOSINE RECEPTOR AFFINITY AND ANTINOCICEPTIVE ACTIVITY | 1-gen-2013 | Petrelli, Riccardo; Torquati, Ilaria; Vita, Patrizia; L., Luongo; K. N., Klotz; S., Kachler; F., Guida; M., De Chiaro; S., Maione; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana | Poster atto convegno su volume | |
SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF NOVEL HYDRAZONE DERIVATIVES | 1-gen-2014 | Petrelli, Riccardo; Torquati, Ilaria; Anders, Hofer; Olivia, Grubbström; Venkateswara Rao, Jonn; Praveen, Kusumanchi; Hiremagalur N., Jayaram; Franchetti, Palmarisa; Grifantini, Mario; Cappellacci, Loredana | Poster atto convegno su volume |
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